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Found 42 with Last Name = 'reverchon' and Initial = 's'
TargetTranscriptional activator protein LuxR(Vibrio fischeri)
Insa Lyon

Curated by ChEMBL
LigandPNGBDBM50350660(CHEMBL1813552)
Affinity DataIC50:  1.40E+3nMAssay Description:Antagonist activity at Vibrio fischeri LuxR assessed as inhibition of 3-oxo-C6-HSL-induced quorum sensing activation mediated bioluminescenceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscriptional activator protein LuxR(Vibrio fischeri)
Insa Lyon

Curated by ChEMBL
LigandPNGBDBM50373056(CHEMBL261163)
Affinity DataIC50:  2.00E+3nMAssay Description:Antagonist activity at LuxR in Vibrio fischeri assessed as inhibition of N-3-oxos-hexanoyl-L-homoserine lactone induced luminescenceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscriptional activator protein LuxR(Vibrio fischeri)
Insa Lyon

Curated by ChEMBL
LigandPNGBDBM50350661(CHEMBL1813553)
Affinity DataIC50:  2.70E+3nMAssay Description:Antagonist activity at Vibrio fischeri LuxR assessed as inhibition of 3-oxo-C6-HSL-induced quorum sensing activation mediated bioluminescenceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscriptional activator protein LuxR(Vibrio fischeri)
Insa Lyon

Curated by ChEMBL
LigandPNGBDBM50373048(CHEMBL184106)
Affinity DataIC50:  3.00E+3nMAssay Description:Antagonist activity at LuxR in Vibrio fischeri assessed as inhibition of N-3-oxos-hexanoyl-L-homoserine lactone induced luminescenceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscriptional activator protein LuxR(Vibrio fischeri)
Insa Lyon

Curated by ChEMBL
LigandPNGBDBM50350666(CHEMBL1813558)
Affinity DataIC50:  3.40E+3nMAssay Description:Antagonist activity at Vibrio fischeri LuxR assessed as inhibition of 3-oxo-C6-HSL-induced quorum sensing activation mediated bioluminescenceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscriptional activator protein LuxR(Vibrio fischeri)
Insa Lyon

Curated by ChEMBL
LigandPNGBDBM50373057(CHEMBL261162)
Affinity DataIC50:  3.60E+3nMAssay Description:Antagonist activity at LuxR in Vibrio fischeri assessed as inhibition of N-3-oxos-hexanoyl-L-homoserine lactone induced luminescenceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscriptional activator protein LuxR(Vibrio fischeri)
Insa Lyon

Curated by ChEMBL
LigandPNGBDBM50350659(CHEMBL1813551)
Affinity DataIC50:  4.00E+3nMAssay Description:Antagonist activity at Vibrio fischeri LuxR assessed as inhibition of 3-oxo-C6-HSL-induced quorum sensing activation mediated bioluminescenceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscriptional activator protein LuxR(Vibrio fischeri)
Insa Lyon

Curated by ChEMBL
LigandPNGBDBM50350669(CHEMBL1813546)
Affinity DataIC50:  4.90E+3nMAssay Description:Antagonist activity at Vibrio fischeri LuxR assessed as inhibition of 3-oxo-C6-HSL-induced quorum sensing activation mediated bioluminescenceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscriptional activator protein LuxR(Vibrio fischeri)
Insa Lyon

Curated by ChEMBL
LigandPNGBDBM50373055(CHEMBL408369)
Affinity DataIC50:  5.00E+3nMAssay Description:Antagonist activity at LuxR in Vibrio fischeri assessed as inhibition of N-3-oxos-hexanoyl-L-homoserine lactone induced luminescenceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscriptional activator protein LuxR(Vibrio fischeri)
Insa Lyon

Curated by ChEMBL
LigandPNGBDBM50373047(CHEMBL260235)
Affinity DataIC50:  5.00E+3nMAssay Description:Antagonist activity at LuxR in Vibrio fischeri assessed as inhibition of N-3-oxos-hexanoyl-L-homoserine lactone induced luminescenceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscriptional activator protein LuxR(Vibrio fischeri)
Insa Lyon

Curated by ChEMBL
LigandPNGBDBM50350649(CHEMBL1813536)
Affinity DataIC50:  5.20E+3nMAssay Description:Antagonist activity at Vibrio fischeri LuxR assessed as inhibition of 3-oxo-C6-HSL-induced quorum sensing activation mediated bioluminescenceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscriptional activator protein LuxR(Vibrio fischeri)
Insa Lyon

Curated by ChEMBL
LigandPNGBDBM50350670(CHEMBL1813559)
Affinity DataIC50:  5.30E+3nMAssay Description:Antagonist activity at Vibrio fischeri LuxR assessed as inhibition of 3-oxo-C6-HSL-induced quorum sensing activation mediated bioluminescenceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscriptional activator protein LuxR(Vibrio fischeri)
Insa Lyon

Curated by ChEMBL
LigandPNGBDBM50350653(CHEMBL1813540)
Affinity DataIC50:  5.80E+3nMAssay Description:Antagonist activity at Vibrio fischeri LuxR assessed as inhibition of 3-oxo-C6-HSL-induced quorum sensing activation mediated bioluminescenceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscriptional activator protein LuxR(Vibrio fischeri)
Insa Lyon

Curated by ChEMBL
LigandPNGBDBM50350648(CHEMBL1813535)
Affinity DataIC50:  6.10E+3nMAssay Description:Antagonist activity at Vibrio fischeri LuxR assessed as inhibition of 3-oxo-C6-HSL-induced quorum sensing activation mediated bioluminescenceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscriptional activator protein LuxR(Vibrio fischeri)
Insa Lyon

Curated by ChEMBL
LigandPNGBDBM50350654(CHEMBL1813541)
Affinity DataIC50:  6.20E+3nMAssay Description:Antagonist activity at Vibrio fischeri LuxR assessed as inhibition of 3-oxo-C6-HSL-induced quorum sensing activation mediated bioluminescenceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscriptional activator protein LuxR(Vibrio fischeri)
Insa Lyon

Curated by ChEMBL
LigandPNGBDBM50373052(CHEMBL404926)
Affinity DataIC50:  6.40E+3nMAssay Description:Antagonist activity at LuxR in Vibrio fischeri assessed as inhibition of N-3-oxos-hexanoyl-L-homoserine lactone induced luminescenceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscriptional activator protein LuxR(Vibrio fischeri)
Insa Lyon

Curated by ChEMBL
LigandPNGBDBM50262515(CHEMBL453930 | N-(4-bromo-2-oxo-2,5-dihydrofuran-3...)
Affinity DataIC50:  6.50E+3nMAssay Description:Inhibition of LuxR-dependent Vibrio fischeri quorum sensing assessed as reduction in 3-oxo-hexanoyihomoserine-induced bioluminescenceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscriptional activator protein LuxR(Vibrio fischeri)
Insa Lyon

Curated by ChEMBL
LigandPNGBDBM50350657(CHEMBL1813547)
Affinity DataIC50:  6.50E+3nMAssay Description:Antagonist activity at Vibrio fischeri LuxR assessed as inhibition of 3-oxo-C6-HSL-induced quorum sensing activation mediated bioluminescenceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscriptional activator protein LuxR(Vibrio fischeri)
Insa Lyon

Curated by ChEMBL
LigandPNGBDBM50262517(CHEMBL448263 | N-(4-chloro-2-oxo-2,5-dihydrofuran-...)
Affinity DataIC50:  6.90E+3nMAssay Description:Inhibition of LuxR-dependent Vibrio fischeri quorum sensing assessed as reduction in 3-oxo-hexanoyihomoserine-induced bioluminescenceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscriptional activator protein LuxR(Vibrio fischeri)
Insa Lyon

Curated by ChEMBL
LigandPNGBDBM50373054(CHEMBL408296)
Affinity DataIC50:  7.20E+3nMAssay Description:Antagonist activity at LuxR in Vibrio fischeri assessed as inhibition of N-3-oxos-hexanoyl-L-homoserine lactone induced luminescenceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscriptional activator protein LuxR(Vibrio fischeri)
Insa Lyon

Curated by ChEMBL
LigandPNGBDBM50350650(CHEMBL1813537)
Affinity DataIC50:  7.30E+3nMAssay Description:Antagonist activity at Vibrio fischeri LuxR assessed as inhibition of 3-oxo-C6-HSL-induced quorum sensing activation mediated bioluminescenceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscriptional activator protein LuxR(Vibrio fischeri)
Insa Lyon

Curated by ChEMBL
LigandPNGBDBM50373053(CHEMBL260905)
Affinity DataIC50:  7.80E+3nMAssay Description:Antagonist activity at LuxR in Vibrio fischeri assessed as inhibition of N-3-oxos-hexanoyl-L-homoserine lactone induced luminescenceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscriptional activator protein LuxR(Vibrio fischeri)
Insa Lyon

Curated by ChEMBL
LigandPNGBDBM50350668(CHEMBL1813545)
Affinity DataIC50:  8.90E+3nMAssay Description:Antagonist activity at Vibrio fischeri LuxR assessed as inhibition of 3-oxo-C6-HSL-induced quorum sensing activation mediated bioluminescenceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscriptional activator protein LuxR(Vibrio fischeri)
Insa Lyon

Curated by ChEMBL
LigandPNGBDBM50373050(CHEMBL258584)
Affinity DataIC50:  9.40E+3nMAssay Description:Antagonist activity at LuxR in Vibrio fischeri assessed as inhibition of N-3-oxos-hexanoyl-L-homoserine lactone induced luminescenceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscriptional activator protein LuxR(Vibrio fischeri)
Insa Lyon

Curated by ChEMBL
LigandPNGBDBM50350652(CHEMBL1813539)
Affinity DataIC50:  9.80E+3nMAssay Description:Antagonist activity at Vibrio fischeri LuxR assessed as inhibition of 3-oxo-C6-HSL-induced quorum sensing activation mediated bioluminescenceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscriptional activator protein LuxR(Vibrio fischeri)
Insa Lyon

Curated by ChEMBL
LigandPNGBDBM50350665(CHEMBL1813557)
Affinity DataIC50:  1.10E+4nMAssay Description:Antagonist activity at Vibrio fischeri LuxR assessed as inhibition of 3-oxo-C6-HSL-induced quorum sensing activation mediated bioluminescenceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscriptional activator protein LuxR(Vibrio fischeri)
Insa Lyon

Curated by ChEMBL
LigandPNGBDBM50373051(CHEMBL404924)
Affinity DataIC50:  1.30E+4nMAssay Description:Antagonist activity at LuxR in Vibrio fischeri assessed as inhibition of N-3-oxos-hexanoyl-L-homoserine lactone induced luminescenceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscriptional activator protein LuxR(Vibrio fischeri)
Insa Lyon

Curated by ChEMBL
LigandPNGBDBM50373049(CHEMBL408121)
Affinity DataIC50:  1.30E+4nMAssay Description:Antagonist activity at LuxR in Vibrio fischeri assessed as inhibition of N-3-oxos-hexanoyl-L-homoserine lactone induced luminescenceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscriptional activator protein LuxR(Vibrio fischeri)
Insa Lyon

Curated by ChEMBL
LigandPNGBDBM50350662(CHEMBL1813554)
Affinity DataIC50:  1.47E+4nMAssay Description:Antagonist activity at Vibrio fischeri LuxR assessed as inhibition of 3-oxo-C6-HSL-induced quorum sensing activation mediated bioluminescenceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscriptional activator protein LuxR(Vibrio fischeri)
Insa Lyon

Curated by ChEMBL
LigandPNGBDBM50350647(CHEMBL1813534)
Affinity DataIC50:  1.80E+4nMAssay Description:Antagonist activity at Vibrio fischeri LuxR assessed as inhibition of 3-oxo-C6-HSL-induced quorum sensing activation mediated bioluminescenceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscriptional activator protein LuxR(Vibrio fischeri)
Insa Lyon

Curated by ChEMBL
LigandPNGBDBM50350664(CHEMBL1813556)
Affinity DataIC50:  3.30E+4nMAssay Description:Antagonist activity at Vibrio fischeri LuxR assessed as inhibition of 3-oxo-C6-HSL-induced quorum sensing activation mediated bioluminescenceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscriptional activator protein LuxR(Vibrio fischeri)
Insa Lyon

Curated by ChEMBL
LigandPNGBDBM50350658(CHEMBL1813550)
Affinity DataIC50:  3.50E+4nMAssay Description:Antagonist activity at Vibrio fischeri LuxR assessed as inhibition of 3-oxo-C6-HSL-induced quorum sensing activation mediated bioluminescenceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscriptional activator protein LuxR(Vibrio fischeri)
Insa Lyon

Curated by ChEMBL
LigandPNGBDBM50350656(CHEMBL1813544)
Affinity DataIC50:  5.20E+4nMAssay Description:Antagonist activity at Vibrio fischeri LuxR assessed as inhibition of 3-oxo-C6-HSL-induced quorum sensing activation mediated bioluminescenceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscriptional activator protein LuxR(Vibrio fischeri)
Insa Lyon

Curated by ChEMBL
LigandPNGBDBM50262465(3-oxo-N-(2-oxo-2,5-dihydrofuran-3-yl)hexanamide | ...)
Affinity DataIC50:  5.50E+4nMAssay Description:Inhibition of LuxR-dependent Vibrio fischeri quorum sensing assessed as reduction in 3-oxo-hexanoyihomoserine-induced bioluminescenceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscriptional activator protein LuxR(Vibrio fischeri)
Insa Lyon

Curated by ChEMBL
LigandPNGBDBM50350651(CHEMBL1813538)
Affinity DataIC50:  6.30E+4nMAssay Description:Antagonist activity at Vibrio fischeri LuxR assessed as inhibition of 3-oxo-C6-HSL-induced quorum sensing activation mediated bioluminescenceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscriptional activator protein LuxR(Vibrio fischeri)
Insa Lyon

Curated by ChEMBL
LigandPNGBDBM50350663(CHEMBL1813555)
Affinity DataIC50:  6.80E+4nMAssay Description:Antagonist activity at Vibrio fischeri LuxR assessed as inhibition of 3-oxo-C6-HSL-induced quorum sensing activation mediated bioluminescenceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscriptional activator protein LuxR(Vibrio fischeri)
Insa Lyon

Curated by ChEMBL
LigandPNGBDBM50350655(CHEMBL1813542)
Affinity DataIC50:  7.50E+4nMAssay Description:Antagonist activity at Vibrio fischeri LuxR assessed as inhibition of 3-oxo-C6-HSL-induced quorum sensing activation mediated bioluminescenceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscriptional activator protein LuxR(Vibrio fischeri)
Insa Lyon

Curated by ChEMBL
LigandPNGBDBM50350646(CHEMBL1813533)
Affinity DataIC50:  7.60E+4nMAssay Description:Antagonist activity at Vibrio fischeri LuxR assessed as inhibition of 3-oxo-C6-HSL-induced quorum sensing activation mediated bioluminescenceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscriptional activator protein LuxR(Vibrio fischeri)
Insa Lyon

Curated by ChEMBL
LigandPNGBDBM50262516(CHEMBL478391 | N-(4-bromo-2-oxo-2,5-dihydrofuran-3...)
Affinity DataIC50:  8.40E+4nMAssay Description:Inhibition of LuxR-dependent Vibrio fischeri quorum sensing assessed as reduction in 3-oxo-hexanoyihomoserine-induced bioluminescenceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscriptional activator protein LuxR(Vibrio fischeri)
Insa Lyon

Curated by ChEMBL
LigandPNGBDBM50262464(CHEMBL478634 | N-(2-oxo-2,5-dihydrofuran-3-yl)hexa...)
Affinity DataIC50:  8.50E+4nMAssay Description:Inhibition of LuxR-dependent Vibrio fischeri quorum sensing assessed as reduction in 3-oxo-hexanoyihomoserine-induced bioluminescenceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscriptional activator protein LuxR(Vibrio fischeri)
Insa Lyon

Curated by ChEMBL
LigandPNGBDBM50350667(CHEMBL1813560)
Affinity DataIC50:  8.60E+4nMAssay Description:Antagonist activity at Vibrio fischeri LuxR assessed as inhibition of 3-oxo-C6-HSL-induced quorum sensing activation mediated bioluminescenceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscriptional activator protein LuxR(Vibrio fischeri)
Insa Lyon

Curated by ChEMBL
LigandPNGBDBM50350645(CHEMBL1813532)
Affinity DataIC50:  1.53E+5nMAssay Description:Antagonist activity at Vibrio fischeri LuxR assessed as inhibition of 3-oxo-C6-HSL-induced quorum sensing activation mediated bioluminescenceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed