BDBM23891 3-amidinophenylalanine deriv., 35::CHEMBL107955::ethyl 4-[(2S)-3-(3-carbamimidoylphenyl)-2-{[2,4,6-tris(propan-2-yl)benzene]sulfonamido}propanoyl]piperazine-1-carboxylate
SMILES CCOC(=O)N1CCN(CC1)C(=O)[C@H](Cc1cccc(c1)C(N)=N)NS(=O)(=O)c1c(cc(cc1C(C)C)C(C)C)C(C)C
InChI Key InChIKey=ISJSHQTWOHGCMM-NDEPHWFRSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 25 hits for monomerid = 23891
Affinity DataKi: 37nMAssay Description:Compound was tested for inhibition of trypsinMore data for this Ligand-Target Pair
Affinity DataKi: 320nM ΔG°: -8.85kcal/molepH: 8.0 T: 25°CAssay Description:The measurements were carried out on a microplate reader. Two concentrations of the substrate and five concentrations of the inhibitor were used. Af...More data for this Ligand-Target Pair
Affinity DataKi: 370nMAssay Description:Inhibition of matriptase (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 390nMAssay Description:Inhibition of human plasma plasmin using pyroGlu-Pro-Arg-p-NA.HCl as substrate preincubated for 15 mins prior sustrate addition measured for 10 mins ...More data for this Ligand-Target Pair
Affinity DataKi: 390nMAssay Description:The measurements were carried out on a microplate reader. Two concentrations of the substrate and five concentrations of the inhibitor were used. Af...More data for this Ligand-Target Pair
Affinity DataKi: 390nMAssay Description:Compound was tested for inhibition of plasminMore data for this Ligand-Target Pair
Affinity DataKi: 390nMAssay Description:Inhibition of human plasminMore data for this Ligand-Target Pair
Affinity DataKi: 410nMAssay Description:The measurements were carried out on a microplate reader. Two concentrations of the substrate and five concentrations of the inhibitor were used. Af...More data for this Ligand-Target Pair
Affinity DataKi: 410nMAssay Description:Inhibition of human uPA using pyroGlu-Gly-Arg-p-NA.HCl as substrate preincubated for 15 mins prior sustrate addition measured for 10 mins by spectrop...More data for this Ligand-Target Pair
Affinity DataKi: 410nMAssay Description:Inhibition of uPA (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 410nMAssay Description:Compound was tested for inhibition of plasminogen activator urokinase(microPa)More data for this Ligand-Target Pair
Affinity DataKi: 490nMAssay Description:Inhibition of human plasma thrombin using pyroGlu-Pro-Arg-p-NA.HCl as substrate preincubated for 15 mins prior sustrate addition measured for 10 mins...More data for this Ligand-Target Pair
Affinity DataKi: 490nMAssay Description:The measurements were carried out on a microplate reader. Two concentrations of the substrate and five concentrations of the inhibitor were used. Af...More data for this Ligand-Target Pair
Affinity DataKi: 490nMAssay Description:Compound was tested for inhibition of thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 500nMAssay Description:Inhibition of thrombin (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 650nMAssay Description:Inhibition of uPA (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 980nMAssay Description:Inhibition of factor 10a (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 1.46E+3nMAssay Description:Inhibition of plasmin (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 1.70E+3nMAssay Description:Compound was tested for inhibition of Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 1.70E+3nMAssay Description:The measurements were carried out on a microplate reader. Two concentrations of the substrate and five concentrations of the inhibitor were used. Af...More data for this Ligand-Target Pair
Affinity DataKi: 2.51E+3nMAssay Description:Inhibition of tPA (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 4.90E+3nMAssay Description:Inhibition of recombinant tPA using H-D-Ile-Pro-Arg-pNA.2HCl as substrate preincubated for 15 mins prior sustrate addition measured for 10 mins by sp...More data for this Ligand-Target Pair
Affinity DataKi: 6.30E+3nMAssay Description:Compound was tested for inhibition of tryptaseMore data for this Ligand-Target Pair
Affinity DataKi: 7.20E+3nMAssay Description:Compound was tested for inhibition of plasma kallikreinMore data for this Ligand-Target Pair