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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 5 hits in this display   

TargetSuppressor of tumorigenicity 14 protein(Homo sapiens (Human))
Curacyte Chemistry

LigandPNGBDBM23869(3-[(2S)-3-[4-(3-aminopropanoyl)piperazin-1-yl]-3-o...)
Affinity DataKi:  170nM ΔG°:  -38.6kJ/molepH: 8.0 T: 2°CAssay Description:The measurements were carried out on a microplate reader. Two concentrations of the substrate and five concentrations of the inhibitor were used. Af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen(Homo sapiens (Human))
Curacyte Chemistry

LigandPNGBDBM23869(3-[(2S)-3-[4-(3-aminopropanoyl)piperazin-1-yl]-3-o...)
Affinity DataKi:  440nMAssay Description:The measurements were carried out on a microplate reader. Two concentrations of the substrate and five concentrations of the inhibitor were used. Af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Curacyte Chemistry

LigandPNGBDBM23869(3-[(2S)-3-[4-(3-aminopropanoyl)piperazin-1-yl]-3-o...)
Affinity DataKi:  640nMAssay Description:The measurements were carried out on a microplate reader. Two concentrations of the substrate and five concentrations of the inhibitor were used. Af...More data for this Ligand-Target Pair
TargetProthrombin(Bos taurus (Bovine))
Curacyte Chemistry

LigandPNGBDBM23869(3-[(2S)-3-[4-(3-aminopropanoyl)piperazin-1-yl]-3-o...)
Affinity DataKi:  3.30E+3nMAssay Description:The measurements were carried out on a microplate reader. Two concentrations of the substrate and five concentrations of the inhibitor were used. Af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Bos taurus)
Curacyte Chemistry

LigandPNGBDBM23869(3-[(2S)-3-[4-(3-aminopropanoyl)piperazin-1-yl]-3-o...)
Affinity DataKi:  1.50E+4nMAssay Description:The measurements were carried out on a microplate reader. Two concentrations of the substrate and five concentrations of the inhibitor were used. Af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed