Target
Casein kinase I isoform delta
Ligand
BDBM50013720
Substrate
n/a
Ki
9900±n/a nM
Comments
PDSP_6411
Citation
 Bain, JMcLauchlan, HElliott, MCohen, P The specificities of protein kinase inhibitors: an update. Biochem J 371:199-204 (2003) [PubMed]  Article 
Target
Name:
Casein kinase I isoform delta
Synonyms:
Casein kinase 1 Delta | Casein kinase I isoform delta | CK1, delta | casein kinase 1, delta | Casein kinase I delta | KC1D_RAT | Csnk1d | Hckid
Type:
Enzyme
Mol. Mass.:
47342.73
Organism:
Rat
Description:
Q06486
Residue:
415
Sequence:
MELRVGNRYRLGRKIGSGSFGDIYLGTDIAAGEEVAIKLECVKTKHPQLHIESKIYKMMQGGVGIPTIRWCGAEGDYNVMVMELLGPSLEDLFNFCSRKFSLKTVLLLADQMISRIEYIHSKNFIHRDVKPDNFLMGLGKKGNLVYIIDFGLAKKYRDARTHQHIPYRENKNLTGTARYASINTHLGIEQSRRDDLESLGYVLMYFNLGSLPWQGLKAATKRQKYERISEKKMSTPIEVLCKGYPSEFATYLNFCRSLRFDDKPDYSYLRQLFRNLFHRQGFSYDYVFDWNMLKFGASRAADDAERERRDREERLRHSRNPATRGLPSTASGRLRGTQEVAPPTPLTPTSHTANTSPRPVSGMERERKVSMRLHRGAPVNVSSSDLTGRQDTSRMSTSQIPGRVASSGLQSVVHR
  
Inhibitor
Name:
BDBM50013720
Synonyms:
CHEMBL65063 | PP3 | cid_4879 | 1-Phenyl-1H-pyrazolo[3,4-d]pyrimidin-4-ylamine
Type:
Small organic molecule
Emp. Form.:
TBD
Mol. Mass.:
TBD
SMILES:
TBD
Structure:
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