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Found 50 with Last Name = 'pearson' and Initial = 'n'
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50359538(CHEMBL1235773)
Affinity DataIC50:  500nMAssay Description:Displacement of [3H]dofetilide from human ERG by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50359538(CHEMBL1235773)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of human ERG expressed in HEK293 cells by patch-clamp electrophysiologyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50359535(CHEMBL1927163)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of human ERG expressed in HEK293 cells by patch-clamp electrophysiologyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50359457(CHEMBL1926867)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of human ERG by whole cell patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50359535(CHEMBL1927163)
Affinity DataIC50:  2.00E+3nMAssay Description:Displacement of [3H]dofetilide from human ERG by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50359537(CHEMBL1927167)
Affinity DataIC50:  3.00E+3nMAssay Description:Inhibition of human ERG expressed in HEK293 cells by patch-clamp electrophysiologyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50359540(CHEMBL1927161)
Affinity DataIC50:  4.00E+3nMAssay Description:Inhibition of human ERG expressed in HEK293 cells by patch-clamp electrophysiologyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50359544(CHEMBL1927168)
Affinity DataIC50:  4.90E+3nMAssay Description:Displacement of [3H]dofetilide from human ERG by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50359541(CHEMBL1927162)
Affinity DataIC50:  5.00E+3nMAssay Description:Displacement of [3H]dofetilide from human ERG by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50359536(CHEMBL1927165)
Affinity DataIC50:  5.00E+3nMAssay Description:Inhibition of human ERG expressed in HEK293 cells by patch-clamp electrophysiologyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50359541(CHEMBL1927162)
Affinity DataIC50:  6.00E+3nMAssay Description:Inhibition of human ERG expressed in HEK293 cells by patch-clamp electrophysiologyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50359542(CHEMBL1927164)
Affinity DataIC50:  7.90E+3nMAssay Description:Displacement of [3H]dofetilide from human ERG by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50359537(CHEMBL1927167)
Affinity DataIC50:  7.90E+3nMAssay Description:Displacement of [3H]dofetilide from human ERG by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50357934(CHEMBL1916532)
Affinity DataIC50:  1.51E+4nMAssay Description:Displacement of [3H]dofetilide from human ERG by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50493332(CHEMBL2424930)
Affinity DataIC50:  1.60E+4nMAssay Description:Inhibition of human ERG by patch clamp assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCytochrome P450 2D6(Homo sapiens (Human))
Merck Healthcare

Curated by ChEMBL
LigandPNGBDBM50600846(CHEMBL5170406)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of CYP2D6 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))
Merck Healthcare

Curated by ChEMBL
LigandPNGBDBM50600846(CHEMBL5170406)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of CYP3A4 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCytochrome P450 2C19(Homo sapiens)
Merck Healthcare

Curated by ChEMBL
LigandPNGBDBM50600846(CHEMBL5170406)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of CYP2C19 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCytochrome P450 2C9(Homo sapiens (Human))
Merck Healthcare

Curated by ChEMBL
LigandPNGBDBM50600846(CHEMBL5170406)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of CYP2C9 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCytochrome P450 2C8(Homo sapiens (Human))
Merck Healthcare

Curated by ChEMBL
LigandPNGBDBM50600846(CHEMBL5170406)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of CYP2C8 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCytochrome P450 2B6(Homo sapiens (Human))
Merck Healthcare

Curated by ChEMBL
LigandPNGBDBM50600846(CHEMBL5170406)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of CYP2B6 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCytochrome P450 1A2(Homo sapiens (Human))
Merck Healthcare

Curated by ChEMBL
LigandPNGBDBM50600846(CHEMBL5170406)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of CYP1A2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50359451(CHEMBL1926763)
Affinity DataIC50:  2.40E+4nMAssay Description:Inhibition of human ERG by whole cell patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50359450(CHEMBL1926762)
Affinity DataIC50:  2.50E+4nMAssay Description:Inhibition of human ERG by whole cell patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50359452(CHEMBL1926765)
Affinity DataIC50:  2.50E+4nMAssay Description:Inhibition of human ERG by whole cell patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50359540(CHEMBL1927161)
Affinity DataIC50:  2.51E+4nMAssay Description:Displacement of [3H]dofetilide from human ERG by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50359454(CHEMBL1926864)
Affinity DataIC50:  2.90E+4nMAssay Description:Inhibition of human ERG by whole cell patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50359545(CHEMBL1927170)
Affinity DataIC50:  2.95E+4nMAssay Description:Displacement of [3H]dofetilide from human ERG by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50359539(CHEMBL548279)
Affinity DataIC50:  3.98E+4nMAssay Description:Displacement of [3H]dofetilide from human ERG by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50156567(CHEMBL3794265)
Affinity DataIC50:  4.20E+4nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50359453(CHEMBL1926766)
Affinity DataIC50:  5.20E+4nMAssay Description:Inhibition of human ERG by whole cell patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50493331(CHEMBL2424931)
Affinity DataIC50:  5.80E+4nMAssay Description:Inhibition of human ERG by patch clamp assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50359543(CHEMBL1927166)
Affinity DataIC50:  6.31E+4nMAssay Description:Displacement of [3H]dofetilide from human ERG by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50359536(CHEMBL1927165)
Affinity DataIC50:  7.94E+4nMAssay Description:Displacement of [3H]dofetilide from human ERG by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50493330(CHEMBL2424933)
Affinity DataIC50:  1.01E+5nMAssay Description:Inhibition of human ERG by patch clamp assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50359455(CHEMBL1926865)
Affinity DataIC50:  1.13E+5nMAssay Description:Inhibition of human ERG by whole cell patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50493331(CHEMBL2424931)
Affinity DataIC50:  1.22E+5nMAssay Description:Inhibition of human ERG transfected in HEK293 cells by patch clamp assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50359456(CHEMBL1926866)
Affinity DataIC50:  2.00E+5nMAssay Description:Inhibition of human ERG by whole cell patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50493330(CHEMBL2424933)
Affinity DataIC50:  2.06E+5nMAssay Description:Inhibition of human ERG transfected in HEK293 cells by patch clamp assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50156545(CHEMBL3793226)
Affinity DataIC50:  2.38E+5nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50254157(CHEMBL2424928)
Affinity DataIC50:  2.39E+5nMAssay Description:Inhibition of human ERG by patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50493333(CHEMBL2424934)
Affinity DataIC50:  2.89E+5nMAssay Description:Inhibition of human ERG by patch clamp assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50254157(CHEMBL2424928)
Affinity DataIC50:  3.10E+5nMAssay Description:Inhibition of human ERG transfected in HEK293 cells by patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscriptional enhancer factor TEF-1(Homo sapiens)
Merck Healthcare

Curated by ChEMBL
LigandPNGBDBM50600845(CHEMBL5173440)
Affinity DataKd:  5.80E+3nMAssay Description:Binding affinity to human TEAD1 (209 to 426 residues) expressed in Escherichia coli BL21 Star (DE3) by surface plasmon resonance assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetTranscriptional enhancer factor TEF-4(Homo sapiens)
Merck Healthcare

Curated by ChEMBL
LigandPNGBDBM50600846(CHEMBL5170406)
Affinity DataKd:  4.60E+3nMAssay Description:Binding affinity to human TEAD2 (217 to 447 residues) expressed in Escherichia coli BL21 Star (DE3) by surface plasmon resonance assayMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetTranscriptional enhancer factor TEF-5(Homo sapiens)
Merck Healthcare

Curated by ChEMBL
LigandPNGBDBM50600846(CHEMBL5170406)
Affinity DataKd:  1.40E+3nMAssay Description:Binding affinity to human TEAD3 (216 to 435 residues) expressed in Escherichia coli BL21 Star (DE3) by surface plasmon resonance assayMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetTranscriptional enhancer factor TEF-1(Homo sapiens)
Merck Healthcare

Curated by ChEMBL
LigandPNGBDBM50600846(CHEMBL5170406)
Affinity DataKd:  120nMAssay Description:Binding affinity to human TEAD1 (209 to 426 residues) expressed in Escherichia coli BL21 Star (DE3) by surface plasmon resonance assayMore data for this Ligand-Target Pair
TargetTranscriptional enhancer factor TEF-3(Homo sapiens)
Merck Healthcare

Curated by ChEMBL
LigandPNGBDBM50600846(CHEMBL5170406)
Affinity DataKd:  5.40E+3nMAssay Description:Binding affinity to human TEAD4 (217 to 434 residues) expressed in Escherichia coli BL21 Star (DE3) by surface plasmon resonance assayMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetTranscriptional enhancer factor TEF-3(Homo sapiens)
Merck Healthcare

Curated by ChEMBL
LigandPNGBDBM50600845(CHEMBL5173440)
Affinity DataKd:  7.60E+3nMAssay Description:Binding affinity to human TEAD4 (217 to 434 residues) expressed in Escherichia coli BL21 Star (DE3) by surface plasmon resonance assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetTranscriptional enhancer factor TEF-4(Homo sapiens)
Merck Healthcare

Curated by ChEMBL
LigandPNGBDBM50600845(CHEMBL5173440)
Affinity DataKd:  4.30E+4nMAssay Description:Binding affinity to human TEAD2 (217 to 447 residues) expressed in Escherichia coli BL21 Star (DE3) by surface plasmon resonance assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed