Reaction Details Report a problem with these data
Target
Norepinephrine transporter
Ligand
BDBM35229
Substrate
n/a
Ki
0.06±n/a nM
Comments
PDSP_638
Citation
 Davids, E; Zhang, K; Kula, NS; Tarazi, FI; Baldessarini, RJ Effects of norepinephrine and serotonin transporter inhibitors on hyperactivity induced by neonatal 6-hydroxydopamine lesioning in rats. J Pharmacol Exp Ther 301:1097-102 (2002) [PubMed]  Article 
Target
Name:
Norepinephrine transporter
Synonyms:
n/a
Type:
Enzyme Catalytic Domain
Mol. Mass.:
2082.45
Organism:
Rat
Description:
Norepinephrine transporter 0 RAT::Q9JIA2
Residue:
19
Sequence:
MLLARMKPQVQPELGGADQ
  
Inhibitor
Name:
BDBM35229
Synonyms:
Desmethylimipramine | 3-(10,11-dihydro-5H-dibenzo[b,f]azepin-5-yl)-N-methylpropan-1-amine | monodemethylimipramine | Desipramin | 5-(gamma-methylaminopropyl)iminodibenzyl | norimipramine | CHEMBL72 | DESIPRAMINE HYDROCHLORIDE | demethylimipramine | N-(3-methylaminopropyl)iminobibenzyl | DMI | Desipramine | US9944618, Compound ID No. 174
Type:
Small organic molecule
Emp. Form.:
TBD
Mol. Mass.:
TBD
SMILES:
TBD
Structure:
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