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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 7 hits in this display   

TargetKappa-type opioid receptor(Mus musculus (Mouse))
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50095703(3-But-3-enyl-6,11-dimethyl-1,2,3,4,5,6-hexahydro-2...)
Affinity DataKi:  1.30nMAssay Description:Ki value determined against Opioid receptor kappa 1 using [3H]U69, 593 at the Kd concentration 0.95 nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Macaca mulatta)
University Of Catania

Curated by ChEMBL
LigandPNGBDBM50458148(CHEMBL4214248)
Affinity DataKi:  1.30nMAssay Description:Displacement of [3H]U69,593 from KOR in monkey brain cortex membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(MOUSE)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50095703(3-But-3-enyl-6,11-dimethyl-1,2,3,4,5,6-hexahydro-2...)
Affinity DataKi:  2.10nMAssay Description:Ki value determined against Opioid receptor mu 1 using [3H]-DAMGO at the Kd concentration 0.57 nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Macaca mulatta)
University Of Catania

Curated by ChEMBL
LigandPNGBDBM50458148(CHEMBL4214248)
Affinity DataKi:  2.10nMAssay Description:Displacement of [3H]DAMGO from MOR in monkey brain cortex membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50095703(3-But-3-enyl-6,11-dimethyl-1,2,3,4,5,6-hexahydro-2...)
Affinity DataKi:  21nMAssay Description:Ki value determined against Opioid receptor delta 1 using [3H]-DPDPE at the Kd concentration 2.1 nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOpioid receptor delta 1(Macaca mulatta)
University Of Catania

Curated by ChEMBL
LigandPNGBDBM50458148(CHEMBL4214248)
Affinity DataKi:  21nMAssay Description:Displacement of [3H]naltrindole from DOR in monkey brain cortex membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Mus musculus (Mouse))
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50095703(3-But-3-enyl-6,11-dimethyl-1,2,3,4,5,6-hexahydro-2...)
Affinity DataKi:  1.60E+3nMAssay Description:Ki value determined against Sigma opioid receptor type 1 using [(+)-[3H]pentazocaine at the Kd concentration 2nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed