Reaction Details Report a problem with these data
Target
Serine/threonine-protein kinase haspin [465-798]
Ligand
BDBM103302
Substrate
n/a
Meas. Tech.
ITC
pH
7.5±0
Temperature
288.15±0 K
Kd
297± 1 nM
Citation
Chaikuad, A; Tacconi, EM; Zimmer, J; Liang, Y; Gray, NS; Tarsounas, M; Knapp, S A unique inhibitor binding site in ER K1/2 is associated with slow binding kinetics Nat Chem Biol 10:853-860 (2014) [PubMed] Article
More Info.:
Target
Name:
Serine/threonine-protein kinase haspin [465-798]
Synonyms:
GSG2 | HASPIN | HASP_HUMAN | Haspin (aa 465-798)
Type:
Protein
Mol. Mass.:
37973.67
Organism:
Homo sapiens (Human)
Description:
Haspin kinase domain 465-798aa (curated by PDB 4QTC)
Residue:
334
Sequence:
GECSQKGPVPFSHCLPTEKLQRCEKIGEGVFGEVFQTIADHTPVAIKIIAIEGPDLVNGSHQKTFEEILPEIIISKELSLLSGEVCNRTEGFIGLNSVHCVQGSYPPLLLKAWDHYNSTKGSANDRPDFFKDDQLFIVLEFEFGGIDLEQMRTKLSSLATAKSILHQLTASLAVAEASLRFEHRDLHWGNVLLKKTSLKKLHYTLNGKSSTIPSCGLQVSIIDYTLSRLERDGIVVFCDVSMDEDLFTGDGDYQFDIYRLMKKENNNRWGEYHPYSNVLWLHYLTDKMLKQMTFKTKCNTPAMKQIKRKIQEFHRTMLNFSSATDLLCQHSLFK