Target
14-3-3 protein eta
Ligand
BDBM50177028
Substrate
n/a
Meas. Tech.
ChEMBL_1582332 (CHEMBL3816075)
Kd
70.0±n/a nM
Citation
 Watanabe, NOsada, H Small molecules that target phosphorylation dependent protein-protein interaction. Bioorg Med Chem 24:3246-54 (2016) [PubMed]  Article 
Target
Name:
14-3-3 protein eta
Synonyms:
14-3-3 protein eta | Protein AS1 | 1433F_HUMAN | YWHAH | YWHA1
Type:
PROTEIN
Mol. Mass.:
28205.81
Organism:
Human
Description:
ChEMBL_110546
Residue:
246
Sequence:
MGDREQLLQRARLAEQAERYDDMASAMKAVTELNEPLSNEDRNLLSVAYKNVVGARRSSWRVISSIEQKTMADGNEKKLEKVKAYREKIEKELETVCNDVLSLLDKFLIKNCNDFQYESKVFYLKMKGDYYRYLAEVASGEKKNSVVEASEAAYKEAFEISKEQMQPTHPIRLGLALNFSVFYYEIQNAPEQACLLAKQAFDDAIAELDTLNEDSYKDSTLIMQLLRDNLTLWTSDQQDEEAGEGN
  
Inhibitor
Name:
BDBM50177028
Synonyms:
CHEMBL3814675
Type:
Small organic molecule
Emp. Form.:
TBD
Mol. Mass.:
TBD
SMILES:
TBD
Structure:
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