Reaction Details Report a problem with these data
Target
Matrilysin
Ligand
BDBM50070942
Substrate
n/a
Meas. Tech.
SPA Assay
pH
7.5000±0.0000
Temperature
295.1500±0.0000 K
IC50
8300±3700 nM
Citation
 Niu, X; Fan, X; Sun, J; Ting, P; Narula, S; Lundell, D Inhibition of fucosyltransferase VII by gallic acid and its derivatives. Arch Biochem Biophys 425:51-7 (2004) [PubMed]  Article 
Target
Name:
Matrilysin
Synonyms:
Matrix metalloproteinase 7 | Matrix metalloproteinase-7 (MMP-7) | MMP7_HUMAN | MMP7 | MPSL1 | PUMP1 | Matrix metalloproteinase-7 (MMP7)
Type:
Enzyme
Mol. Mass.:
29681.54
Organism:
Human
Description:
P09237
Residue:
267
Sequence:
MRLTVLCAVCLLPGSLALPLPQEAGGMSELQWEQAQDYLKRFYLYDSETKNANSLEAKLKEMQKFFGLPITGMLNSRVIEIMQKPRCGVPDVAEYSLFPNSPKWTSKVVTYRIVSYTRDLPHITVDRLVSKALNMWGKEIPLHFRKVVWGTADIMIGFARGAHGDSYPFDGPGNTLAHAFAPGTGLGGDAHFDEDERWTDGSSLGINFLYAATHELGHSLGMGHSSDPNAVMYPTYGNGDPQNFKLSQDDIKGIQKLYGKRSNSRKK
  
Inhibitor
Name:
BDBM50070942
Synonyms:
(-)-Epigallocatechin-3-o-gallate | (-)-Epigallocatechin gallate | Epigallocatechin monogallate, B | cid_65064 | CHEMBL297453 | EGCG | Epigallocatechin 3-gallate | (-)-epigallocatechin 3-gallate | (2R,3R)-5,7-dihydroxy-2-(3,4,5-trihydroxyphenyl)-3,4-dihydro-2H-chromen-3-yl 3,4,5-trihydroxybenzoate | US20240336588, Compound 3
Type:
Small organic molecule
Emp. Form.:
TBD
Mol. Mass.:
TBD
SMILES:
TBD
Structure:
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