TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
University Of Aarhus
Curated by ChEMBL
University Of Aarhus
Curated by ChEMBL
Affinity DataKi: 30nMAssay Description:Displacement of [125I]RTI55 from human DAT transfected in COS1 cellsMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
University Of Aarhus
Curated by ChEMBL
University Of Aarhus
Curated by ChEMBL
Affinity DataKi: 60nMAssay Description:Displacement of [125I]RTI55 from human DAT transfected in COS1 cellsMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
University Of Aarhus
Curated by ChEMBL
University Of Aarhus
Curated by ChEMBL
Affinity DataKi: 70nMAssay Description:Displacement of [125I]RTI55 from human DAT transfected in COS1 cellsMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
University Of Aarhus
Curated by ChEMBL
University Of Aarhus
Curated by ChEMBL
Affinity DataKi: 140nMAssay Description:Displacement of [125I]RTI55 from human DAT transfected in COS1 cellsMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
University Of Aarhus
Curated by ChEMBL
University Of Aarhus
Curated by ChEMBL
Affinity DataKi: 170nMAssay Description:Displacement of [125I]RTI55 from human DAT transfected in COS1 cellsMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
University Of Aarhus
Curated by ChEMBL
University Of Aarhus
Curated by ChEMBL
Affinity DataKi: 220nMAssay Description:Displacement of [125I]RTI55 from human DAT transfected in COS1 cellsMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
University Of Aarhus
Curated by ChEMBL
University Of Aarhus
Curated by ChEMBL
Affinity DataKi: 300nMAssay Description:Displacement of [125I]RTI55 from human DAT transfected in COS1 cellsMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
University Of Aarhus
Curated by ChEMBL
University Of Aarhus
Curated by ChEMBL
Affinity DataKi: 400nMAssay Description:Displacement of [125I]RTI55 from human DAT transfected in COS1 cellsMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
University Of Aarhus
Curated by ChEMBL
University Of Aarhus
Curated by ChEMBL
Affinity DataKi: 500nMAssay Description:Displacement of [125I]RTI55 from human DAT transfected in COS1 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 500nMAssay Description:Inhibition of jack bean Lysosomal alpha-mannosidase assessed as residual hydrolytic activity after 10 to 30 mins by spectrophotometric analysisMore data for this Ligand-Target Pair
Affinity DataKi: 500nMAssay Description:Inhibition of jack bean Lysosomal alpha-mannosidase assessed as residual hydrolytic activity after 10 to 30 mins by spectrophotometric analysisMore data for this Ligand-Target Pair
Affinity DataKi: 500nMAssay Description:Inhibition of jack bean Lysosomal alpha-mannosidase assessed as residual hydrolytic activity after 10 to 30 mins by spectrophotometric analysisMore data for this Ligand-Target Pair
Affinity DataKi: 500nMAssay Description:Inhibition of jack bean Lysosomal alpha-mannosidase assessed as residual hydrolytic activity after 10 to 30 mins by spectrophotometric analysisMore data for this Ligand-Target Pair
Affinity DataKi: 500nMAssay Description:Inhibition of jack bean Lysosomal alpha-mannosidase assessed as residual hydrolytic activity after 10 to 30 mins by spectrophotometric analysisMore data for this Ligand-Target Pair
Affinity DataKi: 500nMAssay Description:Inhibition of jack bean Lysosomal alpha-mannosidase assessed as residual hydrolytic activity after 10 to 30 mins by spectrophotometric analysisMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
University Of Aarhus
Curated by ChEMBL
University Of Aarhus
Curated by ChEMBL
Affinity DataKi: 830nMAssay Description:Displacement of [125I]RTI55 from human DAT transfected in COS1 cellsMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
University Of Aarhus
Curated by ChEMBL
University Of Aarhus
Curated by ChEMBL
Affinity DataKi: 1.50E+3nMAssay Description:Displacement of [125I]RTI55 from human DAT transfected in COS1 cellsMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
University Of Aarhus
Curated by ChEMBL
University Of Aarhus
Curated by ChEMBL
Affinity DataKi: 1.90E+3nMAssay Description:Displacement of [125I]RTI55 from human DAT transfected in COS1 cellsMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
University Of Aarhus
Curated by ChEMBL
University Of Aarhus
Curated by ChEMBL
Affinity DataKi: 2.60E+3nMAssay Description:Displacement of [125I]RTI55 from human DAT transfected in COS1 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 3.20E+3nMAssay Description:Inhibition of jack bean Lysosomal alpha-mannosidase assessed as residual hydrolytic activity after 10 to 30 mins by spectrophotometric analysisMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
University Of Aarhus
Curated by ChEMBL
University Of Aarhus
Curated by ChEMBL
Affinity DataKi: 3.40E+3nMAssay Description:Displacement of [125I]RTI55 from human DAT transfected in COS1 cellsMore data for this Ligand-Target Pair
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
University Of Aarhus
Curated by ChEMBL
University Of Aarhus
Curated by ChEMBL
Affinity DataKi: 5.80E+3nMAssay Description:Displacement of [125I]RTI55 from human NET transfected in COS1 cellsMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
University Of Aarhus
Curated by ChEMBL
University Of Aarhus
Curated by ChEMBL
Affinity DataKi: 6.40E+3nMAssay Description:Displacement of [125I]RTI55 from human DAT transfected in COS1 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 7.00E+3nMAssay Description:Inhibition of jack bean Lysosomal alpha-mannosidase assessed as residual hydrolytic activity after 10 to 30 mins by spectrophotometric analysisMore data for this Ligand-Target Pair
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
University Of Aarhus
Curated by ChEMBL
University Of Aarhus
Curated by ChEMBL
Affinity DataKi: 8.00E+3nMAssay Description:Displacement of [125I]RTI55 from human NET transfected in COS1 cellsMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
University Of Aarhus
Curated by ChEMBL
University Of Aarhus
Curated by ChEMBL
Affinity DataKi: 9.00E+3nMAssay Description:Displacement of [125I]RTI55 from human DAT transfected in COS1 cellsMore data for this Ligand-Target Pair
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
University Of Aarhus
Curated by ChEMBL
University Of Aarhus
Curated by ChEMBL
Affinity DataKi: 9.00E+3nMAssay Description:Displacement of [125I]RTI55 from human NET transfected in COS1 cellsMore data for this Ligand-Target Pair
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
University Of Aarhus
Curated by ChEMBL
University Of Aarhus
Curated by ChEMBL
Affinity DataKi: 9.20E+3nMAssay Description:Displacement of [125I]RTI55 from human NET transfected in COS1 cellsMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
University Of Aarhus
Curated by ChEMBL
University Of Aarhus
Curated by ChEMBL
Affinity DataKi: 1.10E+4nMAssay Description:Displacement of [125I]RTI55 from human DAT transfected in COS1 cellsMore data for this Ligand-Target Pair
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
University Of Aarhus
Curated by ChEMBL
University Of Aarhus
Curated by ChEMBL
Affinity DataKi: 1.10E+4nMAssay Description:Displacement of [125I]RTI55 from human NET transfected in COS1 cellsMore data for this Ligand-Target Pair
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
University Of Aarhus
Curated by ChEMBL
University Of Aarhus
Curated by ChEMBL
Affinity DataKi: 1.20E+4nMAssay Description:Displacement of [125I]RTI55 from human NET transfected in COS1 cellsMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
University Of Aarhus
Curated by ChEMBL
University Of Aarhus
Curated by ChEMBL
Affinity DataKi: 1.20E+4nMAssay Description:Displacement of [125I]RTI55 from human DAT transfected in COS1 cellsMore data for this Ligand-Target Pair
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
University Of Aarhus
Curated by ChEMBL
University Of Aarhus
Curated by ChEMBL
Affinity DataKi: 1.80E+4nMAssay Description:Displacement of [125I]RTI55 from human NET transfected in COS1 cellsMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
University Of Aarhus
Curated by ChEMBL
University Of Aarhus
Curated by ChEMBL
Affinity DataKi: 2.40E+4nMAssay Description:Displacement of [125I]RTI55 from human SERT transfected in COS1 cellsMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
University Of Aarhus
Curated by ChEMBL
University Of Aarhus
Curated by ChEMBL
Affinity DataKi: 2.40E+4nMAssay Description:Displacement of [125I]RTI55 from human SERT transfected in COS1 cellsMore data for this Ligand-Target Pair
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
University Of Aarhus
Curated by ChEMBL
University Of Aarhus
Curated by ChEMBL
Affinity DataKi: 2.60E+4nMAssay Description:Displacement of [125I]RTI55 from human NET transfected in COS1 cellsMore data for this Ligand-Target Pair
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
University Of Aarhus
Curated by ChEMBL
University Of Aarhus
Curated by ChEMBL
Affinity DataKi: 3.30E+4nMAssay Description:Displacement of [125I]RTI55 from human NET transfected in COS1 cellsMore data for this Ligand-Target Pair
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
University Of Aarhus
Curated by ChEMBL
University Of Aarhus
Curated by ChEMBL
Affinity DataKi: 4.20E+4nMAssay Description:Displacement of [125I]RTI55 from human NET transfected in COS1 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 4.50E+4nMpH: 6.8Assay Description:Inhibition of almond beta glucosidase at pH 6.8More data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
University Of Aarhus
Curated by ChEMBL
University Of Aarhus
Curated by ChEMBL
Affinity DataKi: 5.00E+4nMAssay Description:Displacement of [125I]RTI55 from human SERT transfected in COS1 cellsMore data for this Ligand-Target Pair
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
University Of Aarhus
Curated by ChEMBL
University Of Aarhus
Curated by ChEMBL
Affinity DataKi: 5.00E+4nMAssay Description:Displacement of [125I]RTI55 from human NET transfected in COS1 cellsMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
University Of Aarhus
Curated by ChEMBL
University Of Aarhus
Curated by ChEMBL
Affinity DataKi: 5.80E+4nMAssay Description:Displacement of [125I]RTI55 from human DAT transfected in COS1 cellsMore data for this Ligand-Target Pair
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
University Of Aarhus
Curated by ChEMBL
University Of Aarhus
Curated by ChEMBL
Affinity DataKi: 6.10E+4nMAssay Description:Displacement of [125I]RTI55 from human NET transfected in COS1 cellsMore data for this Ligand-Target Pair
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
University Of Aarhus
Curated by ChEMBL
University Of Aarhus
Curated by ChEMBL
Affinity DataKi: 8.50E+4nMAssay Description:Displacement of [125I]RTI55 from human NET transfected in COS1 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 9.20E+4nMpH: 5.0Assay Description:Inhibition of almond beta glucosidase at pH 5More data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
University Of Aarhus
Curated by ChEMBL
University Of Aarhus
Curated by ChEMBL
Affinity DataKi: 9.40E+4nMAssay Description:Displacement of [125I]RTI55 from human DAT transfected in COS1 cellsMore data for this Ligand-Target Pair
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
University Of Aarhus
Curated by ChEMBL
University Of Aarhus
Curated by ChEMBL
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [125I]RTI55 from human NET transfected in COS1 cellsMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
University Of Aarhus
Curated by ChEMBL
University Of Aarhus
Curated by ChEMBL
Affinity DataKi: 1.10E+5nMAssay Description:Displacement of [125I]RTI55 from human SERT transfected in COS1 cellsMore data for this Ligand-Target Pair
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
University Of Aarhus
Curated by ChEMBL
University Of Aarhus
Curated by ChEMBL
Affinity DataKi: 1.30E+5nMAssay Description:Displacement of [125I]RTI55 from human NET transfected in COS1 cellsMore data for this Ligand-Target Pair
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
University Of Aarhus
Curated by ChEMBL
University Of Aarhus
Curated by ChEMBL
Affinity DataKi: 1.70E+5nMAssay Description:Displacement of [125I]RTI55 from human NET transfected in COS1 cellsMore data for this Ligand-Target Pair