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Found 206 with Last Name = 'marguet' and Initial = 'f'
TargetTranslocator protein(Rattus norvegicus (rat))
Institute Of Biomedical Imaging (I2Bm)

Curated by ChEMBL
LigandPNGBDBM50210860(CHEMBL3936390)
Affinity DataKi:  0.25nMAssay Description:Displacement of [3H]PK11195 from TSPO in rat heart membranes after 15 mins by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Institute Of Biomedical Imaging (I2Bm)

Curated by ChEMBL
LigandPNGBDBM50210866(CHEMBL3979767)
Affinity DataKi:  0.260nMAssay Description:Displacement of [3H]PK11195 from TSPO in rat heart membranes after 15 mins by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Institute Of Biomedical Imaging (I2Bm)

Curated by ChEMBL
LigandPNGBDBM50210858(CHEMBL3906952)
Affinity DataKi:  0.300nMAssay Description:Displacement of [3H]PK11195 from TSPO in rat heart membranes after 15 mins by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Institute Of Biomedical Imaging (I2Bm)

Curated by ChEMBL
LigandPNGBDBM50117259(CHEMBL3613363)
Affinity DataKi:  0.300nMAssay Description:Displacement of [3H]-PK11195 from rat heart membrane TSPOMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Institute Of Biomedical Imaging (I2Bm)

Curated by ChEMBL
LigandPNGBDBM50005293(CHEMBL3125363)
Affinity DataKi:  0.350nMAssay Description:Displacement of [3H]PK11195 from TSPO in rat heart membrane homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Institute Of Biomedical Imaging (I2Bm)

Curated by ChEMBL
LigandPNGBDBM50243008(CHEMBL469682 | N,N-Diethyl-2-(2-(4-(3-fluoropropox...)
Affinity DataKi:  0.370nMAssay Description:Displacement of [3H]PK11195 from TSPO in rat heart membranes after 15 mins by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Institute Of Biomedical Imaging (I2Bm)

Curated by ChEMBL
LigandPNGBDBM50117212(CHEMBL3613360)
Affinity DataKi:  0.400nMAssay Description:Displacement of [3H]-PK11195 from rat heart membrane TSPOMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Institute Of Biomedical Imaging (I2Bm)

Curated by ChEMBL
LigandPNGBDBM50117211(CHEMBL3613361)
Affinity DataKi:  0.420nMAssay Description:Displacement of [3H]-PK11195 from rat heart membrane TSPOMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Institute Of Biomedical Imaging (I2Bm)

Curated by ChEMBL
LigandPNGBDBM50005295(CHEMBL3125361)
Affinity DataKi:  0.540nMAssay Description:Displacement of [3H]PK11195 from TSPO in rat heart membrane homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Institute Of Biomedical Imaging (I2Bm)

Curated by ChEMBL
LigandPNGBDBM50117258(CHEMBL3613358)
Affinity DataKi:  0.680nMAssay Description:Displacement of [3H]-PK11195 from rat heart membrane TSPOMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Institute Of Biomedical Imaging (I2Bm)

Curated by ChEMBL
LigandPNGBDBM50005294(CHEMBL3125362)
Affinity DataKi:  0.740nMAssay Description:Displacement of [3H]PK11195 from TSPO in rat heart membrane homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Institute Of Biomedical Imaging (I2Bm)

Curated by ChEMBL
LigandPNGBDBM50005292(CHEMBL3125364)
Affinity DataKi:  0.790nMAssay Description:Displacement of [3H]PK11195 from TSPO in rat heart membrane homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Institute Of Biomedical Imaging (I2Bm)

Curated by ChEMBL
LigandPNGBDBM50255226((7-chloro-N,N,5-trimethyl-4-oxo-3-phenyl-3,5-dihyd...)
Affinity DataKi:  0.830nMAssay Description:Displacement of [3H]-PK11195 from rat heart membrane TSPOMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Institute Of Biomedical Imaging (I2Bm)

Curated by ChEMBL
LigandPNGBDBM50243007(2-(2-(4-(2-Fluoroethoxy)phenyl)-5,7-dimethylpyrazo...)
Affinity DataKi:  0.910nMAssay Description:Displacement of [3H]PK11195 from TSPO in rat heart membranes after 15 mins by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Institute Of Biomedical Imaging (I2Bm)

Curated by ChEMBL
LigandPNGBDBM50243007(2-(2-(4-(2-Fluoroethoxy)phenyl)-5,7-dimethylpyrazo...)
Affinity DataKi:  0.910nMAssay Description:Displacement of [3H]PK11195 from TSPO in rat heart membrane homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Institute Of Biomedical Imaging (I2Bm)

Curated by ChEMBL
LigandPNGBDBM50117265(CHEMBL3613362)
Affinity DataKi:  0.960nMAssay Description:Displacement of [3H]-PK11195 from rat heart membrane TSPOMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Institute Of Biomedical Imaging (I2Bm)

Curated by ChEMBL
LigandPNGBDBM50210857(CHEMBL3938340)
Affinity DataKi:  1.10nMAssay Description:Displacement of [3H]PK11195 from TSPO in rat heart membranes after 15 mins by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRelaxin receptor 1(Homo sapiens (Human))
Sanofi R&D

Curated by ChEMBL
LigandPNGBDBM50563230(CHEMBL4754949)
Affinity DataKi:  1.10nMAssay Description:Displacement of Eu3+-labelled H2 relaxin from human RXFP1 expressed in human HEK-293T cells in presence of 10 % FCS by competition binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Institute Of Biomedical Imaging (I2Bm)

Curated by ChEMBL
LigandPNGBDBM50210864(CHEMBL3960249)
Affinity DataKi:  1.20nMAssay Description:Displacement of [3H]PK11195 from TSPO in rat heart membranes after 15 mins by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Institute Of Biomedical Imaging (I2Bm)

Curated by ChEMBL
LigandPNGBDBM50117210(CHEMBL3613359)
Affinity DataKi:  1.40nMAssay Description:Displacement of [3H]-PK11195 from rat heart membrane TSPOMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Institute Of Biomedical Imaging (I2Bm)

Curated by ChEMBL
LigandPNGBDBM50117266(CHEMBL3613365)
Affinity DataKi:  1.5nMAssay Description:Displacement of [3H]-PK11195 from rat heart membrane TSPOMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Institute Of Biomedical Imaging (I2Bm)

Curated by ChEMBL
LigandPNGBDBM50210867(CHEMBL3923539)
Affinity DataKi:  2.20nMAssay Description:Displacement of [3H]PK11195 from TSPO in rat heart membranes after 15 mins by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Institute Of Biomedical Imaging (I2Bm)

Curated by ChEMBL
LigandPNGBDBM50210863(CHEMBL3929294)
Affinity DataKi:  2.80nMAssay Description:Displacement of [3H]PK11195 from TSPO in rat heart membranes after 15 mins by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Institute Of Biomedical Imaging (I2Bm)

Curated by ChEMBL
LigandPNGBDBM50117213(CHEMBL3613366)
Affinity DataKi:  4.10nMAssay Description:Displacement of [3H]-PK11195 from rat heart membrane TSPOMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Institute Of Biomedical Imaging (I2Bm)

Curated by ChEMBL
LigandPNGBDBM50117205(CHEMBL3613370)
Affinity DataKi:  4.20nMAssay Description:Displacement of [3H]-PK11195 from rat heart membrane TSPOMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Institute Of Biomedical Imaging (I2Bm)

Curated by ChEMBL
LigandPNGBDBM50117267(CHEMBL3613364)
Affinity DataKi:  4.20nMAssay Description:Displacement of [3H]-PK11195 from rat heart membrane TSPOMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Institute Of Biomedical Imaging (I2Bm)

Curated by ChEMBL
LigandPNGBDBM50117206(CHEMBL3613369)
Affinity DataKi:  8.10nMAssay Description:Displacement of [3H]-PK11195 from rat heart membrane TSPOMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Institute Of Biomedical Imaging (I2Bm)

Curated by ChEMBL
LigandPNGBDBM50210859(CHEMBL3908452)
Affinity DataKi:  15nMAssay Description:Displacement of [3H]PK11195 from TSPO in rat heart membranes after 15 mins by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Institute Of Biomedical Imaging (I2Bm)

Curated by ChEMBL
LigandPNGBDBM50210865(CHEMBL3909555)
Affinity DataKi:  17nMAssay Description:Displacement of [3H]PK11195 from TSPO in rat heart membranes after 15 mins by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Institute Of Biomedical Imaging (I2Bm)

Curated by ChEMBL
LigandPNGBDBM50210861(CHEMBL3896806)
Affinity DataKi:  26nMAssay Description:Displacement of [3H]PK11195 from TSPO in rat heart membranes after 15 mins by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Institute Of Biomedical Imaging (I2Bm)

Curated by ChEMBL
LigandPNGBDBM50210868(CHEMBL3981447)
Affinity DataKi:  27nMAssay Description:Displacement of [3H]PK11195 from TSPO in rat heart membranes after 15 mins by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Institute Of Biomedical Imaging (I2Bm)

Curated by ChEMBL
LigandPNGBDBM50210856(CHEMBL3906707)
Affinity DataKi:  32nMAssay Description:Displacement of [3H]PK11195 from TSPO in rat heart membranes after 15 mins by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Institute Of Biomedical Imaging (I2Bm)

Curated by ChEMBL
LigandPNGBDBM50117209(CHEMBL3613367)
Affinity DataKi:  61nMAssay Description:Displacement of [3H]-PK11195 from rat heart membrane TSPOMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Institute Of Biomedical Imaging (I2Bm)

Curated by ChEMBL
LigandPNGBDBM50117208(CHEMBL3613368)
Affinity DataKi:  120nMAssay Description:Displacement of [3H]-PK11195 from rat heart membrane TSPOMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Institute Of Biomedical Imaging (I2Bm)

Curated by ChEMBL
LigandPNGBDBM50117202(CHEMBL3613371)
Affinity DataKi:  130nMAssay Description:Displacement of [3H]-PK11195 from rat heart membrane TSPOMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Institute Of Biomedical Imaging (I2Bm)

Curated by ChEMBL
LigandPNGBDBM50210862(CHEMBL3920384)
Affinity DataKi:  260nMAssay Description:Displacement of [3H]PK11195 from TSPO in rat heart membranes after 15 mins by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Institute Of Biomedical Imaging (I2Bm)

Curated by ChEMBL
LigandPNGBDBM50117201(CHEMBL3613372)
Affinity DataKi:  920nMAssay Description:Displacement of [3H]-PK11195 from rat heart membrane TSPOMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRelaxin receptor 1(Homo sapiens (Human))
Sanofi R&D

Curated by ChEMBL
LigandPNGBDBM50563231(CHEMBL4780098)
Affinity DataKi:  2.88E+3nMAssay Description:Displacement of Eu3+-labelled H2 relaxin from human RXFP1 expressed in human HEK-293T cells in presence of 10 % FCS by competition binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCasein kinase I isoform epsilon(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM207015(US9233965, 100)
Affinity DataIC50: >1nMpH: 7.5 T: 2°CAssay Description:"U"-bottomed Falcon plates are prepared by placing 5 uL of solutions of the compounds according to the invention at concentrations of 10, 1, 0.1, 0.0...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCasein kinase I isoform epsilon(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM207003(US9233965, 86)
Affinity DataIC50: <1nMpH: 7.5 T: 2°CAssay Description:"U"-bottomed Falcon plates are prepared by placing 5 uL of solutions of the compounds according to the invention at concentrations of 10, 1, 0.1, 0.0...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCasein kinase I isoform epsilon(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM207001(US9233965, 84)
Affinity DataIC50:  1nMpH: 7.5 T: 2°CAssay Description:"U"-bottomed Falcon plates are prepared by placing 5 uL of solutions of the compounds according to the invention at concentrations of 10, 1, 0.1, 0.0...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCasein kinase I isoform epsilon(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM207024(US9233965, 2)
Affinity DataIC50: <1nMpH: 7.5 T: 2°CAssay Description:"U"-bottomed Falcon plates are prepared by placing 5 uL of solutions of the compounds according to the invention at concentrations of 10, 1, 0.1, 0.0...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCasein kinase I isoform epsilon(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM207023(US9233965, 110)
Affinity DataIC50: <1nMpH: 7.5 T: 2°CAssay Description:"U"-bottomed Falcon plates are prepared by placing 5 uL of solutions of the compounds according to the invention at concentrations of 10, 1, 0.1, 0.0...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCasein kinase I isoform epsilon(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM207020(US9233965, 107)
Affinity DataIC50: <1nMpH: 7.5 T: 2°CAssay Description:"U"-bottomed Falcon plates are prepared by placing 5 uL of solutions of the compounds according to the invention at concentrations of 10, 1, 0.1, 0.0...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCasein kinase I isoform epsilon(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM206925(US9233965, 105)
Affinity DataIC50: <1nMpH: 7.5 T: 2°CAssay Description:"U"-bottomed Falcon plates are prepared by placing 5 uL of solutions of the compounds according to the invention at concentrations of 10, 1, 0.1, 0.0...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCasein kinase I isoform epsilon(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM206924(US9233965, 104)
Affinity DataIC50: <1nMpH: 7.5 T: 2°CAssay Description:"U"-bottomed Falcon plates are prepared by placing 5 uL of solutions of the compounds according to the invention at concentrations of 10, 1, 0.1, 0.0...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCasein kinase I isoform epsilon(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM206926(US9233965, 87)
Affinity DataIC50: <1nMpH: 7.5 T: 2°CAssay Description:"U"-bottomed Falcon plates are prepared by placing 5 uL of solutions of the compounds according to the invention at concentrations of 10, 1, 0.1, 0.0...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCasein kinase I isoform epsilon(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM206971(US9233965, 48)
Affinity DataIC50:  1.5nMpH: 7.5 T: 2°CAssay Description:"U"-bottomed Falcon plates are prepared by placing 5 uL of solutions of the compounds according to the invention at concentrations of 10, 1, 0.1, 0.0...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCasein kinase I isoform epsilon(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM206920(US9233965, 64)
Affinity DataIC50:  2nMpH: 7.5 T: 2°CAssay Description:"U"-bottomed Falcon plates are prepared by placing 5 uL of solutions of the compounds according to the invention at concentrations of 10, 1, 0.1, 0.0...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCasein kinase I isoform epsilon(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM206981(US9233965, 62)
Affinity DataIC50:  2nMpH: 7.5 T: 2°CAssay Description:"U"-bottomed Falcon plates are prepared by placing 5 uL of solutions of the compounds according to the invention at concentrations of 10, 1, 0.1, 0.0...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
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