Reaction Details
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Target
Acyl-protein thioesterase 2 [L78I,A85S,P86Q]
Ligand
BDBM207991
Substrate
n/a
Meas. Tech.
Steady-State Kinetic Assays
pH
6.5000±n/a
Ki
3400±260 nM
Comments
extracted
Citation

More Info.:
Target
Name:
Acyl-protein thioesterase 2 [L78I,A85S,P86Q]
Synonyms:
LYPA2_HUMAN | LYPLA2 | APT2 | Acyl-protein thioesterase 2 (APT2 L78I/A85S/P86Q)
Type:
Protein
Mol. Mass.:
24787.24
Organism:
Human
Description:
Human APT2 with L78I/A85S/P86Q mutations
Residue:
231
Sequence:
MCGNTMSVPLLTDAATVSGAERETAAVIFLHGLGDTGHSWADALSTIRLPHVKYICPHAPRIPVTLNMKMVMPSWFDIMGLSPDSQEDEAGIKKAAENIKALIEHEMKNGIPANRIVLGGFSQGGALSLYTALTCPHPLAGIVALSCWLPLHRAFPQAANGSAKDLAILQCHGELDPMVPVRFGALTAEKLRSVVTPARVQFKTYPGVMHSSCPQEMAAVKEFLEKLLPPV