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Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
5
hits in this display
Target
Suppressor of tumorigenicity 14 protein
(Homo sapiens (Human))
Curacyte Chemistry
Ligand
BDBM23883
(3-[(2S)-3-[4-(3-carbamimidamidopropanoyl)piperazin...)
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Affinity Data
Ki: 400nM ΔG°: -36.5kJ/mole
pH: 8.0 T: 2°C
Assay Description:
The measurements were carried out on a microplate reader. Two concentrations of the substrate and five concentrations of the inhibitor were used. Af...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
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Target
Prothrombin
(Bos taurus (Bovine))
Curacyte Chemistry
Ligand
BDBM23883
(3-[(2S)-3-[4-(3-carbamimidamidopropanoyl)piperazin...)
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Affinity Data
Ki: 2.60E+3nM
Assay Description:
The measurements were carried out on a microplate reader. Two concentrations of the substrate and five concentrations of the inhibitor were used. Af...
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
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Target
Plasminogen
(Homo sapiens (Human))
Curacyte Chemistry
Ligand
BDBM23883
(3-[(2S)-3-[4-(3-carbamimidamidopropanoyl)piperazin...)
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Affinity Data
Ki: 1.20E+4nM
Assay Description:
The measurements were carried out on a microplate reader. Two concentrations of the substrate and five concentrations of the inhibitor were used. Af...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
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Target
Urokinase-type plasminogen activator
(Homo sapiens (Human))
Curacyte Chemistry
Ligand
BDBM23883
(3-[(2S)-3-[4-(3-carbamimidamidopropanoyl)piperazin...)
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Affinity Data
Ki: 4.30E+4nM
Assay Description:
The measurements were carried out on a microplate reader. Two concentrations of the substrate and five concentrations of the inhibitor were used. Af...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
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Target
Coagulation factor X
(Bos taurus)
Curacyte Chemistry
Ligand
BDBM23883
(3-[(2S)-3-[4-(3-carbamimidamidopropanoyl)piperazin...)
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Affinity Data
Ki: 1.30E+5nM
Assay Description:
The measurements were carried out on a microplate reader. Two concentrations of the substrate and five concentrations of the inhibitor were used. Af...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
GoogleScholar
Ligand Info
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI