Reaction Details Report a problem with these data
Target
C-C chemokine receptor type 5
Ligand
BDBM50378977
Substrate
n/a
Meas. Tech.
ChEMBL_809511 (CHEMBL2015428)
Kd
49000±n/a nM
Citation
 Navratilova, I; Besnard, J; Hopkins, AL Screening for GPCR Ligands Using Surface Plasmon Resonance. ACS Med Chem Lett 2:549-554 (2011) [PubMed]  Article 
Target
Name:
C-C chemokine receptor type 5
Synonyms:
CCR-5 | C-C CKR-5 | CC-CKR-5 | CHEMR13 | CCR5/mu opioid receptor complex | HIV-1 fusion coreceptor | CD_antigen=CD195 | CCR5_HUMAN | CCR5 | CMKBR5 | C-C chemokine receptor type 5
Type:
Enzyme
Mol. Mass.:
40540.21
Organism:
Human
Description:
P51681
Residue:
352
Sequence:
MDYQVSSPIYDINYYTSEPCQKINVKQIAARLLPPLYSLVFIFGFVGNMLVILILINCKRLKSMTDIYLLNLAISDLFFLLTVPFWAHYAAAQWDFGNTMCQLLTGLYFIGFFSGIFFIILLTIDRYLAVVHAVFALKARTVTFGVVTSVITWVVAVFASLPGIIFTRSQKEGLHYTCSSHFPYSQYQFWKNFQTLKIVILGLVLPLLVMVICYSGILKTLLRCRNEKKRHRAVRLIFTIMIVYFLFWAPYNIVLLLNTFQEFFGLNNCSSSNRLDQAMQVTETLGMTHCCINPIIYAFVGEKFRNYLLVFFQKHIAKRFCKCCSIFQQEAPERASSVYTRSTGEQEISVGL
  
Inhibitor
Name:
BDBM50378977
Synonyms:
CHEMBL1621896
Type:
Small organic molecule
Emp. Form.:
TBD
Mol. Mass.:
TBD
SMILES:
TBD
Structure:
Search PDB for entries with ligand similarity: