Affinity DataIC50: 3nMAssay Description:Ability to inhibit Trypsin was evaluated by amidolytic method using fluorogenic or chromogenic substratesChecked by AuthorMore data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Membrane Research Group Of The Hungarian Academy Of Sciences
Curated by ChEMBL
Membrane Research Group Of The Hungarian Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 5nMAssay Description:TP_TRANSPORTER: efflux of Hoechst33342 in BCRP-expressing Sf9 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 9nMAssay Description:Ability to inhibit Thrombin was evaluated by amidolytic method using fluorogenic or chromogenic substratesChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataIC50: 22.3nMAssay Description:Amidolytic activity of THP.1 cell lysate against IL-1 beta converting enzyme using C1-Asp-AMC as a substrateChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataIC50: 70nMAssay Description:Ability to inhibit papain was evaluated by amidolytic method using fluorogenic or chromogenic substratesChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataIC50: 130nMAssay Description:Ability to inhibit papain was evaluated by amidolytic method using fluorogenic or chromogenic substratesChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataIC50: 190nMAssay Description:Ability to inhibit Thrombin was evaluated by amidolytic method using fluorogenic or chromogenic substratesChecked by AuthorMore data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Membrane Research Group Of The Hungarian Academy Of Sciences
Curated by ChEMBL
Membrane Research Group Of The Hungarian Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 200nMAssay Description:TP_TRANSPORTER: efflux of Hoechst33342 in BCRP-expressing Sf9 cellsMore data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Membrane Research Group Of The Hungarian Academy Of Sciences
Curated by ChEMBL
Membrane Research Group Of The Hungarian Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 400nMAssay Description:TP_TRANSPORTER: efflux of Hoechst33342 in BCRP-expressing Sf9 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 438nMAssay Description:Amidolytic activity of THP.1 cell lysate against Caspase-3 using C3-Asp-AMC as a substrateChecked by AuthorMore data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Membrane Research Group Of The Hungarian Academy Of Sciences
Curated by ChEMBL
Membrane Research Group Of The Hungarian Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 500nMAssay Description:TP_TRANSPORTER: inhibition of ATPase activity in BCRP-expressing Sf9 cellsMore data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Membrane Research Group Of The Hungarian Academy Of Sciences
Curated by ChEMBL
Membrane Research Group Of The Hungarian Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 900nMAssay Description:TP_TRANSPORTER: efflux of Hoechst33342 in BCRP-expressing Sf9 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 1.76E+3nMAssay Description:Ability to inhibit Trypsin was evaluated by amidolytic method using fluorogenic or chromogenic substratesChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataIC50: 1.79E+3nMAssay Description:Ability to inhibit Trypsin was evaluated by amidolytic method using fluorogenic or chromogenic substratesChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataIC50: 2.00E+3nMAssay Description:Ability to inhibit IL-1 beta converting enzyme was evaluated in LPS-stimulated human whole bloodChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataIC50: 2.90E+3nMAssay Description:Ability to inhibit IL-1 beta converting enzyme was evaluated in LPS-stimulated human whole bloodChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataIC50: 5.44E+3nMAssay Description:Ability to inhibit Thrombin was evaluated by amidolytic method using fluorogenic or chromogenic substratesChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataIC50: 8.50E+3nMAssay Description:Ability to inhibit papain was evaluated by amidolytic method using fluorogenic or chromogenic substratesChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataIC50: 1.25E+4nMAssay Description:Ability to inhibit papain was evaluated by amidolytic method using fluorogenic or chromogenic substratesChecked by AuthorMore data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Membrane Research Group Of The Hungarian Academy Of Sciences
Curated by ChEMBL
Membrane Research Group Of The Hungarian Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: >5.00E+4nMAssay Description:TP_TRANSPORTER: efflux of Hoechst33342 in BCRP-expressing Sf9 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 6.50E+4nMAssay Description:Ability to inhibit papain was evaluated by amidolytic method using fluorogenic or chromogenic substratesChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataIC50: 6.80E+4nMAssay Description:Amidolytic activity of THP.1 cell lysate against IL-1 beta converting enzyme using C1-Asp-AMC as a substrateChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataIC50: 7.00E+4nMAssay Description:Amidolytic activity of THP.1 cell lysate against IL-1 beta converting enzyme using C1-Asp-AMC as a substrateChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataIC50: 1.05E+5nMAssay Description:Ability to inhibit papain was evaluated by amidolytic method using fluorogenic or chromogenic substratesChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataIC50: 1.42E+5nMAssay Description:Amidolytic activity of THP.1 cell lysate against IL-1 beta converting enzyme using C1-Asp-AMC as a substrateChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataIC50: 1.90E+5nMAssay Description:Amidolytic activity of THP.1 cell lysate against Caspase-3 using C3-Asp-AMC as a substrateChecked by AuthorMore data for this Ligand-Target Pair