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Found 41 with Last Name = 'barassin' and Initial = 's'
Target3-oxo-5-alpha-steroid 4-dehydrogenase 2(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50334788((17beta-(N-tert-butylcarbamoyl)-4-aza-5alpha-andro...)
Affinity DataIC50:  5nMAssay Description:Inhibition of Steroid 5-alpha-reductase type 2 from human benign prostatic hyperplasia (BPH) tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

Target3-oxo-5-alpha-steroid 4-dehydrogenase 2(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50116431(CHEMBL113726 | {4-[1-(2,2-Dicyclohexyl-acetyl)-pip...)
Affinity DataIC50:  6nMAssay Description:Inhibition of Steroid 5-alpha-reductase type 2 from human benign prostatic hyperplasia (BPH) tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-oxo-5-alpha-steroid 4-dehydrogenase 2(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50116424(CHEMBL115438 | {4-[1-(2,2-Dicyclohexyl-acetyl)-pip...)
Affinity DataIC50:  7nMAssay Description:Inhibition of Steroid 5-alpha-reductase type 2 from human benign prostatic hyperplasia (BPH) tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-oxo-5-alpha-steroid 4-dehydrogenase 1(Rattus norvegicus)
Saarland University

Curated by ChEMBL
LigandPNGBDBM50334788((17beta-(N-tert-butylcarbamoyl)-4-aza-5alpha-andro...)
Affinity DataIC50:  10nMAssay Description:Inhibition of Steroid 5-alpha-reductase type I from rat ventral prostate (RVP)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-oxo-5-alpha-steroid 4-dehydrogenase 2(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50116419(4-[1-(2,2-Dicyclohexyl-acetyl)-piperidin-4-ylidene...)
Affinity DataIC50:  11nMAssay Description:Inhibition of Steroid 5-alpha-reductase type 2 from human benign prostatic hyperplasia (BPH) tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-oxo-5-alpha-steroid 4-dehydrogenase 2(Rattus norvegicus)
Saarland University

Curated by ChEMBL
LigandPNGBDBM50334788((17beta-(N-tert-butylcarbamoyl)-4-aza-5alpha-andro...)
Affinity DataIC50:  11nMAssay Description:Inhibition of Steroid 5-alpha-reductase type 2 of rat ventral prostate (RVP)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-oxo-5-alpha-steroid 4-dehydrogenase 2(Rattus norvegicus)
Saarland University

Curated by ChEMBL
LigandPNGBDBM50116424(CHEMBL115438 | {4-[1-(2,2-Dicyclohexyl-acetyl)-pip...)
Affinity DataIC50:  38nMAssay Description:Inhibition of Steroid 5-alpha-reductase type 2 of rat ventral prostate (RVP)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-oxo-5-alpha-steroid 4-dehydrogenase 1(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50334788((17beta-(N-tert-butylcarbamoyl)-4-aza-5alpha-andro...)
Affinity DataIC50:  41nMAssay Description:In vitro inhibitory activity against Steroid 5-alpha-reductase type I of human DU 145 prostatic tumor cell lineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-oxo-5-alpha-steroid 4-dehydrogenase 2(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50116429(4-[1-(2,2-Dicyclohexyl-acetyl)-piperidin-4-ylidene...)
Affinity DataIC50:  60nMAssay Description:Inhibition of Steroid 5-alpha-reductase type 2 from human benign prostatic hyperplasia (BPH) tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-oxo-5-alpha-steroid 4-dehydrogenase 1(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50116418(CHEMBL323856 | [4-(1-Diphenylacetyl-piperidin-4-yl...)
Affinity DataIC50:  75nMAssay Description:In vitro inhibitory activity against Steroid 5-alpha-reductase type 2 of human benign prostatic hyperplasia (BPH) tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-oxo-5-alpha-steroid 4-dehydrogenase 2(Rattus norvegicus)
Saarland University

Curated by ChEMBL
LigandPNGBDBM50116429(4-[1-(2,2-Dicyclohexyl-acetyl)-piperidin-4-ylidene...)
Affinity DataIC50:  80nMAssay Description:Inhibition of Steroid 5-alpha-reductase type 2 of rat ventral prostate (RVP)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-oxo-5-alpha-steroid 4-dehydrogenase 2(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50116421(4-[1-(2,2-Dicyclohexyl-acetyl)-piperidin-4-ylidene...)
Affinity DataIC50:  130nMAssay Description:Inhibition of Steroid 5-alpha-reductase type 2 from human benign prostatic hyperplasia (BPH) tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-oxo-5-alpha-steroid 4-dehydrogenase 2(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50116416(4-[1-(Adamantane-1-carbonyl)-piperidin-4-ylideneme...)
Affinity DataIC50:  210nMAssay Description:Inhibition of Steroid 5-alpha-reductase type 2 from human benign prostatic hyperplasia (BPH) tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-oxo-5-alpha-steroid 4-dehydrogenase 2(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50116426(4-[1-(Adamantane-1-carbonyl)-piperidin-4-ylideneme...)
Affinity DataIC50:  260nMAssay Description:Inhibition of Steroid 5-alpha-reductase type 2 from human benign prostatic hyperplasia (BPH) tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-oxo-5-alpha-steroid 4-dehydrogenase 2(Rattus norvegicus)
Saarland University

Curated by ChEMBL
LigandPNGBDBM50116423(4-(1-Diphenylacetyl-piperidin-4-ylidenemethyl)-ben...)
Affinity DataIC50:  370nMAssay Description:Inhibition of Steroid 5-alpha-reductase type 2 of rat ventral prostate (RVP)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-oxo-5-alpha-steroid 4-dehydrogenase 2(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50116432(4-(1-Diphenylacetyl-piperidin-4-ylidenemethyl)-3-f...)
Affinity DataIC50:  410nMAssay Description:Inhibition of Steroid 5-alpha-reductase type 2 from human benign prostatic hyperplasia (BPH) tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-oxo-5-alpha-steroid 4-dehydrogenase 2(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50116433(4-[1-(Adamantane-1-carbonyl)-piperidin-4-yloxy]-be...)
Affinity DataIC50:  430nMAssay Description:Inhibition of Steroid 5-alpha-reductase type 2 from human benign prostatic hyperplasia (BPH) tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-oxo-5-alpha-steroid 4-dehydrogenase 2(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50116423(4-(1-Diphenylacetyl-piperidin-4-ylidenemethyl)-ben...)
Affinity DataIC50:  530nMAssay Description:Inhibition of Steroid 5-alpha-reductase type 2 from human benign prostatic hyperplasia (BPH) tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-oxo-5-alpha-steroid 4-dehydrogenase 1(Rattus norvegicus)
Saarland University

Curated by ChEMBL
LigandPNGBDBM50116417(4-(1-Diphenylcarbamoyl-piperidin-4-ylidenemethyl)-...)
Affinity DataIC50:  540nMAssay Description:Inhibition of Steroid 5-alpha-reductase type I from rat ventral prostate (RVP)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-oxo-5-alpha-steroid 4-dehydrogenase 2(Rattus norvegicus)
Saarland University

Curated by ChEMBL
LigandPNGBDBM50116417(4-(1-Diphenylcarbamoyl-piperidin-4-ylidenemethyl)-...)
Affinity DataIC50:  690nMAssay Description:Inhibition of Steroid 5-alpha-reductase type 2 of rat ventral prostate (RVP)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-oxo-5-alpha-steroid 4-dehydrogenase 1(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50116420(3-[1-(2,2-Dicyclohexyl-acetyl)-piperidin-4-ylidene...)
Affinity DataIC50:  700nMAssay Description:In vitro inhibitory activity against Steroid 5-alpha-reductase type 2 of human benign prostatic hyperplasia (BPH) tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-oxo-5-alpha-steroid 4-dehydrogenase 2(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50116417(4-(1-Diphenylcarbamoyl-piperidin-4-ylidenemethyl)-...)
Affinity DataIC50:  830nMAssay Description:Inhibition of Steroid 5-alpha-reductase type 2 from human benign prostatic hyperplasia (BPH) tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-oxo-5-alpha-steroid 4-dehydrogenase 2(Rattus norvegicus)
Saarland University

Curated by ChEMBL
LigandPNGBDBM50116422(4-[1-(3,3-Diphenyl-propionyl)-piperidin-4-ylidenem...)
Affinity DataIC50:  880nMAssay Description:Inhibition of Steroid 5-alpha-reductase type 2 of rat ventral prostate (RVP)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-oxo-5-alpha-steroid 4-dehydrogenase 2(Rattus norvegicus)
Saarland University

Curated by ChEMBL
LigandPNGBDBM50116428(4-(1-Diphenylacetyl-piperidin-4-ylidenemethyl)-3-m...)
Affinity DataIC50:  940nMAssay Description:Inhibition of Steroid 5-alpha-reductase type 2 of rat ventral prostate (RVP)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-oxo-5-alpha-steroid 4-dehydrogenase 1(Rattus norvegicus)
Saarland University

Curated by ChEMBL
LigandPNGBDBM50116432(4-(1-Diphenylacetyl-piperidin-4-ylidenemethyl)-3-f...)
Affinity DataIC50:  1.10E+3nMAssay Description:Inhibition of Steroid 5-alpha-reductase type I from rat ventral prostate (RVP)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-oxo-5-alpha-steroid 4-dehydrogenase 2(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50116422(4-[1-(3,3-Diphenyl-propionyl)-piperidin-4-ylidenem...)
Affinity DataIC50:  1.10E+3nMAssay Description:Inhibition of Steroid 5-alpha-reductase type 2 from human benign prostatic hyperplasia (BPH) tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-oxo-5-alpha-steroid 4-dehydrogenase 2(Rattus norvegicus)
Saarland University

Curated by ChEMBL
LigandPNGBDBM50116432(4-(1-Diphenylacetyl-piperidin-4-ylidenemethyl)-3-f...)
Affinity DataIC50:  1.10E+3nMAssay Description:Inhibition of Steroid 5-alpha-reductase type 2 of rat ventral prostate (RVP)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-oxo-5-alpha-steroid 4-dehydrogenase 2(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50116430(4-[1-(Adamantane-1-carbonyl)-piperidin-4-ylideneme...)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibition of Steroid 5-alpha-reductase type 2 from human benign prostatic hyperplasia (BPH) tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-oxo-5-alpha-steroid 4-dehydrogenase 1(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50116425(4-(1-Diphenylacetyl-piperidin-4-yloxy)-benzoic aci...)
Affinity DataIC50:  1.30E+3nMAssay Description:In vitro inhibitory activity against Steroid 5-alpha-reductase type 2 of human benign prostatic hyperplasia (BPH) tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-oxo-5-alpha-steroid 4-dehydrogenase 1(Rattus norvegicus)
Saarland University

Curated by ChEMBL
LigandPNGBDBM50116422(4-[1-(3,3-Diphenyl-propionyl)-piperidin-4-ylidenem...)
Affinity DataIC50:  1.60E+3nMAssay Description:Inhibition of Steroid 5-alpha-reductase type I from rat ventral prostate (RVP)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-oxo-5-alpha-steroid 4-dehydrogenase 1(Rattus norvegicus)
Saarland University

Curated by ChEMBL
LigandPNGBDBM50116419(4-[1-(2,2-Dicyclohexyl-acetyl)-piperidin-4-ylidene...)
Affinity DataIC50:  1.80E+3nMAssay Description:In vitro inhibitory activity against steroid Steroid 5-alpha-reductase type I of rat ventral prostate (RVP)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-oxo-5-alpha-steroid 4-dehydrogenase 1(Rattus norvegicus)
Saarland University

Curated by ChEMBL
LigandPNGBDBM50116428(4-(1-Diphenylacetyl-piperidin-4-ylidenemethyl)-3-m...)
Affinity DataIC50:  1.90E+3nMAssay Description:Inhibition of Steroid 5-alpha-reductase type I from rat ventral prostate (RVP)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-oxo-5-alpha-steroid 4-dehydrogenase 2(Rattus norvegicus)
Saarland University

Curated by ChEMBL
LigandPNGBDBM50116426(4-[1-(Adamantane-1-carbonyl)-piperidin-4-ylideneme...)
Affinity DataIC50:  2.50E+3nMAssay Description:Inhibition of Steroid 5-alpha-reductase type 2 of rat ventral prostate (RVP)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-oxo-5-alpha-steroid 4-dehydrogenase 1(Rattus norvegicus)
Saarland University

Curated by ChEMBL
LigandPNGBDBM50116416(4-[1-(Adamantane-1-carbonyl)-piperidin-4-ylideneme...)
Affinity DataIC50:  2.70E+3nMAssay Description:Inhibition of Steroid 5-alpha-reductase type I from rat ventral prostate (RVP)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-oxo-5-alpha-steroid 4-dehydrogenase 2(Rattus norvegicus)
Saarland University

Curated by ChEMBL
LigandPNGBDBM50116419(4-[1-(2,2-Dicyclohexyl-acetyl)-piperidin-4-ylidene...)
Affinity DataIC50:  3.00E+3nMAssay Description:Inhibition of Steroid 5-alpha-reductase type 2 of rat ventral prostate (RVP)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-oxo-5-alpha-steroid 4-dehydrogenase 1(Rattus norvegicus)
Saarland University

Curated by ChEMBL
LigandPNGBDBM50116424(CHEMBL115438 | {4-[1-(2,2-Dicyclohexyl-acetyl)-pip...)
Affinity DataIC50:  3.20E+3nMAssay Description:Inhibition of Steroid 5-alpha-reductase type I from rat ventral prostate (RVP)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-oxo-5-alpha-steroid 4-dehydrogenase 1(Rattus norvegicus)
Saarland University

Curated by ChEMBL
LigandPNGBDBM50116423(4-(1-Diphenylacetyl-piperidin-4-ylidenemethyl)-ben...)
Affinity DataIC50:  3.40E+3nMAssay Description:Inhibition of Steroid 5-alpha-reductase type I from rat ventral prostate (RVP)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-oxo-5-alpha-steroid 4-dehydrogenase 2(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50116428(4-(1-Diphenylacetyl-piperidin-4-ylidenemethyl)-3-m...)
Affinity DataIC50:  3.50E+3nMAssay Description:Inhibition of Steroid 5-alpha-reductase type 2 from human benign prostatic hyperplasia (BPH) tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-oxo-5-alpha-steroid 4-dehydrogenase 2(Rattus norvegicus)
Saarland University

Curated by ChEMBL
LigandPNGBDBM50116416(4-[1-(Adamantane-1-carbonyl)-piperidin-4-ylideneme...)
Affinity DataIC50:  3.50E+3nMAssay Description:Inhibition of Steroid 5-alpha-reductase type 2 of rat ventral prostate (RVP)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-oxo-5-alpha-steroid 4-dehydrogenase 1(Rattus norvegicus)
Saarland University

Curated by ChEMBL
LigandPNGBDBM50116418(CHEMBL323856 | [4-(1-Diphenylacetyl-piperidin-4-yl...)
Affinity DataIC50:  4.50E+3nMAssay Description:Inhibition of Steroid 5-alpha-reductase type I from rat ventral prostate (RVP)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-oxo-5-alpha-steroid 4-dehydrogenase 1(Rattus norvegicus)
Saarland University

Curated by ChEMBL
LigandPNGBDBM50116426(4-[1-(Adamantane-1-carbonyl)-piperidin-4-ylideneme...)
Affinity DataIC50:  5.60E+3nMAssay Description:Inhibition of Steroid 5-alpha-reductase type I from rat ventral prostate (RVP)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed