Reaction Details Report a problem with these data
Target
C-X-C chemokine receptor type 4
Ligand
BDBM50196241
Substrate
n/a
Meas. Tech.
ChEMBL_1618265 (CHEMBL3860434)
EC50
81±n/a nM
Citation
 Mona, CE; Besserer-Offroy, É; Cabana, J; Lefrançois, M; Boulais, PE; Lefebvre, MR; Leduc, R; Lavigne, P; Heveker, N; Marsault, É; Escher, E Structure-Activity Relationship and Signaling of New Chimeric CXCR4 Agonists. J Med Chem 59:7512-24 (2016) [PubMed]  Article 
Target
Name:
C-X-C chemokine receptor type 4
Synonyms:
C-X-C chemokine receptor type 4 | NPYRL | CXCR-4 | HM89 | CXC-R4 | SDF-1 receptor | CD_antigen=CD184 | Stromal cell-derived factor 1 receptor | LCR1 | LESTR | Fusin | Leukocyte-derived seven transmembrane domain receptor | FB22 | C-X-C chemokine receptor type 4 (CXCR4) | CXCR4_HUMAN | CXCR4
Type:
Enzyme
Mol. Mass.:
39754.61
Organism:
Human
Description:
P61073
Residue:
352
Sequence:
MEGISIYTSDNYTEEMGSGDYDSMKEPCFREENANFNKIFLPTIYSIIFLTGIVGNGLVILVMGYQKKLRSMTDKYRLHLSVADLLFVITLPFWAVDAVANWYFGNFLCKAVHVIYTVNLYSSVLILAFISLDRYLAIVHATNSQRPRKLLAEKVVYVGVWIPALLLTIPDFIFANVSEADDRYICDRFYPNDLWVVVFQFQHIMVGLILPGIVILSCYCIIISKLSHSKGHQKRKALKTTVILILAFFACWLPYYIGISIDSFILLEIIKQGCEFENTVHKWISITEALAFFHCCLNPILYAFLGAKFKTSAQHALTSVSRGSSLKILSKGKRGGHSSVSTESESSSFHSS
  
Inhibitor
Name:
BDBM50196241
Synonyms:
CHEMBL3902240
Type:
Small organic molecule
Emp. Form.:
TBD
Mol. Mass.:
TBD
SMILES:
TBD
Structure:
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