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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 27 hits in this display   

Target72 kDa type IV collagenase(Homo sapiens (Human))
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM50100927((S)-N-(1-(4,4-dimethyl-2,5-dioxoimidazolidin-1-yl)...)
Affinity DataIC50:  4nMAssay Description:Inhibition of MMP-2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails PubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM50100927((S)-N-(1-(4,4-dimethyl-2,5-dioxoimidazolidin-1-yl)...)
Affinity DataIC50:  4nMAssay Description:Inhibition of MMP2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM50100927((S)-N-(1-(4,4-dimethyl-2,5-dioxoimidazolidin-1-yl)...)
Affinity DataIC50:  4nMAssay Description:In vitro inhibition of human Matrix metalloproteinase-2.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM50100922(CHEMBL43411 | N-[2-(4,4-Dimethyl-2,5-dioxo-imidazo...)
Affinity DataIC50:  6nMAssay Description:In vitro inhibition of human Matrix metalloproteinase-2.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50100927((S)-N-(1-(4,4-dimethyl-2,5-dioxoimidazolidin-1-yl)...)
Affinity DataIC50:  42nMAssay Description:Inhibition of Matrix metalloproteinase-3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50100927((S)-N-(1-(4,4-dimethyl-2,5-dioxoimidazolidin-1-yl)...)
Affinity DataIC50:  42nMAssay Description:Inhibition of MMP-3 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetStromelysin-1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50100927((S)-N-(1-(4,4-dimethyl-2,5-dioxoimidazolidin-1-yl)...)
Affinity DataIC50:  42nMAssay Description:Inhibition of MMP3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrix metalloproteinase-9(Homo sapiens (Human))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50100927((S)-N-(1-(4,4-dimethyl-2,5-dioxoimidazolidin-1-yl)...)
Affinity DataIC50:  120nMAssay Description:Inhibition of MMP9More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrix metalloproteinase-9(Homo sapiens (Human))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50100927((S)-N-(1-(4,4-dimethyl-2,5-dioxoimidazolidin-1-yl)...)
Affinity DataIC50:  120nMAssay Description:Inhibition of matrix metalloproteinase-9More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrix metalloproteinase-9(Homo sapiens (Human))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50100927((S)-N-(1-(4,4-dimethyl-2,5-dioxoimidazolidin-1-yl)...)
Affinity DataIC50:  120nMAssay Description:Inhibition of MMP-9 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails PubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM50100923(CHEMBL41943 | N-[(R)-2-(4,4-Dimethyl-2,5-dioxo-imi...)
Affinity DataIC50:  180nMAssay Description:In vitro inhibition of human Matrix metalloproteinase-2.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM50100923(CHEMBL41943 | N-[(R)-2-(4,4-Dimethyl-2,5-dioxo-imi...)
Affinity DataIC50:  180nMAssay Description:Inhibition of MMP-2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMatrix metalloproteinase-9(Homo sapiens (Human))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50100923(CHEMBL41943 | N-[(R)-2-(4,4-Dimethyl-2,5-dioxo-imi...)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibition of MMP-9 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMatrix metalloproteinase-9(Homo sapiens (Human))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50100923(CHEMBL41943 | N-[(R)-2-(4,4-Dimethyl-2,5-dioxo-imi...)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibition of matrix metalloproteinase-9More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50100923(CHEMBL41943 | N-[(R)-2-(4,4-Dimethyl-2,5-dioxo-imi...)
Affinity DataIC50:  3.10E+3nMAssay Description:Inhibition of MMP-3 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetStromelysin-1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50100923(CHEMBL41943 | N-[(R)-2-(4,4-Dimethyl-2,5-dioxo-imi...)
Affinity DataIC50:  3.10E+3nMAssay Description:Inhibition of Matrix metalloproteinase-3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInterstitial collagenase(Homo sapiens (Human))
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM50100927((S)-N-(1-(4,4-dimethyl-2,5-dioxoimidazolidin-1-yl)...)
Affinity DataIC50:  4.60E+3nMAssay Description:Inhibition of MMP-1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetInterstitial collagenase(Homo sapiens (Human))
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM50100927((S)-N-(1-(4,4-dimethyl-2,5-dioxoimidazolidin-1-yl)...)
Affinity DataIC50:  4.60E+3nMAssay Description:Inhibition of MMP1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInterstitial collagenase(Homo sapiens (Human))
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM50100927((S)-N-(1-(4,4-dimethyl-2,5-dioxoimidazolidin-1-yl)...)
Affinity DataIC50:  4.60E+3nMAssay Description:In vitro inhibition of human Matrix metalloproteinase-1.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInterstitial collagenase(Homo sapiens (Human))
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM50100922(CHEMBL43411 | N-[2-(4,4-Dimethyl-2,5-dioxo-imidazo...)
Affinity DataIC50:  8.60E+3nMAssay Description:In vitro inhibition of human Matrix metalloproteinase-1.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrilysin(Homo sapiens (Human))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50100927((S)-N-(1-(4,4-dimethyl-2,5-dioxoimidazolidin-1-yl)...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of MMP7More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInterstitial collagenase(Homo sapiens (Human))
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM50100923(CHEMBL41943 | N-[(R)-2-(4,4-Dimethyl-2,5-dioxo-imi...)
Affinity DataIC50: >1.00E+4nMAssay Description:In vitro inhibition of human Matrix metalloproteinase-1.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrilysin(Homo sapiens (Human))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50100923(CHEMBL41943 | N-[(R)-2-(4,4-Dimethyl-2,5-dioxo-imi...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of Matrix metalloproteinase-7More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrilysin(Homo sapiens (Human))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50100927((S)-N-(1-(4,4-dimethyl-2,5-dioxoimidazolidin-1-yl)...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of MMP-7 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMatrilysin(Homo sapiens (Human))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50100923(CHEMBL41943 | N-[(R)-2-(4,4-Dimethyl-2,5-dioxo-imi...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of MMP-7 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMatrilysin(Homo sapiens (Human))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50100927((S)-N-(1-(4,4-dimethyl-2,5-dioxoimidazolidin-1-yl)...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of Matrix metalloproteinase-7More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInterstitial collagenase(Homo sapiens (Human))
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM50100923(CHEMBL41943 | N-[(R)-2-(4,4-Dimethyl-2,5-dioxo-imi...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of MMP-1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails PubMed