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Found 294 with Last Name = 'kharkar' and Initial = 'p'
TargetD(3) dopamine receptor(Homo sapiens (Human))
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50303799((-)-(S)-6-(Propyl(2-(4-(quinolin-4-yl)piperazin-1-...)
Affinity DataKi:  0.190nMAssay Description:Displacement of [3H]spiperone from human dopamine D3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50303799((-)-(S)-6-(Propyl(2-(4-(quinolin-4-yl)piperazin-1-...)
Affinity DataKi:  0.400nMAssay Description:Displacement of [3H]spiperone from human dopamine D3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50303796(7-((2-(4-(Naphthalen-1-yl)-piperazin-1-yl)ethyl)(p...)
Affinity DataKi:  0.435nMAssay Description:Displacement of [3H]spiperone from human dopamine D3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50303795(7-((2-(4-(Isoquinolin-1-yl)piperazin-1-yl)ethyl)(p...)
Affinity DataKi:  0.441nMAssay Description:Displacement of [3H]spiperone from human dopamine D3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50303793((S)-(4-(2-((5-hydroxy-1,2,3,4-tetrahydronaphthalen...)
Affinity DataKi:  0.570nMAssay Description:Displacement of [3H]spiperone from human dopamine D3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
Bharati Vidyapeeth'S College Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50054653(CHEMBL3323211)
Affinity DataKi:  0.590nMAssay Description:Inhibition of human carbonic anhydrase 12 preincubated for 15 mins by stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
Bharati Vidyapeeth'S College Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50054648(CHEMBL3323207)
Affinity DataKi:  0.630nMAssay Description:Inhibition of human carbonic anhydrase 12 preincubated for 15 mins by stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
Bharati Vidyapeeth'S College Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50054646(CHEMBL3323209)
Affinity DataKi:  0.650nMAssay Description:Inhibition of human carbonic anhydrase 12 preincubated for 15 mins by stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
Bharati Vidyapeeth'S College Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50054652(CHEMBL3323212)
Affinity DataKi:  0.660nMAssay Description:Inhibition of human carbonic anhydrase 12 preincubated for 15 mins by stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
Bharati Vidyapeeth'S College Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50054650(CHEMBL3323205)
Affinity DataKi:  0.680nMAssay Description:Inhibition of human carbonic anhydrase 12 preincubated for 15 mins by stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50303797(7-((2-(4-(Naphthalen-2-yl)piperazin-1-yl)ethyl)(pr...)
Affinity DataKi:  0.685nMAssay Description:Displacement of [3H]spiperone from human dopamine D3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
Bharati Vidyapeeth'S College Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50054651(CHEMBL3323213)
Affinity DataKi:  0.710nMAssay Description:Inhibition of human carbonic anhydrase 12 preincubated for 15 mins by stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
Bharati Vidyapeeth'S College Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50054649(CHEMBL3323206)
Affinity DataKi:  0.720nMAssay Description:Inhibition of human carbonic anhydrase 12 preincubated for 15 mins by stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
Bharati Vidyapeeth'S College Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50054658(CHEMBL3323210)
Affinity DataKi:  0.790nMAssay Description:Inhibition of human carbonic anhydrase 12 preincubated for 15 mins by stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
Bharati Vidyapeeth'S College Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50054647(CHEMBL3323208)
Affinity DataKi:  0.790nMAssay Description:Inhibition of human carbonic anhydrase 12 preincubated for 15 mins by stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50273939((R)-6-((2-(4-phenylpiperazin-1-yl)ethyl)(propyl)am...)
Affinity DataKi:  0.825nMAssay Description:Displacement of [3H]spiperone from human dopamine D3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50273938((-)-(S)-6-((2-(4-phenylpiperazin-1-yl)ethyl)(propy...)
Affinity DataKi:  0.825nMAssay Description:Displacement of [3H]Spiperone from rat dopamine D3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50273996((S)-N*6*-[2-(4-Biphenyl-4-yl-piperazin-1-yl)-ethyl...)
Affinity DataKi:  0.920nMAssay Description:Displacement of [3H]spiperone from human dopamine D3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50273996((S)-N*6*-[2-(4-Biphenyl-4-yl-piperazin-1-yl)-ethyl...)
Affinity DataKi:  0.925nMAssay Description:Displacement of [3H]Spiperone from rat dopamine D3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50303794((-)-(S)-N6-Propyl-N6-(2-(4-(quinolin-5-yl)piperazi...)
Affinity DataKi:  1.21nMAssay Description:Displacement of [3H]spiperone from human dopamine D3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50303798(7-(Propyl(2-(4-(quinolin-5-yl)piperazin-1-yl)ethyl...)
Affinity DataKi:  1.27nMAssay Description:Displacement of [3H]spiperone from human dopamine D3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50020221((-)-5-hydroxy-2-(dipropylamino)tetralin | (-)-6-(d...)
Affinity DataKi:  1.36nMAssay Description:Displacement of [3H]spiperone from human dopamine D3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50273937((+)-(R)-7-((2-(4-phenylpiperazin-1-yl)ethyl)(propy...)
Affinity DataKi:  1.77nMAssay Description:Displacement of [3H]Spiperone from rat dopamine D3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50273937((+)-(R)-7-((2-(4-phenylpiperazin-1-yl)ethyl)(propy...)
Affinity DataKi:  1.77nMAssay Description:Displacement of [3H]spiperone from human dopamine D3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50303791((-)-(S)-N6-(2-(4-(Isoquinolin-1-yl)piperazin-1-yl)...)
Affinity DataKi:  2.23nMAssay Description:Displacement of [3H]spiperone from human dopamine D3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50054067((2R)-7-Dipropylamino-5,6,7,8-tetrahydro-naphthalen...)
Affinity DataKi:  2.35nMAssay Description:Displacement of [3H]spiperone from human dopamine D3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50303792((-)-(S)-N6-Propyl-N6-(2-(4-(quinolin-4-yl)piperazi...)
Affinity DataKi:  2.61nMAssay Description:Displacement of [3H]spiperone from human dopamine D3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50303800(7-(Propyl(2-(4-(quinolin-4-yl)piperazin-1-yl)ethyl...)
Affinity DataKi:  2.65nMAssay Description:Displacement of [3H]spiperone from human dopamine D3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
Bharati Vidyapeeth'S College Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50054648(CHEMBL3323207)
Affinity DataKi:  3.5nMAssay Description:Inhibition of human carbonic anhydrase 2 preincubated for 15 mins by stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
Bharati Vidyapeeth'S College Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50054651(CHEMBL3323213)
Affinity DataKi:  3.60nMAssay Description:Inhibition of human carbonic anhydrase 2 preincubated for 15 mins by stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50303799((-)-(S)-6-(Propyl(2-(4-(quinolin-4-yl)piperazin-1-...)
Affinity DataKi:  3.74nMAssay Description:Displacement of [3H]spiperone from human dopamine D2L receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
Bharati Vidyapeeth'S College Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50054652(CHEMBL3323212)
Affinity DataKi:  3.80nMAssay Description:Inhibition of human carbonic anhydrase 2 preincubated for 15 mins by stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
Bharati Vidyapeeth'S College Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50054647(CHEMBL3323208)
Affinity DataKi:  3.90nMAssay Description:Inhibition of human carbonic anhydrase 2 preincubated for 15 mins by stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50273994((S)-N6-(2-(4-phenylpiperazin-1-yl)ethyl)-N6-propyl...)
Affinity DataKi:  4.15nMAssay Description:Displacement of [3H]Spiperone from rat dopamine D3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
Bharati Vidyapeeth'S College Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50054650(CHEMBL3323205)
Affinity DataKi:  4.30nMAssay Description:Inhibition of human carbonic anhydrase 2 preincubated for 15 mins by stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50303790((-)-(S)-N6-Propyl-N6-(2-(4-(4-(pyridin-4-yl)phenyl...)
Affinity DataKi:  4.78nMAssay Description:Displacement of [3H]spiperone from human dopamine D3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50303799((-)-(S)-6-(Propyl(2-(4-(quinolin-4-yl)piperazin-1-...)
Affinity DataKi:  4.89nMAssay Description:Displacement of [3H]spiperone from human dopamine D2L receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50273418((+/-)-trans-4-(2-(4-Phenylpiperazin-1-yl)ethyl)-1,...)
Affinity DataKi:  4.95nMAssay Description:Displacement of [3H]Spiperone from rat dopamine D3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50273418((+/-)-trans-4-(2-(4-Phenylpiperazin-1-yl)ethyl)-1,...)
Affinity DataKi:  4.95nMAssay Description:Displacement of [3H]Spiperone from rat dopamine D3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50303798(7-(Propyl(2-(4-(quinolin-5-yl)piperazin-1-yl)ethyl...)
Affinity DataKi:  5.22nMAssay Description:Displacement of [3H]spiperone from human dopamine D2L receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
Bharati Vidyapeeth'S College Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM10880(AZA | AZA2 | AZM acetazolamide | Acerazolamide, AA...)
Affinity DataKi:  5.80nMAssay Description:Inhibition of human carbonic anhydrase 12 preincubated for 15 mins by stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
TargetCarbonic anhydrase 2(Homo sapiens (Human))
Bharati Vidyapeeth'S College Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50054658(CHEMBL3323210)
Affinity DataKi:  6nMAssay Description:Inhibition of human carbonic anhydrase 2 preincubated for 15 mins by stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
Bharati Vidyapeeth'S College Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50054646(CHEMBL3323209)
Affinity DataKi:  6.10nMAssay Description:Inhibition of human carbonic anhydrase 2 preincubated for 15 mins by stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50020222((+/-)-7-(dipropylamino)-5,6,7,8-tetrahydronaphthal...)
Affinity DataKi:  6.19nMAssay Description:Displacement of [3H]Spiperone from rat dopamine D3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50303800(7-(Propyl(2-(4-(quinolin-4-yl)piperazin-1-yl)ethyl...)
Affinity DataKi:  7.08nMAssay Description:Displacement of [3H]spiperone from human dopamine D2L receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50303797(7-((2-(4-(Naphthalen-2-yl)piperazin-1-yl)ethyl)(pr...)
Affinity DataKi:  8.85nMAssay Description:Displacement of [3H]spiperone from human dopamine D2L receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
Bharati Vidyapeeth'S College Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM10880(AZA | AZA2 | AZM acetazolamide | Acerazolamide, AA...)
Affinity DataKi:  12nMAssay Description:Inhibition of human carbonic anhydrase 2 preincubated for 15 mins by stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Homo sapiens (Human))
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50303796(7-((2-(4-(Naphthalen-1-yl)-piperazin-1-yl)ethyl)(p...)
Affinity DataKi:  13.5nMAssay Description:Displacement of [3H]spiperone from human dopamine D2L receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
Bharati Vidyapeeth'S College Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50054649(CHEMBL3323206)
Affinity DataKi:  14nMAssay Description:Inhibition of human carbonic anhydrase 2 preincubated for 15 mins by stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50273939((R)-6-((2-(4-phenylpiperazin-1-yl)ethyl)(propyl)am...)
Affinity DataKi:  18.4nMAssay Description:Displacement of [3H]Spiperone from rat dopamine D3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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