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Target
Delta-type opioid receptor
Ligand
BDBM50126765
Substrate
n/a
Meas. Tech.
ChEMBL_147038 (CHEMBL753341)
Ki
>10000±n/a nM
Citation
 Holzgrabe, U; Brandt, W Mechanism of action of the diazabicyclononanone-type kappa-agonists. J Med Chem 46:1383-9 (2003) [PubMed]  Article 
Target
Name:
Delta-type opioid receptor
Synonyms:
Delta-type opioid receptor (DOR) | OPIATE Delta | Opioid receptor | DOR-1 | Delta-type opioid receptor | Opioid receptor A | Delta opioid receptor | Voltage-gated potassium channel | Opiate Delta 1 | Cytochrome P450 3A4 | OPRD_RAT | Oprd1 | Ror-a | Opioid receptors; mu & delta
Type:
G Protein-Coupled Receptor (GPCR)
Mol. Mass.:
40465.04
Organism:
Rat
Description:
Competition binding assays were using CHO-K1 cell membranes expressing the opioid receptor.
Residue:
372
Sequence:
MEPVPSARAELQFSLLANVSDTFPSAFPSASANASGSPGARSASSLALAIAITALYSAVCAVGLLGNVLVMFGIVRYTKLKTATNIYIFNLALADALATSTLPFQSAKYLMETWPFGELLCKAVLSIDYYNMFTSIFTLTMMSVDRYIAVCHPVKALDFRTPAKAKLINICIWVLASGVGVPIMVMAVTQPRDGAVVCTLQFPSPSWYWDTVTKICVFLFAFVVPILIITVCYGLMLLRLRSVRLLSGSKEKDRSLRRITRMVLVVVGAFVVCWAPIHIFVIVWTLVDINRRDPLVVAALHLCIALGYANSSLNPVLYAFLDENFKRCFRQLCRAPCGGQEPGSLRRPRQATARERVTACTPSDGPGGGAAA
  
Inhibitor
Name:
BDBM50126765
Synonyms:
3,7-Dimethyl-2,4-di-pyridin-2-yl-3,7-diaza-bicyclo[3.3.1]nonan-9-one | CHEMBL287392
Type:
Small organic molecule
Emp. Form.:
TBD
Mol. Mass.:
TBD
SMILES:
TBD
Structure:
Search PDB for entries with ligand similarity: