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Target
Cannabinoid receptor 2
Ligand
BDBM50117099
Substrate
n/a
Meas. Tech.
[35S]GTPγS Binding Assay
pH
7.5000±n/a
EC50
18.3±n/a nM
Comments
extracted
Citation
 Mechoulam, R; Magid, L; Shohami, E; Bab, I Arylated camphenes, processes for their preparation and uses thereof US Patent  US9365534 Publication Date 6/14/2016 
Target
Name:
Cannabinoid receptor 2
Synonyms:
CB2 | CB2A | CB2B | CNR2 | CNR2_HUMAN | CANNABINOID CB2 | CB-2 | CX5 | Cannabinoid CB2 receptor | Cannabinoid receptor 2 (CB2) | Cannabinoid receptor 2 (CB2R) | hCB2
Type:
G Protein-Coupled Receptor (GPCR)
Mol. Mass.:
39690.94
Organism:
Human
Description:
P34972
Residue:
360
Sequence:
MEECWVTEIANGSKDGLDSNPMKDYMILSGPQKTAVAVLCTLLGLLSALENVAVLYLILSSHQLRRKPSYLFIGSLAGADFLASVVFACSFVNFHVFHGVDSKAVFLLKIGSVTMTFTASVGSLLLTAIDRYLCLRYPPSYKALLTRGRALVTLGIMWVLSALVSYLPLMGWTCCPRPCSELFPLIPNDYLLSWLLFIAFLFSGIIYTYGHVLWKAHQHVASLSGHQDRQVPGMARMRLDVRLAKTLGLVLAVLLICWFPVLALMAHSLATTLSDQVKKAFAFCSMLCLINSMVNPVIYALRSGEIRSSAHHCLAHWKKCVRGLGSEAKEEAPRSSVTETEADGKITPWPDSRDLDLSDC
  
Inhibitor
Name:
BDBM50117099
Synonyms:
CHEMBL3613118 | US9365534, HU-308
Type:
Small organic molecule
Emp. Form.:
C27H42O3
Mol. Mass.:
414.31
SMILES:
[H][C@@]12C[C@@]([H])(C(CO)=C[C@H]1c1c(OC)cc(cc1OC)C(C)(C)CCCCCC)C2(C)C |r,c:7,TLB:10:9:29:2,THB:6:5:29:2|
Structure:
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