Target
Chromobox protein homolog 7
Ligand
BDBM50538814
Substrate
n/a
Meas. Tech.
ChEMBL_1977189 (CHEMBL4610324)
Kd
1500±n/a nM
Citation
 Milosevich, NMcFarlane, JGignac, MCLi, JBrown, TMWilson, CRDevorkin, LCroft, CSHof, RPaci, ILum, JJHof, F Pan-specific and partially selective dye-labeled peptidic inhibitors of the polycomb paralog proteins. Bioorg Med Chem 28:0 (2020) [PubMed]  Article 
Target
Name:
Chromobox protein homolog 7
Synonyms:
Chromobox protein homolog 7 | CBX7_HUMAN | CBX7 | Chromobox protein homolog 7 (CBX7)
Type:
Protein
Mol. Mass.:
28351.76
Organism:
Human
Description:
n/a
Residue:
251
Sequence:
MELSAIGEQVFAVESIRKKRVRKGKVEYLVKWKGWPPKYSTWEPEEHILDPRLVMAYEEKEERDRASGYRKRGPKPKRLLLQRLYSMDLRSSHKAKGKEKLCFSLTCPLGSGSPEGVVKAGAPELVDKGPLVPTLPFPLRKPRKAHKYLRLSRKKFPPRGPNLESHSHRRELFLQEPPAPDVLQAAGEWEPAAQPPEEEADADLAEGPPPWTPALPSSEVTVTDITANSITVTFREAQAAEGFFRDRSGKF
  
Inhibitor
Name:
BDBM50538814
Synonyms:
CHEMBL4640186
Type:
Small organic molecule
Emp. Form.:
TBD
Mol. Mass.:
TBD
SMILES:
TBD
Structure:
Search PDB for entries with ligand similarity: