Target
Chromobox protein homolog 6
Ligand
BDBM50538808
Substrate
n/a
Meas. Tech.
ChEMBL_1977188 (CHEMBL4610323)
Kd
900±n/a nM
Citation
 Milosevich, NMcFarlane, JGignac, MCLi, JBrown, TMWilson, CRDevorkin, LCroft, CSHof, RPaci, ILum, JJHof, F Pan-specific and partially selective dye-labeled peptidic inhibitors of the polycomb paralog proteins. Bioorg Med Chem 28:0 (2020) [PubMed]  Article 
Target
Name:
Chromobox protein homolog 6
Synonyms:
Chromobox protein homolog 6 | CBX6_HUMAN | CBX6
Type:
PROTEIN
Mol. Mass.:
43924.51
Organism:
Human
Description:
ChEMBL_116765
Residue:
412
Sequence:
MELSAVGERVFAAESIIKRRIRKGRIEYLVKWKGWAIKYSTWEPEENILDSRLIAAFEQKERERELYGPKKRGPKPKTFLLKARAQAEALRISDVHFSVKPSASASSPKLHSSAAVHRLKKDIRRCHRMSRRPLPRPDPQGGSPGLRPPISPFSETVRIINRKVKPREPKRNRIILNLKVIDKGAGGGGAGQGAGALARPKVPSRNRVIGKSKKFSESVLRTQIRHMKFGAFALYKPPPAPLVAPSPGKAEASAPGPGLLLAAPAAPYDARSSGSSGCPSPTPQSSDPDDTPPKLLPETVSPSAPSWREPEVLDLSLPPESAATSKRAPPEVTAAAGPAPPTAPEPAGASSEPEAGDWRPEMSPCSNVVVTDVTSNLLTVTIKEFCNPEDFEKVAAGVAGAAGGGGSIGASK
  
Inhibitor
Name:
BDBM50538808
Synonyms:
CHEMBL4646516
Type:
Small organic molecule
Emp. Form.:
TBD
Mol. Mass.:
TBD
SMILES:
TBD
Structure:
Search PDB for entries with ligand similarity: