Target
Aminoacyl tRNA synthase complex-interacting multifunctional protein 2
Ligand
BDBM50514847
Substrate
n/a
Meas. Tech.
ChEMBL_1858838 (CHEMBL4359567)
Kd
3070±n/a nM
Citation
 Sivaraman, AKim, DGBhattarai, DKim, MLee, HYLim, SKong, JGoo, JIShim, SLee, SSuh, YGChoi, YKim, SLee, K Synthesis and Structure-Activity Relationships of Arylsulfonamides as AIMP2-DX2 Inhibitors for the Development of a Novel Anticancer Therapy. J Med Chem 63:5139-5158 (2020) [PubMed]  Article 
Target
Name:
Aminoacyl tRNA synthase complex-interacting multifunctional protein 2
Synonyms:
Aminoacyl tRNA synthase complex-interacting multifunctional protein 2 | JTV1 | Multisynthase complex auxiliary component p38 | Protein JTV-1 | AIMP2_HUMAN | AIMP2 | JTV1
Type:
PROTEIN
Mol. Mass.:
35355.45
Organism:
Human
Description:
ChEMBL_119035
Residue:
320
Sequence:
MPMYQVKPYHGGGAPLRVELPTCMYRLPNVHGRSYGPAPGAGHVQEESNLSLQALESRQDDILKRLYELKAAVDGLSKMIQTPDADLDVTNIIQADEPTTLTTNALDLNSVLGKDYGALKDIVINANPASPPLSLLVLHRLLCEHFRVLSTVHTHSSVKSVPENLLKCFGEQNKKQPRQDYQLGFTLIWKNVPKTQMKFSIQTMCPIEGEGNIARFLFSLFGQKHNAVNATLIDSWVDIAIFQLKEGSSKEKAAVFRSMNSALGKSPWLAGNELTVADVVLWSVLQQIGGCSVTVPANVQRWMRSCENLAPFNTALKLLK
  
Inhibitor
Name:
BDBM50514847
Synonyms:
CHEMBL4558745
Type:
Small organic molecule
Emp. Form.:
TBD
Mol. Mass.:
TBD
SMILES:
TBD
Structure:
Search PDB for entries with ligand similarity: