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Found 109 with Last Name = 'jolibois' and Initial = 'k'
TargetSqualene synthase(Rattus norvegicus)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50031845((4-Biphenyl-4-yl-1-phosphono-butyl)-phosphonic aci...)
Affinity DataIC50:  0.700nMAssay Description:Inhibitory activity against rat liver microsomal squalene synthase was determined using [3H]-FPP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSqualene synthase(Rattus norvegicus)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50031845((4-Biphenyl-4-yl-1-phosphono-butyl)-phosphonic aci...)
Affinity DataIC50:  0.700nMAssay Description:Inhibition rat liver microsomal squalene synthaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSqualene synthase(Rattus norvegicus)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50049232(CHEMBL348349 | Tetrasodium salt of 4-(4'-Methyl-bi...)
Affinity DataIC50:  1nMAssay Description:Inhibitory activity against rat liver microsomal squalene synthase was determined using [3H]-FPP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSqualene synthase(Rattus norvegicus)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50031839(((E)-6,10-Dimethyl-1-phosphono-undeca-5,9-dienyl)-...)
Affinity DataIC50:  1nMAssay Description:Inhibition rat liver microsomal squalene synthaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSqualene synthase(Rattus norvegicus)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50031843(((E)-8,12-Dimethyl-1-phosphono-trideca-7,11-dienyl...)
Affinity DataIC50:  2.5nMAssay Description:Inhibition rat liver microsomal squalene synthaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSqualene synthase(Rattus norvegicus)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50031848(((E)-7,11-Dimethyl-1-phosphono-dodeca-6,10-dienyl)...)
Affinity DataIC50:  2.60nMAssay Description:Inhibition rat liver microsomal squalene synthaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMicrosomal triglyceride transfer protein large subunit(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50153193(CHEMBL186836 | Trans-9-{4-[5-(2-Benzooxazol-2-yl-b...)
Affinity DataIC50:  3nMAssay Description:In vitro inhibitory concentration against human Microsomal triglyceride transfer proteinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSqualene synthase(Rattus norvegicus)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50031844(((E)-1-Hydroxyphosphinoyl-6,10-dimethyl-undeca-5,9...)
Affinity DataIC50:  4nMAssay Description:Inhibition rat liver microsomal squalene synthaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSqualene synthase(Rattus norvegicus)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50031851(((E)-10,14-Dimethyl-1-phosphono-pentadeca-9,13-die...)
Affinity DataIC50:  4.20nMAssay Description:Inhibition rat liver microsomal squalene synthaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSqualene synthase(Rattus norvegicus)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50031842(CHEMBL86867 | [(5E,9E)-1-(Hydroxy-hydroxymethyl-ph...)
Affinity DataIC50:  4.70nMAssay Description:Inhibition rat liver microsomal squalene synthaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMicrosomal triglyceride transfer protein large subunit(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50153191(9-(4-{1-Oxy-4-[(4''-trifluoromethyl-biphenyl-2-car...)
Affinity DataIC50:  5nMAssay Description:In vitro inhibitory concentration against human Microsomal triglyceride transfer proteinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSqualene synthase(Rattus norvegicus)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50049227(CHEMBL158707 | Trisodium salt of [1-(Dimethoxy-pho...)
Affinity DataIC50:  5.70nMAssay Description:Inhibitory activity against rat liver microsomal squalene synthase was determined using [3H]-FPP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSqualene synthase(Rattus norvegicus)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50031847(((5E,9E)-6,10,14-Trimethyl-1-phosphono-pentadeca-5...)
Affinity DataIC50:  5.70nMAssay Description:Inhibition rat liver microsomal squalene synthaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSqualene synthase(Rattus norvegicus)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50031832(CHEMBL87922 | [(6E,10E)-1-(Hydroxy-methyl-phosphin...)
Affinity DataIC50:  6.5nMAssay Description:Inhibition rat liver microsomal squalene synthaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSqualene synthase(Rattus norvegicus)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50031859(CHEMBL314797 | [(5E,9E)-1-(Hydroxy-methoxymethyl-p...)
Affinity DataIC50:  6.5nMAssay Description:Inhibition rat liver microsomal squalene synthaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMicrosomal triglyceride transfer protein large subunit(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50153189(CHEMBL365687 | Cis-9-(4-{2-Oxo-5-[(4''-trifluorome...)
Affinity DataIC50:  7nMAssay Description:In vitro inhibitory concentration against human Microsomal triglyceride transfer proteinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMicrosomal triglyceride transfer protein large subunit(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50153189(CHEMBL365687 | Cis-9-(4-{2-Oxo-5-[(4''-trifluorome...)
Affinity DataIC50:  7nMAssay Description:In vitro inhibitory concentration against human Microsomal triglyceride transfer proteinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMicrosomal triglyceride transfer protein large subunit(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50098320(9-(4-{4-[(4''-Trifluoromethyl-biphenyl-2-carbonyl)...)
Affinity DataIC50:  8nMAssay Description:In vitro inhibitory concentration against human Microsomal triglyceride transfer proteinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetSqualene synthase(Rattus norvegicus)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50031862(CHEMBL84629 | [(E)-1-(Hydroxy-methyl-phosphinoyl)-...)
Affinity DataIC50:  8.70nMAssay Description:Inhibition rat liver microsomal squalene synthaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMicrosomal triglyceride transfer protein large subunit(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50153195(CHEMBL186494 | Trans-9-{4-[5-(2-Benzothiazol-2-yl-...)
Affinity DataIC50:  9nMAssay Description:In vitro inhibitory concentration against human Microsomal triglyceride transfer proteinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMicrosomal triglyceride transfer protein large subunit(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50153188(CHEMBL360146 | Trans-1-Phenyl-piperidine-2-carboxy...)
Affinity DataIC50:  9nMAssay Description:In vitro inhibitory concentration against human Microsomal triglyceride transfer proteinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMicrosomal triglyceride transfer protein large subunit(Bos taurus)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50126193(CHEMBL27660 | {4-[9-(2,2,2-Trifluoro-ethylcarbamoy...)
Affinity DataIC50:  11nMAssay Description:Inhibitory activity against microsomal triglyceride transfer protein (MTP)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMicrosomal triglyceride transfer protein large subunit(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50153190(CHEMBL185866 | Trans-9-[4-(5-Benzoylamino-2-oxo-2l...)
Affinity DataIC50:  11nMAssay Description:In vitro inhibitory concentration against human Microsomal triglyceride transfer proteinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSqualene synthase(Rattus norvegicus)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50031836(((8E,12E)-9,13,17-Trimethyl-1-phosphono-octadeca-8...)
Affinity DataIC50:  11.8nMAssay Description:Inhibition rat liver microsomal squalene synthaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMicrosomal triglyceride transfer protein large subunit(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50153196(CHEMBL187076 | Trans-9-{4-[5-(2-Morpholin-4-yl-ben...)
Affinity DataIC50:  12nMAssay Description:In vitro inhibitory concentration against human Microsomal triglyceride transfer proteinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSqualene synthase(Rattus norvegicus)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50031849(CHEMBL86918 | [(5E,9E)-1-(Hydroxy-methyl-phosphino...)
Affinity DataIC50:  12.9nMAssay Description:Inhibition rat liver microsomal squalene synthaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSqualene synthase(Rattus norvegicus)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50049217(CHEMBL158517 | Tripotassium salt of 1-Phosphono-4-...)
Affinity DataIC50:  13nMAssay Description:Inhibitory activity against rat liver microsomal squalene synthase was determined using [3H]-FPP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSqualene synthase(Rattus norvegicus)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50031837(CHEMBL87489 | [(E)-1-(Hydroxy-methoxymethyl-phosph...)
Affinity DataIC50:  13.1nMAssay Description:Inhibition rat liver microsomal squalene synthaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMicrosomal triglyceride transfer protein large subunit(Bos taurus)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50126188(CHEMBL28348 | [4-(9-Propylcarbamoyl-9H-fluoren-9-y...)
Affinity DataIC50:  14nMAssay Description:Inhibitory activity against microsomal triglyceride transfer protein (MTP)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMicrosomal triglyceride transfer protein large subunit(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50153194(CHEMBL187696 | Cis-(2-Oxo-2-{4-[9-(2,2,2-trifluoro...)
Affinity DataIC50:  14nMAssay Description:In vitro inhibitory concentration against human Microsomal triglyceride transfer proteinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSqualene synthase(Rattus norvegicus)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50031840(CHEMBL84961 | [4-Biphenyl-4-yl-1-(hydroxy-methoxym...)
Affinity DataIC50:  14.8nMAssay Description:Inhibition rat liver microsomal squalene synthaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSqualene synthase(Rattus norvegicus)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50049233(CHEMBL160240 | Tripotassium salt of 4-Biphenyl-4-y...)
Affinity DataIC50:  15nMAssay Description:Inhibitory activity against rat liver microsomal squalene synthase was determined using [3H]-FPP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSqualene synthase(Rattus norvegicus)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50049230(CHEMBL160267 | Tripotassium salt of 4-{3-[2-(4-Met...)
Affinity DataIC50:  17nMAssay Description:Inhibitory activity against rat liver microsomal squalene synthase was determined using [3H]-FPP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSqualene synthase(Rattus norvegicus)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50031854(((E)-9,13-Dimethyl-1-phosphono-tetradeca-8,12-dien...)
Affinity DataIC50:  17.6nMAssay Description:Inhibition rat liver microsomal squalene synthaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSqualene synthase(Rattus norvegicus)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50049215(1-Phosphono-4-[3-(2-benzylphenoxy)phenyl]butylsulf...)
Affinity DataIC50:  18nMAssay Description:Inhibitory activity against rat liver microsomal squalene synthase was determined using [3H]-FPP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSqualene synthase(Rattus norvegicus)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50049228(CHEMBL158448 | Tripotassium salt of 4-{3-[2-(3-Met...)
Affinity DataIC50:  19nMAssay Description:Inhibitory activity against rat liver microsomal squalene synthase was determined using [3H]-FPP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMicrosomal triglyceride transfer protein large subunit(Bos taurus)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50126207((4-{9-[2-(4-Methoxy-phenyl)-ethylcarbamoyl]-9H-flu...)
Affinity DataIC50:  21nMAssay Description:Inhibitory activity against microsomal triglyceride transfer protein (MTP)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMicrosomal triglyceride transfer protein large subunit(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50126201(CHEMBL282785 | {4-[9-(2,2,2-Trifluoro-ethylcarbamo...)
Affinity DataIC50:  22nMAssay Description:In vitro inhibitory concentration against human Microsomal triglyceride transfer proteinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMicrosomal triglyceride transfer protein large subunit(Bos taurus)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50126201(CHEMBL282785 | {4-[9-(2,2,2-Trifluoro-ethylcarbamo...)
Affinity DataIC50:  22nMAssay Description:Inhibitory activity against microsomal triglyceride transfer protein (MTP)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMicrosomal triglyceride transfer protein large subunit(Bos taurus)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50126201(CHEMBL282785 | {4-[9-(2,2,2-Trifluoro-ethylcarbamo...)
Affinity DataIC50:  22nMAssay Description:Inhibitory activity against microsomal triglyceride transfer protein (MTP)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSqualene synthase(Rattus norvegicus)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50031855(CHEMBL86621 | [4-Biphenyl-4-yl-1-(hydroxy-hydroxym...)
Affinity DataIC50:  23.9nMAssay Description:Inhibition rat liver microsomal squalene synthaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMicrosomal triglyceride transfer protein large subunit(Bos taurus)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50126209(CHEMBL283897 | {4-[9-(2,2,2-Trifluoro-ethylcarbamo...)
Affinity DataIC50:  24nMAssay Description:Inhibitory activity against microsomal triglyceride transfer protein (MTP)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMicrosomal triglyceride transfer protein large subunit(Bos taurus)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50126225(CHEMBL26665 | {4-[9-(2,2,2-Trifluoro-ethylcarbamoy...)
Affinity DataIC50:  25nMAssay Description:Inhibitory activity against microsomal triglyceride transfer protein (MTP)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMicrosomal triglyceride transfer protein large subunit(Bos taurus)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50126212(CHEMBL280283 | {4-[9-(2,2,2-Trifluoro-ethylcarbamo...)
Affinity DataIC50:  27nMAssay Description:Inhibitory activity against microsomal triglyceride transfer protein (MTP)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSqualene synthase(Rattus norvegicus)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50031850(CHEMBL420416 | [(E)-1-(Hydroxy-methyl-phosphinoyl)...)
Affinity DataIC50:  30.7nMAssay Description:Inhibition rat liver microsomal squalene synthaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSqualene synthase(Rattus norvegicus)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50031853(((3E,7E)-4,8,12-Trimethyl-1-phosphono-trideca-3,7,...)
Affinity DataIC50:  32.4nMAssay Description:Inhibition rat liver microsomal squalene synthaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMicrosomal triglyceride transfer protein large subunit(Bos taurus)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50126223(CHEMBL282564 | {4-[9-(2,2,2-Trifluoro-ethylcarbamo...)
Affinity DataIC50:  33nMAssay Description:Inhibitory activity against microsomal triglyceride transfer protein (MTP)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSqualene synthase(Rattus norvegicus)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50049223(CHEMBL158851 | Tripotassium salt of4-[3-(2-Butyl-p...)
Affinity DataIC50:  35nMAssay Description:Inhibitory activity against rat liver microsomal squalene synthase was determined using [3H]-FPP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSqualene synthase(Rattus norvegicus)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50049224(CHEMBL158862 | Tripotassium salt of 1-Phosphono-4-...)
Affinity DataIC50:  35nMAssay Description:Inhibitory activity against rat liver microsomal squalene synthase was determined using [3H]-FPP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSqualene synthase(Rattus norvegicus)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50031846(((E)-4,8-Dimethyl-1-phosphono-nona-3,7-dienyl)-pho...)
Affinity DataIC50:  35.5nMAssay Description:Inhibition rat liver microsomal squalene synthaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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