Target
14-3-3 protein beta/alpha
Ligand
BDBM50177028
Substrate
n/a
Meas. Tech.
ChEMBL_1582330 (CHEMBL3816073)
Kd
70.0±n/a nM
Citation
 Watanabe, NOsada, H Small molecules that target phosphorylation dependent protein-protein interaction. Bioorg Med Chem 24:3246-54 (2016) [PubMed]  Article 
Target
Name:
14-3-3 protein beta/alpha
Synonyms:
14-3-3 protein beta/alpha | 14-3-3 protein beta/alpha, N-terminally processed | KCIP-1 | Protein 1054 | Protein kinase C inhibitor protein 1 | 1433B_HUMAN | YWHAB
Type:
PROTEIN
Mol. Mass.:
28068.98
Organism:
Human
Description:
ChEMBL_112364
Residue:
246
Sequence:
MTMDKSELVQKAKLAEQAERYDDMAAAMKAVTEQGHELSNEERNLLSVAYKNVVGARRSSWRVISSIEQKTERNEKKQQMGKEYREKIEAELQDICNDVLELLDKYLIPNATQPESKVFYLKMKGDYFRYLSEVASGDNKQTTVSNSQQAYQEAFEISKKEMQPTHPIRLGLALNFSVFYYEILNSPEKACSLAKTAFDEAIAELDTLNEESYKDSTLIMQLLRDNLTLWTSENQGDEGDAGEGEN
  
Inhibitor
Name:
BDBM50177028
Synonyms:
CHEMBL3814675
Type:
Small organic molecule
Emp. Form.:
TBD
Mol. Mass.:
TBD
SMILES:
TBD
Structure:
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