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Target
Kappa-type opioid receptor
Ligand
BDBM50008984
Substrate
n/a
Meas. Tech.
ChEBML_146364
Ki
1130±n/a nM
Citation
 Wang, C; McFadyen, IJ; Traynor, JR; Mosberg, HI Design of a high affinity peptidomimetic opioid agonist from peptide pharmacophore models. Bioorg Med Chem Lett 8:2685-8 (1999) [PubMed]  Article 
Target
Name:
Kappa-type opioid receptor
Synonyms:
Kappa Opioid Receptor | OPIATE Kappa | Opiate Kappa 1 | OPRK_CAVPO | OPRK1 | mu/kappa opioid receptor
Type:
G Protein-Coupled Receptor (GPCR)
Mol. Mass.:
42744.99
Organism:
Guinea pig
Description:
P41144
Residue:
380
Sequence:
MGRRRQGPAQPASELPARNACLLPNGSAWLPGWAEPDGNGSAGPQDEQLEPAHISPAIPVIITAVYSVVFVVGLVGNSLVMFVIIRYTKMKTATNIYIFNLALADALVTTTMPFQSTVYLMNSWPFGDVLCKIVISIDYYNMFTSIFTLTMMSVDRYIAVCHPVKALDFRTPLKAKIINICIWLLSSSVGISAIILGGTKVREDVDIIECSLQFPDDDYSWWDLFMKICVFVFAFVIPVLIIIVCYTLMILRLKSVRLLSGSREKDRNLRRITRLVLVVVAVFIICWTPIHIFILVEALGSTSHSTAALSSYYFCIALGYTNSSLNPILYAFLDENFKRCFRDFCFPIKMRMERQSTSRVRNTVQDPAYMRNVDGVNKPV
  
Inhibitor
Name:
BDBM50008984
Synonyms:
N-(1-Phenethyl-piperidin-4-yl)-N-phenyl-propionamide(Fentanyl) | CHEMBL596 | Fentora | 4-(4-Chloro-benzyl)-2-(1-methyl-azepan-4-yl)-2H-phthalazin-1-one | Ionsys | Duragesic-100 | Fentanyl-75 | Duragesic-25 | Fentanyl-50 | N-(1-Phenethyl-piperidin-4-yl)-N-phenyl-propionamide | FENTANYL CITRATE | Duragesic-12 | Duragesic-50 | Innovar | Duragesic-75 | FENTANYL-HCl | Fentanyl-100 | N-(1-phenethylpiperidin-4-yl)-N-phenylpropionamide | Fentanyl-12 | Fentanyl-25 | FENTANYL | US20230399418, Compound Fentanyl
Type:
Small organic molecule
Emp. Form.:
TBD
Mol. Mass.:
TBD
SMILES:
TBD
Structure:
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