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Target
Chymotrypsinogen A
Ligand
BDBM50633735
Substrate
n/a
Meas. Tech.
ChEMBL_2378831
IC50
2700±n/a nM
Citation
 Holland, DC; Schroder, WA; Calcott, MJ; Kaemmerer, E; Avery, VM; Ekins, MG; Carroll, AR Cyclotheonellazoles D-I, Potent Elastase Inhibitory Thiazole-Containing Cyclic Peptides from  J Nat Prod 86:2216-2227 (2023) [PubMed] 
Target
Name:
Chymotrypsinogen A
Synonyms:
Chymotrypsin A chain A | Chymotrypsin A chain B | Chymotrypsin A chain C | Chymotrypsinogen A | alpha-Chymotrypsin (α-Chymotrypsin) | Chymotrypsin A | CTRA_BOVIN | Alpha-chymotrypsin
Type:
Serine protease
Mol. Mass.:
25670.88
Organism:
Bovine
Description:
n/a
Residue:
245
Sequence:
CGVPAIQPVLSGLSRIVNGEEAVPGSWPWQVSLQDKTGFHFCGGSLINENWVVTAAHCGVTTSDVVVAGEFDQGSSSEKIQKLKIAKVFKNSKYNSLTINNDITLLKLSTAASFSQTVSAVCLPSASDDFAAGTTCVTTGWGLTRYTNANTPDRLQQASLPLLSNTNCKKYWGTKIKDAMICAGASGVSSCMGDSGGPLVCKKNGAWTLVGIVSWGSSTCSTSTPGVYARVTALVNWVQQTLAAN
  
Inhibitor
Name:
BDBM50633735
Synonyms:
CHEMBL5397807
Type:
Small organic molecule
Emp. Form.:
TBD
Mol. Mass.:
TBD
SMILES:
TBD
Structure:
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