Affinity DataIC50: 15nMAssay Description:Binding affinity of the compound against human melanocortin 4 receptor (hMC4R) using [125I]- agouti related protein (AGRP) as radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 16nMAssay Description:Inhibitory activity of the compound against hMC3R (human melanocortin receptor) using I-AGRP as radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 19nMAssay Description:Binding affinity of the compound against human melanocortin 4 receptor (hMC4R) using [125I]- NDP-MSH as radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 1.90E+3nMAssay Description:Binding affinity of the compound against human melanocortin 4 receptor (hMC4R) using [125I]- ([Nle4]alpha-MSH) as radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 1.90E+3nMAssay Description:Binding affinity of the compound against human melanocortin 4 receptor (hMC4R) using [125I]- agouti related protein (AGRP) as radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 2.10E+3nMAssay Description:Inhibitory activity of the compound against hMC4R (human melanocortin receptor) using I-AGRP as radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 3.10E+3nMAssay Description:Binding affinity of the compound against human melanocortin 4 receptor (hMC4R) using [125I]- ([Nle4]alpha-MSH) as radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 3.10E+3nMAssay Description:Binding affinity of the compound against human melanocortin 4 receptor (hMC4R) using [125I]- ([Nle4]alpha-MSH) as radioligandMore data for this Ligand-Target Pair
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
University Of California
Curated by ChEMBL
University Of California
Curated by ChEMBL
Affinity DataIC50: 9.10E+3nMAssay Description:Inhibitory activity of the compound against hMC1R (human melanocortin receptor) using [125I]-[Nle4] alpha-MSH as radioligandMore data for this Ligand-Target Pair
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
University Of California
Curated by ChEMBL
University Of California
Curated by ChEMBL
Affinity DataIC50: 2.50E+4nMAssay Description:Inhibitory activity of the compound against hMC1R (human melanocortin receptor) using [125I]- ASIP Y radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 4.80E+4nMAssay Description:Inhibitory activity of the compound against hMC3R (human melanocortin receptor) using [125I]-[Nle4] alpha-MSH as radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibitory activity of the compound against hMC4R (human melanocortin receptor) using [125I]-[Nle4] alpha-MSH as radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+5nMAssay Description:Binding affinity of the compound against human melanocortin 4 receptor (hMC4R) using [125I]- NDP-MSH as radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+5nMAssay Description:Binding affinity of the compound against human melanocortin 4 receptor (hMC4R) using [125I]- ([Nle4]alpha-MSH) as radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+5nMAssay Description:Binding affinity of the compound against human melanocortin 4 receptor (hMC4R) using [125I]- agouti related protein (AGRP) as radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+5nMAssay Description:Binding affinity of the compound against human melanocortin 4 receptor (hMC4R) using [125I]- ([Nle4]alpha-MSH) as radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+5nMAssay Description:Binding affinity of the compound against human melanocortin 4 receptor (hMC4R) using [125I]- agouti related protein (AGRP) as radioligandMore data for this Ligand-Target Pair