Compile Data Set for Download or QSAR
maximum 50k data
Found 51 with Last Name = 'benito' and Initial = 's'
TargetAdenosine receptor A2b(Homo sapiens (Human))
Almirall

Curated by ChEMBL
LigandPNGBDBM50211682(5-{[4'-(2-furyl)-4,5'-bipyrimidin-2'-yl]amino}pyri...)
Affinity DataKi:  16nMAssay Description:Displacement of [3H]DPCPX from human A2B receptor expressed in HEK293 cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Almirall

Curated by ChEMBL
LigandPNGBDBM50211685(4'-(2-furyl)-N-pyridin-3-yl-4,5'-bipyrimidin-2'-am...)
Affinity DataKi:  17nMAssay Description:Displacement of [3H]DPCPX from human A2B receptor expressed in HEK293 cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Almirall

Curated by ChEMBL
LigandPNGBDBM50211680(4'-(2-furyl)-N-pyrimidin-5-yl-4,5'-bipyrimidin-2'-...)
Affinity DataKi:  24nMAssay Description:Displacement of [3H]DPCPX from human A2B receptor expressed in HEK293 cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Almirall

Curated by ChEMBL
LigandPNGBDBM50211688(5-{[4'-(2-furyl)-4,5'-bipyrimidin-2'-yl]amino}-1-m...)
Affinity DataKi:  28nMAssay Description:Displacement of [3H]DPCPX from human A2B receptor expressed in HEK293 cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Almirall

Curated by ChEMBL
LigandPNGBDBM50211679(4'-(2-furyl)-N-(1-oxidopyridin-3-yl)-4,5'-bipyrimi...)
Affinity DataKi:  34nMAssay Description:Displacement of [3H]DPCPX from human A2B receptor expressed in HEK293 cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Almirall

Curated by ChEMBL
LigandPNGBDBM50211684(4'-(2-furyl)-N-(2-methoxypyrimidin-5-yl)-4,5'-bipy...)
Affinity DataKi:  39nMAssay Description:Displacement of [3H]DPCPX from human A2B receptor expressed in HEK293 cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Almirall

Curated by ChEMBL
LigandPNGBDBM50211687(5-{[4'-(2-furyl)-4,5'-bipyrimidin-2'-yl]amino}nico...)
Affinity DataKi:  69nMAssay Description:Displacement of [3H]DPCPX from human A2B receptor expressed in HEK293 cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Almirall

Curated by ChEMBL
LigandPNGBDBM50211681(4'-(2-furyl)-N-(6-methoxypyridin-3-yl)-4,5'-bipyri...)
Affinity DataKi:  115nMAssay Description:Displacement of [3H]DPCPX from human A2B receptor expressed in HEK293 cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Almirall

Curated by ChEMBL
LigandPNGBDBM50211686(4'-(2-furyl)-N-pyrazin-2-yl-4,5'-bipyrimidin-2'-am...)
Affinity DataKi:  116nMAssay Description:Displacement of [3H]DPCPX from human A2B receptor expressed in HEK293 cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Almirall

Curated by ChEMBL
LigandPNGBDBM50211683(1-(cyclopropylmethyl)-5-{[4'-(2-furyl)-4,5'-bipyri...)
Affinity DataKi:  119nMAssay Description:Displacement of [3H]DPCPX from human A2B receptor expressed in HEK293 cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Instituto De Qu£Mica M£Dica

Curated by ChEMBL
LigandPNGBDBM50078147(CHEMBL3417564)
Affinity DataKi:  398nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor transfected in HEK293 cells after 90 mins by liquid scintillation spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Instituto De Qu£Mica M£Dica

Curated by ChEMBL
LigandPNGBDBM50078149(CHEMBL3417566)
Affinity DataKi:  529nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor transfected in HEK293 cells after 90 mins by liquid scintillation spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Instituto De Qu£Mica M£Dica

Curated by ChEMBL
LigandPNGBDBM50078148(CHEMBL3417565)
Affinity DataKi:  597nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor transfected in HEK293 cells after 90 mins by liquid scintillation spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Almirall

Curated by ChEMBL
LigandPNGBDBM50211685(4'-(2-furyl)-N-pyridin-3-yl-4,5'-bipyrimidin-2'-am...)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]DPCPX from human A1 receptor expressed in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Almirall

Curated by ChEMBL
LigandPNGBDBM50211682(5-{[4'-(2-furyl)-4,5'-bipyrimidin-2'-yl]amino}pyri...)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [2H]NECA from human A3 receptor expressed in HeLa cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Almirall

Curated by ChEMBL
LigandPNGBDBM50211687(5-{[4'-(2-furyl)-4,5'-bipyrimidin-2'-yl]amino}nico...)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [2H]NECA from human A3 receptor expressed in HeLa cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Almirall

Curated by ChEMBL
LigandPNGBDBM50211688(5-{[4'-(2-furyl)-4,5'-bipyrimidin-2'-yl]amino}-1-m...)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [2H]NECA from human A3 receptor expressed in HeLa cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Almirall

Curated by ChEMBL
LigandPNGBDBM50211685(4'-(2-furyl)-N-pyridin-3-yl-4,5'-bipyrimidin-2'-am...)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [2H]NECA from human A3 receptor expressed in HeLa cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Almirall

Curated by ChEMBL
LigandPNGBDBM50211681(4'-(2-furyl)-N-(6-methoxypyridin-3-yl)-4,5'-bipyri...)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [2H]NECA from human A3 receptor expressed in HeLa cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Almirall

Curated by ChEMBL
LigandPNGBDBM50211683(1-(cyclopropylmethyl)-5-{[4'-(2-furyl)-4,5'-bipyri...)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [2H]NECA from human A3 receptor expressed in HeLa cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Almirall

Curated by ChEMBL
LigandPNGBDBM50211679(4'-(2-furyl)-N-(1-oxidopyridin-3-yl)-4,5'-bipyrimi...)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [2H]NECA from human A3 receptor expressed in HeLa cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Almirall

Curated by ChEMBL
LigandPNGBDBM50211680(4'-(2-furyl)-N-pyrimidin-5-yl-4,5'-bipyrimidin-2'-...)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [2H]NECA from human A3 receptor expressed in HeLa cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Almirall

Curated by ChEMBL
LigandPNGBDBM50211684(4'-(2-furyl)-N-(2-methoxypyrimidin-5-yl)-4,5'-bipy...)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [2H]NECA from human A3 receptor expressed in HeLa cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Almirall

Curated by ChEMBL
LigandPNGBDBM50211686(4'-(2-furyl)-N-pyrazin-2-yl-4,5'-bipyrimidin-2'-am...)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [2H]NECA from human A3 receptor expressed in HeLa cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Almirall

Curated by ChEMBL
LigandPNGBDBM50211682(5-{[4'-(2-furyl)-4,5'-bipyrimidin-2'-yl]amino}pyri...)
Affinity DataKi: >2.50E+3nMAssay Description:Displacement of [3H]ZM241385 from human A2A receptor expressed in HeLa cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Almirall

Curated by ChEMBL
LigandPNGBDBM50211687(5-{[4'-(2-furyl)-4,5'-bipyrimidin-2'-yl]amino}nico...)
Affinity DataKi: >2.50E+3nMAssay Description:Displacement of [3H]ZM241385 from human A2A receptor expressed in HeLa cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Almirall

Curated by ChEMBL
LigandPNGBDBM50211683(1-(cyclopropylmethyl)-5-{[4'-(2-furyl)-4,5'-bipyri...)
Affinity DataKi: >2.50E+3nMAssay Description:Displacement of [3H]ZM241385 from human A2A receptor expressed in HeLa cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Almirall

Curated by ChEMBL
LigandPNGBDBM50211681(4'-(2-furyl)-N-(6-methoxypyridin-3-yl)-4,5'-bipyri...)
Affinity DataKi: >2.50E+3nMAssay Description:Displacement of [3H]ZM241385 from human A2A receptor expressed in HeLa cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Almirall

Curated by ChEMBL
LigandPNGBDBM50211684(4'-(2-furyl)-N-(2-methoxypyrimidin-5-yl)-4,5'-bipy...)
Affinity DataKi: >2.50E+3nMAssay Description:Displacement of [3H]ZM241385 from human A2A receptor expressed in HeLa cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Almirall

Curated by ChEMBL
LigandPNGBDBM50211680(4'-(2-furyl)-N-pyrimidin-5-yl-4,5'-bipyrimidin-2'-...)
Affinity DataKi: >2.50E+3nMAssay Description:Displacement of [3H]ZM241385 from human A2A receptor expressed in HeLa cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Almirall

Curated by ChEMBL
LigandPNGBDBM50211685(4'-(2-furyl)-N-pyridin-3-yl-4,5'-bipyrimidin-2'-am...)
Affinity DataKi: >2.50E+3nMAssay Description:Displacement of [3H]ZM241385 from human A2A receptor expressed in HeLa cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Almirall

Curated by ChEMBL
LigandPNGBDBM50211679(4'-(2-furyl)-N-(1-oxidopyridin-3-yl)-4,5'-bipyrimi...)
Affinity DataKi: >2.50E+3nMAssay Description:Displacement of [3H]ZM241385 from human A2A receptor expressed in HeLa cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Almirall

Curated by ChEMBL
LigandPNGBDBM50211688(5-{[4'-(2-furyl)-4,5'-bipyrimidin-2'-yl]amino}-1-m...)
Affinity DataKi: >2.50E+3nMAssay Description:Displacement of [3H]ZM241385 from human A2A receptor expressed in HeLa cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Almirall

Curated by ChEMBL
LigandPNGBDBM50211686(4'-(2-furyl)-N-pyrazin-2-yl-4,5'-bipyrimidin-2'-am...)
Affinity DataKi: >2.50E+3nMAssay Description:Displacement of [3H]ZM241385 from human A2A receptor expressed in HeLa cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Almirall

Curated by ChEMBL
LigandPNGBDBM50211683(1-(cyclopropylmethyl)-5-{[4'-(2-furyl)-4,5'-bipyri...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]DPCPX from human A1 receptor expressed in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Almirall

Curated by ChEMBL
LigandPNGBDBM50211681(4'-(2-furyl)-N-(6-methoxypyridin-3-yl)-4,5'-bipyri...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]DPCPX from human A1 receptor expressed in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Almirall

Curated by ChEMBL
LigandPNGBDBM50211687(5-{[4'-(2-furyl)-4,5'-bipyrimidin-2'-yl]amino}nico...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]DPCPX from human A1 receptor expressed in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Almirall

Curated by ChEMBL
LigandPNGBDBM50211679(4'-(2-furyl)-N-(1-oxidopyridin-3-yl)-4,5'-bipyrimi...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]DPCPX from human A1 receptor expressed in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Almirall

Curated by ChEMBL
LigandPNGBDBM50211688(5-{[4'-(2-furyl)-4,5'-bipyrimidin-2'-yl]amino}-1-m...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]DPCPX from human A1 receptor expressed in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Almirall

Curated by ChEMBL
LigandPNGBDBM50211682(5-{[4'-(2-furyl)-4,5'-bipyrimidin-2'-yl]amino}pyri...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]DPCPX from human A1 receptor expressed in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Almirall

Curated by ChEMBL
LigandPNGBDBM50211686(4'-(2-furyl)-N-pyrazin-2-yl-4,5'-bipyrimidin-2'-am...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]DPCPX from human A1 receptor expressed in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Almirall

Curated by ChEMBL
LigandPNGBDBM50211680(4'-(2-furyl)-N-pyrimidin-5-yl-4,5'-bipyrimidin-2'-...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]DPCPX from human A1 receptor expressed in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Almirall

Curated by ChEMBL
LigandPNGBDBM50211680(4'-(2-furyl)-N-pyrimidin-5-yl-4,5'-bipyrimidin-2'-...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]DPCPX from human A1 receptor expressed in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Almirall

Curated by ChEMBL
LigandPNGBDBM50211684(4'-(2-furyl)-N-(2-methoxypyrimidin-5-yl)-4,5'-bipy...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]DPCPX from human A1 receptor expressed in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Instituto De Qu£Mica M£Dica

Curated by ChEMBL
LigandPNGBDBM50078149(CHEMBL3417566)
Affinity DataKi: >4.00E+4nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor transfected in HEK293 cells after 90 mins by liquid scintillation spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Instituto De Qu£Mica M£Dica

Curated by ChEMBL
LigandPNGBDBM50078148(CHEMBL3417565)
Affinity DataKi: >4.00E+4nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor transfected in HEK293 cells after 90 mins by liquid scintillation spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Instituto De Qu£Mica M£Dica

Curated by ChEMBL
LigandPNGBDBM50078147(CHEMBL3417564)
Affinity DataKi: >4.00E+4nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor transfected in HEK293 cells after 90 mins by liquid scintillation spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Almirall

Curated by ChEMBL
LigandPNGBDBM50211685(4'-(2-furyl)-N-pyridin-3-yl-4,5'-bipyrimidin-2'-am...)
Affinity DataIC50:  321nMAssay Description:Activity at human A2B receptor expressed in HEK293 cells assessed as inhibition of NECA-induced intracellular cAMP levels by ELISAChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Almirall

Curated by ChEMBL
LigandPNGBDBM50211685(4'-(2-furyl)-N-pyridin-3-yl-4,5'-bipyrimidin-2'-am...)
Affinity DataIC50:  340nMAssay Description:Inhibition of NECA-induced IL6 production in human fibroblast after 24 hrs by ELISAChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Mus musculus)
Almirall

Curated by ChEMBL
LigandPNGBDBM50211685(4'-(2-furyl)-N-pyridin-3-yl-4,5'-bipyrimidin-2'-am...)
Affinity DataIC50:  349nMAssay Description:Activity at mouse A2B receptor expressed in CHO cells assessed as inhibition of NECA-induced intracellular cAMP levels by ELISAChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Displayed 1 to 50 (of 51 total ) | Next | Last >>
Jump to: