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Target
Mu-type opioid receptor
Ligand
BDBM50000655
Substrate
n/a
Meas. Tech.
ChEBML_221923
Ki
52±n/a nM
Citation
 Wang, C; McFadyen, IJ; Traynor, JR; Mosberg, HI Design of a high affinity peptidomimetic opioid agonist from peptide pharmacophore models. Bioorg Med Chem Lett 8:2685-8 (1999) [PubMed]  Article 
Target
Name:
Mu-type opioid receptor
Synonyms:
OPIATE Mu | Mu opioid receptor | Mu-type opioid receptor (Mu) | M-OR-1 | MOR-1 | OPRM_CAVPO | OPRM1
Type:
Enzyme Catalytic Domain
Mol. Mass.:
11165.58
Organism:
Guinea pig
Description:
P97266
Residue:
98
Sequence:
YTKMKTATNIYIFNLALADALATSTLPFQSVNYLMGTWPFGTILCKIVISIDYYNMFTSIFTLCTMSVDRYIAVCHPVKALDFRTPRNAKTVNVCNWI
  
Inhibitor
Name:
BDBM50000655
Synonyms:
CHEMBL39192 | 10-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-7-benzyl-3,3-dimethyl-6,9-dioxo-1,2-dithia-5,8-diaza-cycloundecane-4-carboxylic acid | (4R,7S,10R)-10-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-7-benzyl-3,3-dimethyl-6,9-dioxo-1,2-dithia-5,8-diaza-cycloundecane-4-carboxylic acid
Type:
Small organic molecule
Emp. Form.:
TBD
Mol. Mass.:
TBD
SMILES:
TBD
Structure:
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