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Found 17 with Last Name = 'chai' and Initial = 'bx'
TargetMelanocortin receptor 4(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50126395(Ac-Ser-Tyr-Ser-Nle-Glu-His-Phe-Arg-Trp-Gly-Lys-Pro...)
Affinity DataIC50:  15nMAssay Description:Binding affinity of the compound against human melanocortin 4 receptor (hMC4R) using [125I]- agouti related protein (AGRP) as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50126395(Ac-Ser-Tyr-Ser-Nle-Glu-His-Phe-Arg-Trp-Gly-Lys-Pro...)
Affinity DataIC50:  16nMAssay Description:Inhibitory activity of the compound against hMC3R (human melanocortin receptor) using I-AGRP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50126395(Ac-Ser-Tyr-Ser-Nle-Glu-His-Phe-Arg-Trp-Gly-Lys-Pro...)
Affinity DataIC50:  19nMAssay Description:Binding affinity of the compound against human melanocortin 4 receptor (hMC4R) using [125I]- NDP-MSH as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50126393(CHEMBL417853 | N-Benzhydryl-N-{[carbamoylmethyl-((...)
Affinity DataIC50:  1.90E+3nMAssay Description:Binding affinity of the compound against human melanocortin 4 receptor (hMC4R) using [125I]- ([Nle4]alpha-MSH) as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50126393(CHEMBL417853 | N-Benzhydryl-N-{[carbamoylmethyl-((...)
Affinity DataIC50:  1.90E+3nMAssay Description:Binding affinity of the compound against human melanocortin 4 receptor (hMC4R) using [125I]- agouti related protein (AGRP) as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50126393(CHEMBL417853 | N-Benzhydryl-N-{[carbamoylmethyl-((...)
Affinity DataIC50:  2.10E+3nMAssay Description:Inhibitory activity of the compound against hMC4R (human melanocortin receptor) using I-AGRP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50126393(CHEMBL417853 | N-Benzhydryl-N-{[carbamoylmethyl-((...)
Affinity DataIC50:  3.10E+3nMAssay Description:Binding affinity of the compound against human melanocortin 4 receptor (hMC4R) using [125I]- ([Nle4]alpha-MSH) as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50126393(CHEMBL417853 | N-Benzhydryl-N-{[carbamoylmethyl-((...)
Affinity DataIC50:  3.10E+3nMAssay Description:Binding affinity of the compound against human melanocortin 4 receptor (hMC4R) using [125I]- ([Nle4]alpha-MSH) as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50126393(CHEMBL417853 | N-Benzhydryl-N-{[carbamoylmethyl-((...)
Affinity DataIC50:  9.10E+3nMAssay Description:Inhibitory activity of the compound against hMC1R (human melanocortin receptor) using [125I]-[Nle4] alpha-MSH as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50126393(CHEMBL417853 | N-Benzhydryl-N-{[carbamoylmethyl-((...)
Affinity DataIC50:  2.50E+4nMAssay Description:Inhibitory activity of the compound against hMC1R (human melanocortin receptor) using [125I]- ASIP Y radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 3(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50126393(CHEMBL417853 | N-Benzhydryl-N-{[carbamoylmethyl-((...)
Affinity DataIC50:  4.80E+4nMAssay Description:Inhibitory activity of the compound against hMC3R (human melanocortin receptor) using [125I]-[Nle4] alpha-MSH as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 3(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50126393(CHEMBL417853 | N-Benzhydryl-N-{[carbamoylmethyl-((...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibitory activity of the compound against hMC4R (human melanocortin receptor) using [125I]-[Nle4] alpha-MSH as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50126396(CHEMBL30677 | N-Benzyl-N-{[carbamoylmethyl-((R)-1-...)
Affinity DataIC50: >1.00E+5nMAssay Description:Binding affinity of the compound against human melanocortin 4 receptor (hMC4R) using [125I]- NDP-MSH as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50126394(CHEMBL440102 | N-Benzyl-N-[(benzyl-carbamoylmethyl...)
Affinity DataIC50: >1.00E+5nMAssay Description:Binding affinity of the compound against human melanocortin 4 receptor (hMC4R) using [125I]- ([Nle4]alpha-MSH) as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50126394(CHEMBL440102 | N-Benzyl-N-[(benzyl-carbamoylmethyl...)
Affinity DataIC50: >1.00E+5nMAssay Description:Binding affinity of the compound against human melanocortin 4 receptor (hMC4R) using [125I]- agouti related protein (AGRP) as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50126397(2-[Benzyl-(2-{[2-(3-guanidino-propylamino)-acetyl]...)
Affinity DataIC50: >1.00E+5nMAssay Description:Binding affinity of the compound against human melanocortin 4 receptor (hMC4R) using [125I]- ([Nle4]alpha-MSH) as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50126396(CHEMBL30677 | N-Benzyl-N-{[carbamoylmethyl-((R)-1-...)
Affinity DataIC50: >1.00E+5nMAssay Description:Binding affinity of the compound against human melanocortin 4 receptor (hMC4R) using [125I]- agouti related protein (AGRP) as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed