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Target
Carnitine O-palmitoyltransferase 1, liver isoform
Ligand
BDBM50122839
Substrate
n/a
Meas. Tech.
ChEMBL_2444417
Ki
360±n/a nM
Citation
 Fan, Z; Hao, Y; Huo, Y; Cao, F; Li, L; Xu, J; Song, Y; Yang, K Modulators for palmitoylation of proteins and small molecules. Eur J Med Chem 271:0[PubMed] 
Target
Name:
Carnitine O-palmitoyltransferase 1, liver isoform
Synonyms:
CPT I | CPT1-L | CPTI-L | Carnitine O-palmitoyltransferase I, liver isoform | CPT1A_HUMAN | CPT1A | CPT1
Type:
PROTEIN
Mol. Mass.:
88389.31
Organism:
Human
Description:
ChEMBL_887463
Residue:
773
Sequence:
MAEAHQAVAFQFTVTPDGIDLRLSHEALRQIYLSGLHSWKKKFIRFKNGIITGVYPASPSSWLIVVVGVMTTMYAKIDPSLGIIAKINRTLETANCMSSQTKNVVSGVLFGTGLWVALIVTMRYSLKVLLSYHGWMFTEHGKMSRATKIWMGMVKIFSGRKPMLYSFQTSLPRLPVPAVKDTVNRYLQSVRPLMKEEDFKRMTALAQDFAVGLGPRLQWYLKLKSWWATNYVSDWWEEYIYLRGRGPLMVNSNYYAMDLLYILPTHIQAARAGNAIHAILLYRRKLDREEIKPIRLLGSTIPLCSAQWERMFNTSRIPGEETDTIQHMRDSKHIVVYHRGRYFKVWLYHDGRLLKPREMEQQMQRILDNTSEPQPGEARLAALTAGDRVPWARCRQAYFGRGKNKQSLDAVEKAAFFVTLDETEEGYRSEDPDTSMDSYAKSLLHGRCYDRWFDKSFTFVVFKNGKMGLNAEHSWADAPIVAHLWEYVMSIDSLQLGYAEDGHCKGDINPNIPYPTRLQWDIPGECQEVIETSLNTANLLANDVDFHSFPFVAFGKGIIKKCRTSPDAFVQLALQLAHYKDMGKFCLTYEASMTRLFREGRTETVRSCTTESCDFVRAMVDPAQTVEQRLKLFKLASEKHQHMYRLAMTGSGIDRHLFCLYVVSKYLAVESPFLKEVLSEPWRLSTSQTPQQQVELFDLENNPEYVSSGGGFGPVADDGYGVSYILVGENLINFHISSKFSCPETDSHRFGRHLKEAMTDIITLFGLSSNSKK
  
Inhibitor
Name:
BDBM50122839
Synonyms:
[3-Carboxy-2-(3-tetradecyl-ureido)-propyl]-trimethyl-ammonium | CHEMBL106227
Type:
Small organic molecule
Emp. Form.:
n/a
Mol. Mass.:
n/a
SMILES:
CCCCCCCCCCCCCCNC(=O)N[C@H](CC([O-])=O)C[N+](C)(C)C
Structure:
Search PDB for entries with ligand similarity: