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Target
Transcriptional enhancer factor TEF-3
Ligand
BDBM50535722
Substrate
n/a
Meas. Tech.
ChEMBL_1931084 (CHEMBL4434335)
Kd
25±n/a nM
Citation
 Furet, P; Salem, B; Mesrouze, Y; Schmelzle, T; Lewis, I; Kallen, J; Chène, P Structure-based design of potent linear peptide inhibitors of the YAP-TEAD protein-protein interaction derived from the YAP omega-loop sequence. Bioorg Med Chem Lett 29:2316-2319 (2019) [PubMed]  Article 
Target
Name:
Transcriptional enhancer factor TEF-3
Synonyms:
TEA domain family member 4 | TEAD-4 | Transcriptional enhancer factor TEF-3 | Transcription factor 13-like 1 | Transcription factor RTEF-1 | TEAD4_HUMAN | TEAD4 | RTEF1 | TCF13L1 | TEF3
Type:
PROTEIN
Mol. Mass.:
48333.01
Organism:
Human
Description:
ChEMBL_118073
Residue:
434
Sequence:
MEGTAGTITSNEWSSPTSPEGSTASGGSQALDKPIDNDAEGVWSPDIEQSFQEALAIYPPCGRRKIILSDEGKMYGRNELIARYIKLRTGKTRTRKQVSSHIQVLARRKAREIQAKLKDQAAKDKALQSMAAMSSAQIISATAFHSSMALARGPGRPAVSGFWQGALPGQAGTSHDVKPFSQQTYAVQPPLPLPGFESPAGPAPSPSAPPAPPWQGRSVASSKLWMLEFSAFLEQQQDPDTYNKHLFVHIGQSSPSYSDPYLEAVDIRQIYDKFPEKKGGLKDLFERGPSNAFFLVKFWADLNTNIEDEGSSFYGVSSQYESPENMIITCSTKVCSFGKQVVEKVETEYARYENGHYSYRIHRSPLCEYMINFIHKLKHLPEKYMMNSVLENFTILQVVTNRDTQETLLCIAYVFEVSASEHGAQHHIYRLVKE
  
Inhibitor
Name:
BDBM50535722
Synonyms:
CHEMBL4468725
Type:
Small organic molecule
Emp. Form.:
TBD
Mol. Mass.:
TBD
SMILES:
TBD
Structure:
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