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Found 122 with Last Name = 'ortega-caballero' and Initial = 'f'
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
University Of Aarhus

Curated by ChEMBL
LigandPNGBDBM50222175(2-(3,4-dichlorophenyl)-N-(furan-2-ylmethyl)cyclope...)
Affinity DataKi:  30nMAssay Description:Displacement of [125I]RTI55 from human DAT transfected in COS1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
University Of Aarhus

Curated by ChEMBL
LigandPNGBDBM50222179(CHEMBL248824 | m-tolyl 2-(3,4-dichlorophenyl)cyclo...)
Affinity DataKi:  60nMAssay Description:Displacement of [125I]RTI55 from human DAT transfected in COS1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
University Of Aarhus

Curated by ChEMBL
LigandPNGBDBM50222191(2-(3,4-dichlorophenyl)-N-(2-fluoroethyl)cyclopent-...)
Affinity DataKi:  70nMAssay Description:Displacement of [125I]RTI55 from human DAT transfected in COS1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
University Of Aarhus

Curated by ChEMBL
LigandPNGBDBM50222184(2-(3,4-dichlorophenyl)-N-(thiophen-2-ylmethyl)cycl...)
Affinity DataKi:  140nMAssay Description:Displacement of [125I]RTI55 from human DAT transfected in COS1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
University Of Aarhus

Curated by ChEMBL
LigandPNGBDBM50222188(CHEMBL401071 | phenyl 2-(3,4-dichlorophenyl)cyclop...)
Affinity DataKi:  170nMAssay Description:Displacement of [125I]RTI55 from human DAT transfected in COS1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
University Of Aarhus

Curated by ChEMBL
LigandPNGBDBM50222183(CHEMBL403570 | o-tolyl 2-(3,4-dichlorophenyl)cyclo...)
Affinity DataKi:  220nMAssay Description:Displacement of [125I]RTI55 from human DAT transfected in COS1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
University Of Aarhus

Curated by ChEMBL
LigandPNGBDBM50222182(2-hydroxyethyl 2-(3,4-dichlorophenyl)cyclopent-1-e...)
Affinity DataKi:  300nMAssay Description:Displacement of [125I]RTI55 from human DAT transfected in COS1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
University Of Aarhus

Curated by ChEMBL
LigandPNGBDBM50222178(CHEMBL403571 | thiophen-2-ylmethyl 2-(3,4-dichloro...)
Affinity DataKi:  400nMAssay Description:Displacement of [125I]RTI55 from human DAT transfected in COS1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
University Of Aarhus

Curated by ChEMBL
LigandPNGBDBM50222186(2-fluoroethyl 2-(3,4-dichlorophenyl)cyclopent-1-en...)
Affinity DataKi:  500nMAssay Description:Displacement of [125I]RTI55 from human DAT transfected in COS1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-mannosidase(Canavalia ensiformis)
University Of Sevilla

Curated by ChEMBL
LigandPNGBDBM50525020(CHEMBL4518572)
Affinity DataKi:  500nMAssay Description:Inhibition of jack bean Lysosomal alpha-mannosidase assessed as residual hydrolytic activity after 10 to 30 mins by spectrophotometric analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-mannosidase(Canavalia ensiformis)
University Of Sevilla

Curated by ChEMBL
LigandPNGBDBM50525018(CHEMBL4465842)
Affinity DataKi:  500nMAssay Description:Inhibition of jack bean Lysosomal alpha-mannosidase assessed as residual hydrolytic activity after 10 to 30 mins by spectrophotometric analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-mannosidase(Canavalia ensiformis)
University Of Sevilla

Curated by ChEMBL
LigandPNGBDBM50525017(CHEMBL4462117)
Affinity DataKi:  500nMAssay Description:Inhibition of jack bean Lysosomal alpha-mannosidase assessed as residual hydrolytic activity after 10 to 30 mins by spectrophotometric analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-mannosidase(Canavalia ensiformis)
University Of Sevilla

Curated by ChEMBL
LigandPNGBDBM50525014(CHEMBL4475419)
Affinity DataKi:  500nMAssay Description:Inhibition of jack bean Lysosomal alpha-mannosidase assessed as residual hydrolytic activity after 10 to 30 mins by spectrophotometric analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-mannosidase(Canavalia ensiformis)
University Of Sevilla

Curated by ChEMBL
LigandPNGBDBM50525016(CHEMBL4457217)
Affinity DataKi:  500nMAssay Description:Inhibition of jack bean Lysosomal alpha-mannosidase assessed as residual hydrolytic activity after 10 to 30 mins by spectrophotometric analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-mannosidase(Canavalia ensiformis)
University Of Sevilla

Curated by ChEMBL
LigandPNGBDBM50525015(CHEMBL4435118)
Affinity DataKi:  500nMAssay Description:Inhibition of jack bean Lysosomal alpha-mannosidase assessed as residual hydrolytic activity after 10 to 30 mins by spectrophotometric analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
University Of Aarhus

Curated by ChEMBL
LigandPNGBDBM50222185(2-(3,4-dichlorophenyl)-N-methoxycyclopent-1-enecar...)
Affinity DataKi:  830nMAssay Description:Displacement of [125I]RTI55 from human DAT transfected in COS1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
University Of Aarhus

Curated by ChEMBL
LigandPNGBDBM50222187(CHEMBL248825 | furan-2-ylmethyl 2-(3,4-dichlorophe...)
Affinity DataKi:  1.50E+3nMAssay Description:Displacement of [125I]RTI55 from human DAT transfected in COS1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
University Of Aarhus

Curated by ChEMBL
LigandPNGBDBM50211023(CHEMBL245061 | methyl 2-(3,4-dichlorophenyl)cyclop...)
Affinity DataKi:  1.90E+3nMAssay Description:Displacement of [125I]RTI55 from human DAT transfected in COS1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
University Of Aarhus

Curated by ChEMBL
LigandPNGBDBM50222176(CHEMBL401069 | isopropyl 2-(3,4-dichlorophenyl)cyc...)
Affinity DataKi:  2.60E+3nMAssay Description:Displacement of [125I]RTI55 from human DAT transfected in COS1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-mannosidase(Canavalia ensiformis)
University Of Sevilla

Curated by ChEMBL
LigandPNGBDBM50525019(CHEMBL4471561)
Affinity DataKi:  3.20E+3nMAssay Description:Inhibition of jack bean Lysosomal alpha-mannosidase assessed as residual hydrolytic activity after 10 to 30 mins by spectrophotometric analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
University Of Aarhus

Curated by ChEMBL
LigandPNGBDBM50222177(2,2,2-trifluoroethyl 2-(3,4-dichlorophenyl)cyclope...)
Affinity DataKi:  3.40E+3nMAssay Description:Displacement of [125I]RTI55 from human DAT transfected in COS1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
University Of Aarhus

Curated by ChEMBL
LigandPNGBDBM50222186(2-fluoroethyl 2-(3,4-dichlorophenyl)cyclopent-1-en...)
Affinity DataKi:  5.80E+3nMAssay Description:Displacement of [125I]RTI55 from human NET transfected in COS1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
University Of Aarhus

Curated by ChEMBL
LigandPNGBDBM50222192(2-(3,4-dichlorophenyl)-N-methoxy-N-methylcyclopent...)
Affinity DataKi:  6.40E+3nMAssay Description:Displacement of [125I]RTI55 from human DAT transfected in COS1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-mannosidase(Canavalia ensiformis)
University Of Sevilla

Curated by ChEMBL
LigandPNGBDBM50525021(CHEMBL4483772)
Affinity DataKi:  7.00E+3nMAssay Description:Inhibition of jack bean Lysosomal alpha-mannosidase assessed as residual hydrolytic activity after 10 to 30 mins by spectrophotometric analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
University Of Aarhus

Curated by ChEMBL
LigandPNGBDBM50222191(2-(3,4-dichlorophenyl)-N-(2-fluoroethyl)cyclopent-...)
Affinity DataKi:  8.00E+3nMAssay Description:Displacement of [125I]RTI55 from human NET transfected in COS1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
University Of Aarhus

Curated by ChEMBL
LigandPNGBDBM50222189(CHEMBL402924 | N-cyclobutyl-2-(3,4-dichlorophenyl)...)
Affinity DataKi:  9.00E+3nMAssay Description:Displacement of [125I]RTI55 from human DAT transfected in COS1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
University Of Aarhus

Curated by ChEMBL
LigandPNGBDBM50222182(2-hydroxyethyl 2-(3,4-dichlorophenyl)cyclopent-1-e...)
Affinity DataKi:  9.00E+3nMAssay Description:Displacement of [125I]RTI55 from human NET transfected in COS1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
University Of Aarhus

Curated by ChEMBL
LigandPNGBDBM50222185(2-(3,4-dichlorophenyl)-N-methoxycyclopent-1-enecar...)
Affinity DataKi:  9.20E+3nMAssay Description:Displacement of [125I]RTI55 from human NET transfected in COS1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
University Of Aarhus

Curated by ChEMBL
LigandPNGBDBM50222180((2-(3,4-dichlorophenyl)cyclopent-1-enyl)(morpholin...)
Affinity DataKi:  1.10E+4nMAssay Description:Displacement of [125I]RTI55 from human DAT transfected in COS1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
University Of Aarhus

Curated by ChEMBL
LigandPNGBDBM50211023(CHEMBL245061 | methyl 2-(3,4-dichlorophenyl)cyclop...)
Affinity DataKi:  1.10E+4nMAssay Description:Displacement of [125I]RTI55 from human NET transfected in COS1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
University Of Aarhus

Curated by ChEMBL
LigandPNGBDBM50222175(2-(3,4-dichlorophenyl)-N-(furan-2-ylmethyl)cyclope...)
Affinity DataKi:  1.20E+4nMAssay Description:Displacement of [125I]RTI55 from human NET transfected in COS1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
University Of Aarhus

Curated by ChEMBL
LigandPNGBDBM50222190(CHEMBL399430 | cyclohexyl 2-(3,4-dichlorophenyl)cy...)
Affinity DataKi:  1.20E+4nMAssay Description:Displacement of [125I]RTI55 from human DAT transfected in COS1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
University Of Aarhus

Curated by ChEMBL
LigandPNGBDBM50222184(2-(3,4-dichlorophenyl)-N-(thiophen-2-ylmethyl)cycl...)
Affinity DataKi:  1.80E+4nMAssay Description:Displacement of [125I]RTI55 from human NET transfected in COS1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
University Of Aarhus

Curated by ChEMBL
LigandPNGBDBM50222187(CHEMBL248825 | furan-2-ylmethyl 2-(3,4-dichlorophe...)
Affinity DataKi:  2.40E+4nMAssay Description:Displacement of [125I]RTI55 from human SERT transfected in COS1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
University Of Aarhus

Curated by ChEMBL
LigandPNGBDBM50222175(2-(3,4-dichlorophenyl)-N-(furan-2-ylmethyl)cyclope...)
Affinity DataKi:  2.40E+4nMAssay Description:Displacement of [125I]RTI55 from human SERT transfected in COS1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
University Of Aarhus

Curated by ChEMBL
LigandPNGBDBM50222176(CHEMBL401069 | isopropyl 2-(3,4-dichlorophenyl)cyc...)
Affinity DataKi:  2.60E+4nMAssay Description:Displacement of [125I]RTI55 from human NET transfected in COS1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
University Of Aarhus

Curated by ChEMBL
LigandPNGBDBM50222183(CHEMBL403570 | o-tolyl 2-(3,4-dichlorophenyl)cyclo...)
Affinity DataKi:  3.30E+4nMAssay Description:Displacement of [125I]RTI55 from human NET transfected in COS1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
University Of Aarhus

Curated by ChEMBL
LigandPNGBDBM50222178(CHEMBL403571 | thiophen-2-ylmethyl 2-(3,4-dichloro...)
Affinity DataKi:  4.20E+4nMAssay Description:Displacement of [125I]RTI55 from human NET transfected in COS1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-glucosidase(Prunus avium)
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50186735(CHEMBL208021 | D-1,4-dideoxy-4,4-difluoromannonoji...)
Affinity DataKi:  4.50E+4nMpH: 6.8Assay Description:Inhibition of almond beta glucosidase at pH 6.8More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
University Of Aarhus

Curated by ChEMBL
LigandPNGBDBM50222182(2-hydroxyethyl 2-(3,4-dichlorophenyl)cyclopent-1-e...)
Affinity DataKi:  5.00E+4nMAssay Description:Displacement of [125I]RTI55 from human SERT transfected in COS1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
University Of Aarhus

Curated by ChEMBL
LigandPNGBDBM50222189(CHEMBL402924 | N-cyclobutyl-2-(3,4-dichlorophenyl)...)
Affinity DataKi:  5.00E+4nMAssay Description:Displacement of [125I]RTI55 from human NET transfected in COS1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
University Of Aarhus

Curated by ChEMBL
LigandPNGBDBM50222181((2-(3,4-dichlorophenyl)cyclopent-1-enyl)(pyrrolidi...)
Affinity DataKi:  5.80E+4nMAssay Description:Displacement of [125I]RTI55 from human DAT transfected in COS1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
University Of Aarhus

Curated by ChEMBL
LigandPNGBDBM50222187(CHEMBL248825 | furan-2-ylmethyl 2-(3,4-dichlorophe...)
Affinity DataKi:  6.10E+4nMAssay Description:Displacement of [125I]RTI55 from human NET transfected in COS1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
University Of Aarhus

Curated by ChEMBL
LigandPNGBDBM50222188(CHEMBL401071 | phenyl 2-(3,4-dichlorophenyl)cyclop...)
Affinity DataKi:  8.50E+4nMAssay Description:Displacement of [125I]RTI55 from human NET transfected in COS1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-glucosidase(Prunus avium)
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50186735(CHEMBL208021 | D-1,4-dideoxy-4,4-difluoromannonoji...)
Affinity DataKi:  9.20E+4nMpH: 5.0Assay Description:Inhibition of almond beta glucosidase at pH 5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
University Of Aarhus

Curated by ChEMBL
LigandPNGBDBM50222174(2-(3,4-dichlorophenyl)-N,N-diethylcyclopent-1-enec...)
Affinity DataKi:  9.40E+4nMAssay Description:Displacement of [125I]RTI55 from human DAT transfected in COS1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
University Of Aarhus

Curated by ChEMBL
LigandPNGBDBM50222179(CHEMBL248824 | m-tolyl 2-(3,4-dichlorophenyl)cyclo...)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [125I]RTI55 from human NET transfected in COS1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
University Of Aarhus

Curated by ChEMBL
LigandPNGBDBM50222184(2-(3,4-dichlorophenyl)-N-(thiophen-2-ylmethyl)cycl...)
Affinity DataKi:  1.10E+5nMAssay Description:Displacement of [125I]RTI55 from human SERT transfected in COS1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
University Of Aarhus

Curated by ChEMBL
LigandPNGBDBM50222190(CHEMBL399430 | cyclohexyl 2-(3,4-dichlorophenyl)cy...)
Affinity DataKi:  1.30E+5nMAssay Description:Displacement of [125I]RTI55 from human NET transfected in COS1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
University Of Aarhus

Curated by ChEMBL
LigandPNGBDBM50222177(2,2,2-trifluoroethyl 2-(3,4-dichlorophenyl)cyclope...)
Affinity DataKi:  1.70E+5nMAssay Description:Displacement of [125I]RTI55 from human NET transfected in COS1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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