Reaction Details
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C-X-C chemokine receptor type 4
Ligand
BDBM50155311
Substrate
n/a
Meas. Tech.
ChEMBL_1576376 (CHEMBL3802805)
IC50
92±n/a nM
Citation
Zhan, P; Pannecouque, C; De Clercq, E; Liu, X Anti-HIV Drug Discovery and Development: Current Innovations and Future Trends. J Med Chem 59:2849-78 (2016) [PubMed] Article More Info.:
Target
Name:
C-X-C chemokine receptor type 4
Synonyms:
C-X-C chemokine receptor type 4 | NPYRL | CXCR-4 | HM89 | CXC-R4 | SDF-1 receptor | CD_antigen=CD184 | Stromal cell-derived factor 1 receptor | LCR1 | LESTR | Fusin | Leukocyte-derived seven transmembrane domain receptor | FB22 | C-X-C chemokine receptor type 4 (CXCR4) | CXCR4_HUMAN | CXCR4
Type:
Enzyme
Mol. Mass.:
39754.61
Organism:
Human
Description:
P61073
Residue:
352
Sequence:
MEGISIYTSDNYTEEMGSGDYDSMKEPCFREENANFNKIFLPTIYSIIFLTGIVGNGLVILVMGYQKKLRSMTDKYRLHLSVADLLFVITLPFWAVDAVANWYFGNFLCKAVHVIYTVNLYSSVLILAFISLDRYLAIVHATNSQRPRKLLAEKVVYVGVWIPALLLTIPDFIFANVSEADDRYICDRFYPNDLWVVVFQFQHIMVGLILPGIVILSCYCIIISKLSHSKGHQKRKALKTTVILILAFFACWLPYYIGISIDSFILLEIIKQGCEFENTVHKWISITEALAFFHCCLNPILYAFLGAKFKTSAQHALTSVSRGSSLKILSKGKRGGHSSVSTESESSSFHSS
