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Found 101 with Last Name = 'marschner' and Initial = 'a'
TargetMethionine aminopeptidase(Escherichia coli (strain K12))
Heidelberg University

Curated by ChEMBL
LigandPNGBDBM50497521(CHEMBL3337749)
Affinity DataIC50:  190nMAssay Description:Inhibition of C-terminal poly-His-tagged Escherichia coli MetAP expressed in Escherichia coli BL21(DE3) incubated for 30 mins before MGMM substrate a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMethionine aminopeptidase(Escherichia coli (strain K12))
Heidelberg University

Curated by ChEMBL
LigandPNGBDBM50497538(CHEMBL3337748)
Affinity DataIC50:  230nMAssay Description:Inhibition of C-terminal poly-His-tagged Escherichia coli MetAP expressed in Escherichia coli BL21(DE3) incubated for 30 mins before MGMM substrate a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMethionine aminopeptidase(Escherichia coli (strain K12))
Heidelberg University

Curated by ChEMBL
LigandPNGBDBM50497533(CHEMBL3337746)
Affinity DataIC50:  400nMAssay Description:Inhibition of C-terminal poly-His-tagged Escherichia coli MetAP expressed in Escherichia coli BL21(DE3) incubated for 30 mins before MGMM substrate a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMethionine aminopeptidase(Escherichia coli (strain K12))
Heidelberg University

Curated by ChEMBL
LigandPNGBDBM50497531(CHEMBL3337750)
Affinity DataIC50:  670nMAssay Description:Inhibition of C-terminal poly-His-tagged Escherichia coli MetAP expressed in Escherichia coli BL21(DE3) incubated for 30 mins before MGMM substrate a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMethionine aminopeptidase(Escherichia coli (strain K12))
Heidelberg University

Curated by ChEMBL
LigandPNGBDBM50497517(CHEMBL3337739)
Affinity DataIC50:  700nMAssay Description:Inhibition of C-terminal poly-His-tagged Escherichia coli MetAP expressed in Escherichia coli BL21(DE3) incubated for 30 mins before MGMM substrate a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMethionine aminopeptidase(Escherichia coli (strain K12))
Heidelberg University

Curated by ChEMBL
LigandPNGBDBM50497532(CHEMBL3337751)
Affinity DataIC50:  700nMAssay Description:Inhibition of C-terminal poly-His-tagged Escherichia coli MetAP expressed in Escherichia coli BL21(DE3) incubated for 30 mins before MGMM substrate a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMethionine aminopeptidase(Escherichia coli (strain K12))
Heidelberg University

Curated by ChEMBL
LigandPNGBDBM50497528(CHEMBL3337742)
Affinity DataIC50:  720nMAssay Description:Inhibition of C-terminal poly-His-tagged Escherichia coli MetAP expressed in Escherichia coli BL21(DE3) incubated for 30 mins before MGMM substrate a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMethionine aminopeptidase(Escherichia coli (strain K12))
Heidelberg University

Curated by ChEMBL
LigandPNGBDBM50497520(CHEMBL3337747)
Affinity DataIC50:  800nMAssay Description:Inhibition of C-terminal poly-His-tagged Escherichia coli MetAP expressed in Escherichia coli BL21(DE3) incubated for 30 mins before MGMM substrate a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMethionine aminopeptidase(Escherichia coli (strain K12))
Heidelberg University

Curated by ChEMBL
LigandPNGBDBM50497525(CHEMBL3337744)
Affinity DataIC50:  830nMAssay Description:Inhibition of C-terminal poly-His-tagged Escherichia coli MetAP expressed in Escherichia coli BL21(DE3) incubated for 30 mins before MGMM substrate a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMethionine aminopeptidase(Escherichia coli (strain K12))
Heidelberg University

Curated by ChEMBL
LigandPNGBDBM50497527(CHEMBL3337741)
Affinity DataIC50:  840nMAssay Description:Inhibition of C-terminal poly-His-tagged Escherichia coli MetAP expressed in Escherichia coli BL21(DE3) incubated for 30 mins before MGMM substrate a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMethionine aminopeptidase(Escherichia coli (strain K12))
Heidelberg University

Curated by ChEMBL
LigandPNGBDBM50497522(CHEMBL186008)
Affinity DataIC50:  980nMAssay Description:Inhibition of C-terminal poly-His-tagged Escherichia coli MetAP expressed in Escherichia coli BL21(DE3) incubated for 30 mins before MGMM substrate a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMethionine aminopeptidase 1(Homo sapiens (Human))
Heidelberg University

Curated by ChEMBL
LigandPNGBDBM50497538(CHEMBL3337748)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of N-terminal poly-His-tagged human MetAP-1 expressed in Escherichia coli BL21(DE3) incubated for 30 mins before MGMM substrate addition b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMethionine aminopeptidase(Escherichia coli (strain K12))
Heidelberg University

Curated by ChEMBL
LigandPNGBDBM50497518(CHEMBL3337738)
Affinity DataIC50:  1.10E+3nMAssay Description:Inhibition of C-terminal poly-His-tagged Escherichia coli MetAP expressed in Escherichia coli BL21(DE3) incubated for 30 mins before MGMM substrate a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMethionine aminopeptidase(Escherichia coli (strain K12))
Heidelberg University

Curated by ChEMBL
LigandPNGBDBM50497519(CHEMBL3337745)
Affinity DataIC50:  1.70E+3nMAssay Description:Inhibition of C-terminal poly-His-tagged Escherichia coli MetAP expressed in Escherichia coli BL21(DE3) incubated for 30 mins before MGMM substrate a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMethionine aminopeptidase(Escherichia coli (strain K12))
Heidelberg University

Curated by ChEMBL
LigandPNGBDBM50497529(CHEMBL3337743)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of C-terminal poly-His-tagged Escherichia coli MetAP expressed in Escherichia coli BL21(DE3) incubated for 30 mins before MGMM substrate a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMethionine aminopeptidase(Escherichia coli (strain K12))
Heidelberg University

Curated by ChEMBL
LigandPNGBDBM50497536(CHEMBL3337629)
Affinity DataIC50:  2.10E+3nMAssay Description:Inhibition of C-terminal poly-His-tagged Escherichia coli MetAP expressed in Escherichia coli BL21(DE3) incubated for 30 mins before MGMM substrate a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMethionine aminopeptidase(Escherichia coli (strain K12))
Heidelberg University

Curated by ChEMBL
LigandPNGBDBM50497530(CHEMBL3337638)
Affinity DataIC50:  2.80E+3nMAssay Description:Inhibition of C-terminal poly-His-tagged Escherichia coli MetAP expressed in Escherichia coli BL21(DE3) incubated for 30 mins before MGMM substrate a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMethionine aminopeptidase(Escherichia coli (strain K12))
Heidelberg University

Curated by ChEMBL
LigandPNGBDBM50497523(CHEMBL3337736)
Affinity DataIC50:  3.10E+3nMAssay Description:Inhibition of C-terminal poly-His-tagged Escherichia coli MetAP expressed in Escherichia coli BL21(DE3) incubated for 30 mins before MGMM substrate a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMethionine aminopeptidase 1(Homo sapiens (Human))
Heidelberg University

Curated by ChEMBL
LigandPNGBDBM50497521(CHEMBL3337749)
Affinity DataIC50:  3.50E+3nMAssay Description:Inhibition of N-terminal poly-His-tagged human MetAP-1 expressed in Escherichia coli BL21(DE3) incubated for 30 mins before MGMM substrate addition b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMethionine aminopeptidase 1(Homo sapiens (Human))
Heidelberg University

Curated by ChEMBL
LigandPNGBDBM50497528(CHEMBL3337742)
Affinity DataIC50:  3.50E+3nMAssay Description:Inhibition of N-terminal poly-His-tagged human MetAP-1 expressed in Escherichia coli BL21(DE3) incubated for 30 mins before MGMM substrate addition b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMethionine aminopeptidase(Escherichia coli (strain K12))
Heidelberg University

Curated by ChEMBL
LigandPNGBDBM50497537(CHEMBL3337628)
Affinity DataIC50:  3.70E+3nMAssay Description:Inhibition of C-terminal poly-His-tagged Escherichia coli MetAP expressed in Escherichia coli BL21(DE3) incubated for 30 mins before MGMM substrate a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMethionine aminopeptidase(Escherichia coli (strain K12))
Heidelberg University

Curated by ChEMBL
LigandPNGBDBM50497535(CHEMBL3337630)
Affinity DataIC50:  3.80E+3nMAssay Description:Inhibition of C-terminal poly-His-tagged Escherichia coli MetAP expressed in Escherichia coli BL21(DE3) incubated for 30 mins before MGMM substrate a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMethionine aminopeptidase 2(Homo sapiens (Human))
Universit£T Heidelberg

Curated by ChEMBL
LigandPNGBDBM32203(8-quinolinol | CHEMBL310555 | US10005735, Table 1....)
Affinity DataIC50:  5.60E+3nMAssay Description:Inhibition of human MetAP2 expressed in baculovirus infected Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMethionine aminopeptidase(Staphylococcus aureus)
Heidelberg University

Curated by ChEMBL
LigandPNGBDBM50497527(CHEMBL3337741)
Affinity DataIC50:  7.00E+3nMAssay Description:Inhibition of N-terminal poly-His-tagged Staphylococcus aureus COL MetAP expressed in Escherichia coli BL21(DE3) incubated for 30 mins before MGMM su...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMethionine aminopeptidase(Escherichia coli (strain K12))
Heidelberg University

Curated by ChEMBL
LigandPNGBDBM50497526(CHEMBL3337737)
Affinity DataIC50:  7.00E+3nMAssay Description:Inhibition of C-terminal poly-His-tagged Escherichia coli MetAP expressed in Escherichia coli BL21(DE3) incubated for 30 mins before MGMM substrate a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMethionine aminopeptidase 2(Homo sapiens (Human))
Universit£T Heidelberg

Curated by ChEMBL
LigandPNGBDBM50180733(5-Methyl-2-pyridin-2-yl-1H-benzoimidazole | 5-meth...)
Affinity DataIC50:  7.70E+3nMAssay Description:Inhibition of human MetAP2 expressed in baculovirus infected Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMethionine aminopeptidase(Staphylococcus aureus)
Heidelberg University

Curated by ChEMBL
LigandPNGBDBM50497528(CHEMBL3337742)
Affinity DataIC50:  7.80E+3nMAssay Description:Inhibition of N-terminal poly-His-tagged Staphylococcus aureus COL MetAP expressed in Escherichia coli BL21(DE3) incubated for 30 mins before MGMM su...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMethionine aminopeptidase 2(Homo sapiens (Human))
Universit£T Heidelberg

Curated by ChEMBL
LigandPNGBDBM50180747(2-pyridin-2-yl-1H-imidazo[4,5-c]pyridine | CHEMBL2...)
Affinity DataIC50:  8.00E+3nMAssay Description:Inhibition of human MetAP2 expressed in baculovirus infected Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMethionine aminopeptidase 1(Homo sapiens (Human))
Heidelberg University

Curated by ChEMBL
LigandPNGBDBM50129661(CHEMBL89671 | N-(thiazol-2-yl)picolinamide | Pyrid...)
Affinity DataIC50:  8.10E+3nMAssay Description:Inhibition of human MetAP1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMethionine aminopeptidase(Escherichia coli (strain K12))
Heidelberg University

Curated by ChEMBL
LigandPNGBDBM50497524(CHEMBL3245455)
Affinity DataIC50:  8.40E+3nMAssay Description:Inhibition of C-terminal poly-His-tagged Escherichia coli MetAP expressed in Escherichia coli BL21(DE3) incubated for 30 mins before MGMM substrate a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMethionine aminopeptidase(Escherichia coli (strain K12))
Heidelberg University

Curated by ChEMBL
LigandPNGBDBM50497540(CHEMBL3245452)
Affinity DataIC50:  9.10E+3nMAssay Description:Inhibition of C-terminal poly-His-tagged Escherichia coli MetAP expressed in Escherichia coli BL21(DE3) incubated for 30 mins before MGMM substrate a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMethionine aminopeptidase 2(Homo sapiens (Human))
Universit£T Heidelberg

Curated by ChEMBL
LigandPNGBDBM62926(2-(2-pyridinyl)-3H-benzimidazol-5-amine | 2-Pyridi...)
Affinity DataIC50:  9.30E+3nMAssay Description:Inhibition of human MetAP2 expressed in baculovirus infected Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMethionine aminopeptidase 2(Homo sapiens (Human))
Universit£T Heidelberg

Curated by ChEMBL
LigandPNGBDBM50180749(2-(thiazol-4-yl)-1H-benzo[d]imidazol-5-amine | 5-a...)
Affinity DataIC50:  1.01E+4nMAssay Description:Inhibition of human MetAP2 expressed in baculovirus infected Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMethionine aminopeptidase 1(Homo sapiens (Human))
Heidelberg University

Curated by ChEMBL
LigandPNGBDBM50180747(2-pyridin-2-yl-1H-imidazo[4,5-c]pyridine | CHEMBL2...)
Affinity DataIC50:  1.03E+4nMAssay Description:Inhibition of human MetAP1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMethionine aminopeptidase 1(Homo sapiens (Human))
Heidelberg University

Curated by ChEMBL
LigandPNGBDBM50497520(CHEMBL3337747)
Affinity DataIC50:  1.22E+4nMAssay Description:Inhibition of N-terminal poly-His-tagged human MetAP-1 expressed in Escherichia coli BL21(DE3) incubated for 30 mins before MGMM substrate addition b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMethionine aminopeptidase 1(Homo sapiens (Human))
Heidelberg University

Curated by ChEMBL
LigandPNGBDBM50497527(CHEMBL3337741)
Affinity DataIC50:  1.29E+4nMAssay Description:Inhibition of N-terminal poly-His-tagged human MetAP-1 expressed in Escherichia coli BL21(DE3) incubated for 30 mins before MGMM substrate addition b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMethionine aminopeptidase 2(Homo sapiens (Human))
Universit£T Heidelberg

Curated by ChEMBL
LigandPNGBDBM50078834(2-(pyridin-2-yl)-1H-benzo[d]imidazole | 2-pyridin-...)
Affinity DataIC50:  1.33E+4nMAssay Description:Inhibition of human MetAP2 expressed in baculovirus infected Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMethionine aminopeptidase(Staphylococcus aureus)
Heidelberg University

Curated by ChEMBL
LigandPNGBDBM50497533(CHEMBL3337746)
Affinity DataIC50:  1.33E+4nMAssay Description:Inhibition of N-terminal poly-His-tagged Staphylococcus aureus COL MetAP expressed in Escherichia coli BL21(DE3) incubated for 30 mins before MGMM su...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMethionine aminopeptidase 2(Homo sapiens (Human))
Universit£T Heidelberg

Curated by ChEMBL
LigandPNGBDBM50180735(5-fluoro-2-(pyridin-2-yl)-1H-benzo[d]imidazole | 5...)
Affinity DataIC50:  1.49E+4nMAssay Description:Inhibition of human MetAP2 expressed in baculovirus infected Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMethionine aminopeptidase(Staphylococcus aureus)
Heidelberg University

Curated by ChEMBL
LigandPNGBDBM50497517(CHEMBL3337739)
Affinity DataIC50:  1.50E+4nMAssay Description:Inhibition of N-terminal poly-His-tagged Staphylococcus aureus COL MetAP expressed in Escherichia coli BL21(DE3) incubated for 30 mins before MGMM su...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMethionine aminopeptidase 1(Homo sapiens (Human))
Heidelberg University

Curated by ChEMBL
LigandPNGBDBM50497517(CHEMBL3337739)
Affinity DataIC50:  1.62E+4nMAssay Description:Inhibition of N-terminal poly-His-tagged human MetAP-1 expressed in Escherichia coli BL21(DE3) incubated for 30 mins before MGMM substrate addition b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMethionine aminopeptidase 1(Homo sapiens (Human))
Heidelberg University

Curated by ChEMBL
LigandPNGBDBM50497525(CHEMBL3337744)
Affinity DataIC50:  1.65E+4nMAssay Description:Inhibition of N-terminal poly-His-tagged human MetAP-1 expressed in Escherichia coli BL21(DE3) incubated for 30 mins before MGMM substrate addition b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMethionine aminopeptidase(Staphylococcus aureus)
Heidelberg University

Curated by ChEMBL
LigandPNGBDBM50497525(CHEMBL3337744)
Affinity DataIC50:  1.70E+4nMAssay Description:Inhibition of N-terminal poly-His-tagged Staphylococcus aureus COL MetAP expressed in Escherichia coli BL21(DE3) incubated for 30 mins before MGMM su...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMethionine aminopeptidase 2(Homo sapiens (Human))
Universit£T Heidelberg

Curated by ChEMBL
LigandPNGBDBM50180732(5-Chloro-2-pyridin-2-yl-1H-benzoimidazole | 5-chlo...)
Affinity DataIC50:  1.81E+4nMAssay Description:Inhibition of human MetAP2 expressed in baculovirus infected Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMethionine aminopeptidase 1(Homo sapiens (Human))
Heidelberg University

Curated by ChEMBL
LigandPNGBDBM50497531(CHEMBL3337750)
Affinity DataIC50:  1.88E+4nMAssay Description:Inhibition of N-terminal poly-His-tagged human MetAP-1 expressed in Escherichia coli BL21(DE3) incubated for 30 mins before MGMM substrate addition b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMethionine aminopeptidase(Staphylococcus aureus)
Heidelberg University

Curated by ChEMBL
LigandPNGBDBM50497532(CHEMBL3337751)
Affinity DataIC50:  1.89E+4nMAssay Description:Inhibition of N-terminal poly-His-tagged Staphylococcus aureus COL MetAP expressed in Escherichia coli BL21(DE3) incubated for 30 mins before MGMM su...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMethionine aminopeptidase(Staphylococcus aureus)
Heidelberg University

Curated by ChEMBL
LigandPNGBDBM50497519(CHEMBL3337745)
Affinity DataIC50:  1.89E+4nMAssay Description:Inhibition of N-terminal poly-His-tagged Staphylococcus aureus COL MetAP expressed in Escherichia coli BL21(DE3) incubated for 30 mins before MGMM su...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMethionine aminopeptidase 1(Homo sapiens (Human))
Heidelberg University

Curated by ChEMBL
LigandPNGBDBM50180745(2-thiazol-4-yl-1H-imidazo[4,5-c]pyridine | 4-(1H-i...)
Affinity DataIC50:  1.90E+4nMAssay Description:Inhibition of human MetAP1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMethionine aminopeptidase 1(Homo sapiens (Human))
Heidelberg University

Curated by ChEMBL
LigandPNGBDBM50497533(CHEMBL3337746)
Affinity DataIC50:  1.97E+4nMAssay Description:Inhibition of N-terminal poly-His-tagged human MetAP-1 expressed in Escherichia coli BL21(DE3) incubated for 30 mins before MGMM substrate addition b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMethionine aminopeptidase 1(Homo sapiens (Human))
Heidelberg University

Curated by ChEMBL
LigandPNGBDBM32203(8-quinolinol | CHEMBL310555 | US10005735, Table 1....)
Affinity DataIC50:  2.15E+4nMAssay Description:Inhibition of human MetAP1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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