BDBM30075 triazolothiadiazine, 7E

SMILES COc1cccc(c1)C1=Nn2c(SC1)nnc2-c1ccc(OC)cc1OC

InChI Key InChIKey=GCKOBNRYFXDBAO-UHFFFAOYSA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 30075   

TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A(Human)
Nih

LigandBDBM30075(triazolothiadiazine, 7E)Copy SMILESCopy InChI

Affinity DataIC50:  1.34E+4nMpH: 7.2 T: 22°CAssay Description:Inhibition of PDE4A was performed using IMAP technology (Molecular Devices, CA). PDE4A1A mixture was dispensed into 1536-well black/solid bottom assa...More data for this Ligand-Target Pair

Target InfoPDBMMDBReactome pathwayKEGG
UniProtKB/SwissProt
B.MOADDrugBankantibodypediaGoogleScholar

Ligand InfoPC cidPC sidSimilars

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