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Target
Chromobox protein homolog 8
Ligand
BDBM50009526
Substrate
n/a
Meas. Tech.
ChEMBL_1336413 (CHEMBL3242417)
Kd
15000±n/a nM
Citation
 Simhadri, C; Daze, KD; Douglas, SF; Quon, TT; Dev, A; Gignac, MC; Peng, F; Heller, M; Boulanger, MJ; Wulff, JE; Hof, F Chromodomain antagonists that target the polycomb-group methyllysine reader protein chromobox homolog 7 (CBX7). J Med Chem 57:2874-83 (2014) [PubMed]  Article 
Target
Name:
Chromobox protein homolog 8
Synonyms:
Polycomb 3 homolog | Rectachrome 1 | hPc3 | CBX8_HUMAN | CBX8 | PC3 | RC1
Type:
PROTEIN
Mol. Mass.:
43415.86
Organism:
Human
Description:
ChEMBL_108272
Residue:
389
Sequence:
MELSAVGERVFAAEALLKRRIRKGRMEYLVKWKGWSQKYSTWEPEENILDARLLAAFEEREREMELYGPKKRGPKPKTFLLKAQAKAKAKTYEFRSDSARGIRIPYPGRSPQDLASTSRAREGLRNMGLSPPASSTSTSSTCRAEAPRDRDRDRDRDRERDRERERERERERERERERERGTSRVDDKPSSPGDSSKKRGPKPRKELPDPSQRPLGEPSAGLGEYLKGRKLDDTPSGAGKFPAGHSVIQLARRQDSDLVQCGVTSPSSAEATGKLAVDTFPARVIKHRAAFLEAKGQGALDPNGTRVRHGSGPPSSGGGLYRDMGAQGGRPSLIARIPVARILGDPEEESWSPSLTNLEKVVVTDVTSNFLTVTIKESNTDQGFFKEKR
  
Inhibitor
Name:
BDBM50009526
Synonyms:
CHEMBL3234440
Type:
Small organic molecule
Emp. Form.:
TBD
Mol. Mass.:
TBD
SMILES:
TBD
Structure:
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