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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
168
hits in this display
Target
D(4) dopamine receptor
(Homo sapiens (Human))
Washington University
Curated by
PDSP K
i
Database
Ligand
BDBM84637
(CAS_85760-74-3 | CHEMBL240773 | NSC_54562 | QUINPI...)
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Affinity Data
Ki: 0.230nM
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Target
D(3) dopamine receptor
(Homo sapiens (Human))
Università
Curated by
ChEMBL
Ligand
BDBM84637
(CAS_85760-74-3 | CHEMBL240773 | NSC_54562 | QUINPI...)
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Affinity Data
Ki: 0.410nM
Assay Description:
Displacement of [3H]spiroperidol from cloned human dopamine receptor D3 in CHO cell membrane
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Target
D(4) dopamine receptor
(Homo sapiens (Human))
Washington University
Curated by
PDSP K
i
Database
Ligand
BDBM84637
(CAS_85760-74-3 | CHEMBL240773 | NSC_54562 | QUINPI...)
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Affinity Data
Ki: 1.80nM
Assay Description:
High inhibition constant against [3H]-spiperone binding to human Dopamine receptor D4.4 expressed in CHO cells
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Target
D(4) dopamine receptor
(Homo sapiens (Human))
Washington University
Curated by
PDSP K
i
Database
Ligand
BDBM84637
(CAS_85760-74-3 | CHEMBL240773 | NSC_54562 | QUINPI...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 1.80nM
Assay Description:
In vitro for its ability to displace [3H]- spiperone from cloned human Dopamine receptor D4 expressed in CHO cells; high binding affinity
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Target
D(4) dopamine receptor
(Homo sapiens (Human))
Washington University
Curated by
PDSP K
i
Database
Ligand
BDBM84637
(CAS_85760-74-3 | CHEMBL240773 | NSC_54562 | QUINPI...)
Copy SMILES
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Affinity Data
Ki: 1.80nM
Assay Description:
High binding affinity towards human dopamine receptor 4.4 expressed in Chinese hamster ovary cells using [3H]spiperone (0.5 nM) as radioligand
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Target
D(4) dopamine receptor
(Homo sapiens (Human))
Washington University
Curated by
PDSP K
i
Database
Ligand
BDBM84637
(CAS_85760-74-3 | CHEMBL240773 | NSC_54562 | QUINPI...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 1.80nM
Assay Description:
In vitro binding affinity to displace [3H]spiperone from the cloned human dopamine receptor D4 in CHO cells
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Target
Dopamine receptor D4
(CANINE)
University Of Toronto
Curated by
PDSP K
i
Database
Ligand
BDBM84637
(CAS_85760-74-3 | CHEMBL240773 | NSC_54562 | QUINPI...)
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Affinity Data
Ki: 4.80nM
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Target
D(3) dopamine receptor
(Rattus norvegicus (Rat))
U. 109
Curated by
PDSP K
i
Database
Ligand
BDBM84637
(CAS_85760-74-3 | CHEMBL240773 | NSC_54562 | QUINPI...)
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Affinity Data
Ki: 5.10nM
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Target
D(3) dopamine receptor
(Rattus norvegicus (Rat))
U. 109
Curated by
PDSP K
i
Database
Ligand
BDBM84637
(CAS_85760-74-3 | CHEMBL240773 | NSC_54562 | QUINPI...)
Copy SMILES
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Affinity Data
Ki: 5.70nM
Assay Description:
Tested for binding affinity against dopamine receptor D3 expressed in Sf9 cells.
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Target
D(2) dopamine receptor
(Rattus norvegicus (rat))
Dupont Pharmaceuticals
Curated by
PDSP K
i
Database
Ligand
BDBM84637
(CAS_85760-74-3 | CHEMBL240773 | NSC_54562 | QUINPI...)
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Affinity Data
Ki: 8nM
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Target
D(3) dopamine receptor
(Homo sapiens (Human))
Università
Curated by
ChEMBL
Ligand
BDBM84637
(CAS_85760-74-3 | CHEMBL240773 | NSC_54562 | QUINPI...)
Copy SMILES
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Affinity Data
Ki: 12.5nM
Assay Description:
Displacement of [3H]spiroperidol from human cloned dopamine D3 receptor by liquid scintillation counting
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Target
D(2) dopamine receptor
(Homo sapiens (Human))
University Of Toronto
Curated by
PDSP K
i
Database
Ligand
BDBM84637
(CAS_85760-74-3 | CHEMBL240773 | NSC_54562 | QUINPI...)
Copy SMILES
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Affinity Data
Ki: 14nM
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Target
D(3) dopamine receptor
(Homo sapiens (Human))
Università
Curated by
ChEMBL
Ligand
BDBM84637
(CAS_85760-74-3 | CHEMBL240773 | NSC_54562 | QUINPI...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 15nM
Assay Description:
Displacement of [3H]spiperone from human dopamine D3 receptor expressed in CHO cells
More data for this Ligand-Target Pair
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Target
D(2) dopamine receptor
(Rattus norvegicus (rat))
Dupont Pharmaceuticals
Curated by
PDSP K
i
Database
Ligand
BDBM84637
(CAS_85760-74-3 | CHEMBL240773 | NSC_54562 | QUINPI...)
Copy SMILES
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Affinity Data
Ki: 15.5nM
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Target
D(3) dopamine receptor
(Homo sapiens (Human))
Università
Curated by
ChEMBL
Ligand
BDBM84637
(CAS_85760-74-3 | CHEMBL240773 | NSC_54562 | QUINPI...)
Copy SMILES
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Affinity Data
Ki: 17nM
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Target
D(2) dopamine receptor
(Homo sapiens (Human))
University Of Toronto
Curated by
PDSP K
i
Database
Ligand
BDBM84637
(CAS_85760-74-3 | CHEMBL240773 | NSC_54562 | QUINPI...)
Copy SMILES
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Affinity Data
Ki: 18nM
Assay Description:
Displacement of [3H]7-OH-DPAT from human dopamine D2L receptor expressed in CHO cells
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Target
D(3) dopamine receptor
(Rattus norvegicus (Rat))
U. 109
Curated by
PDSP K
i
Database
Ligand
BDBM84637
(CAS_85760-74-3 | CHEMBL240773 | NSC_54562 | QUINPI...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 19.3nM
More data for this Ligand-Target Pair
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Target
D(3) dopamine receptor
(Homo sapiens (Human))
Università
Curated by
ChEMBL
Ligand
BDBM84637
(CAS_85760-74-3 | CHEMBL240773 | NSC_54562 | QUINPI...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 24nM
Assay Description:
High inhibition constant against [3H]-spiperone binding to human Dopamine receptor D3 expressed in CHO cells
More data for this Ligand-Target Pair
Target Info
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Target
D(3) dopamine receptor
(Homo sapiens (Human))
Università
Curated by
ChEMBL
Ligand
BDBM84637
(CAS_85760-74-3 | CHEMBL240773 | NSC_54562 | QUINPI...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 24nM
Assay Description:
In vitro for its ability to displace [3H]- spiperone from cloned human Dopamine receptor D3 expressed in CHO cells; high binding affinity
More data for this Ligand-Target Pair
Target Info
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UniProtKB/SwissProt
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Target
D(3) dopamine receptor
(Homo sapiens (Human))
Università
Curated by
ChEMBL
Ligand
BDBM84637
(CAS_85760-74-3 | CHEMBL240773 | NSC_54562 | QUINPI...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 24nM
Assay Description:
High binding affinity towards human dopamine receptor 3 expressed in Chinese hamster ovary cells using [3H]spiperone (0.5 nM) as radioligand
More data for this Ligand-Target Pair
Target Info
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Copy BDB DOI
Target
D(3) dopamine receptor
(Homo sapiens (Human))
Università
Curated by
ChEMBL
Ligand
BDBM84637
(CAS_85760-74-3 | CHEMBL240773 | NSC_54562 | QUINPI...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 24nM
Assay Description:
In vitro binding affinity to displace [3H]spiperone from the cloned human dopamine receptor D3 in CHO cells
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
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Target
D(2) dopamine receptor
(Rattus norvegicus (rat))
Dupont Pharmaceuticals
Curated by
PDSP K
i
Database
Ligand
BDBM84637
(CAS_85760-74-3 | CHEMBL240773 | NSC_54562 | QUINPI...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 24nM
More data for this Ligand-Target Pair
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Target
D(3) dopamine receptor
(Rattus norvegicus (Rat))
U. 109
Curated by
PDSP K
i
Database
Ligand
BDBM84637
(CAS_85760-74-3 | CHEMBL240773 | NSC_54562 | QUINPI...)
Copy SMILES
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Affinity Data
Ki: 29.4nM
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Target
D(4) dopamine receptor
(Homo sapiens (Human))
Washington University
Curated by
PDSP K
i
Database
Ligand
BDBM84637
(CAS_85760-74-3 | CHEMBL240773 | NSC_54562 | QUINPI...)
Copy SMILES
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Affinity Data
Ki: 33.9nM
More data for this Ligand-Target Pair
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Target
D(4) dopamine receptor
(Homo sapiens (Human))
Washington University
Curated by
PDSP K
i
Database
Ligand
BDBM84637
(CAS_85760-74-3 | CHEMBL240773 | NSC_54562 | QUINPI...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 34nM
More data for this Ligand-Target Pair
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Target
D(2) dopamine receptor
(Homo sapiens (Human))
University Of Toronto
Curated by
PDSP K
i
Database
Ligand
BDBM84637
(CAS_85760-74-3 | CHEMBL240773 | NSC_54562 | QUINPI...)
Copy SMILES
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Affinity Data
Ki: 35nM
Assay Description:
High binding affinity towards human dopamine receptor 2 (short) expressed in Chinese hamster ovary cells using [3H]spiperone (0.5 nM) as radioligand
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Target
D(2) dopamine receptor
(Homo sapiens (Human))
University Of Toronto
Curated by
PDSP K
i
Database
Ligand
BDBM84637
(CAS_85760-74-3 | CHEMBL240773 | NSC_54562 | QUINPI...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 35nM
Assay Description:
High inhibition constant against [3H]-spiperone binding to human Dopamine receptor D2S expressed in CHO cells
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Target
D(4) dopamine receptor
(Homo sapiens (Human))
Washington University
Curated by
PDSP K
i
Database
Ligand
BDBM84637
(CAS_85760-74-3 | CHEMBL240773 | NSC_54562 | QUINPI...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 37.3nM
More data for this Ligand-Target Pair
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Target
D(3) dopamine receptor
(Homo sapiens (Human))
Università
Curated by
ChEMBL
Ligand
BDBM84637
(CAS_85760-74-3 | CHEMBL240773 | NSC_54562 | QUINPI...)
Copy SMILES
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Affinity Data
Ki: 39nM
More data for this Ligand-Target Pair
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Target
D(3) dopamine receptor
(Homo sapiens (Human))
Università
Curated by
ChEMBL
Ligand
BDBM84637
(CAS_85760-74-3 | CHEMBL240773 | NSC_54562 | QUINPI...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 41.7nM
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Target
D(3) dopamine receptor
(Homo sapiens (Human))
Università
Curated by
ChEMBL
Ligand
BDBM84637
(CAS_85760-74-3 | CHEMBL240773 | NSC_54562 | QUINPI...)
Copy SMILES
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Affinity Data
Ki: 43nM
More data for this Ligand-Target Pair
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Target
D(3) dopamine receptor
(Homo sapiens (Human))
Università
Curated by
ChEMBL
Ligand
BDBM84637
(CAS_85760-74-3 | CHEMBL240773 | NSC_54562 | QUINPI...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 43nM
Assay Description:
Displacement of [3H]YM-09151-2 from human dopamine D3 receptor expressed in CHOp cells
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Target
Dopamine receptor D4
(CANINE)
University Of Toronto
Curated by
PDSP K
i
Database
Ligand
BDBM84637
(CAS_85760-74-3 | CHEMBL240773 | NSC_54562 | QUINPI...)
Copy SMILES
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Affinity Data
Ki: 46nM
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Target
D(3) dopamine receptor
(Rattus norvegicus (Rat))
U. 109
Curated by
PDSP K
i
Database
Ligand
BDBM84637
(CAS_85760-74-3 | CHEMBL240773 | NSC_54562 | QUINPI...)
Copy SMILES
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Affinity Data
Ki: 46.8nM
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Target
D(2) dopamine receptor
(Rattus norvegicus (rat))
Dupont Pharmaceuticals
Curated by
PDSP K
i
Database
Ligand
BDBM84637
(CAS_85760-74-3 | CHEMBL240773 | NSC_54562 | QUINPI...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 47nM
More data for this Ligand-Target Pair
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Target
D(2) dopamine receptor
(Rattus norvegicus (rat))
Dupont Pharmaceuticals
Curated by
PDSP K
i
Database
Ligand
BDBM84637
(CAS_85760-74-3 | CHEMBL240773 | NSC_54562 | QUINPI...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 48nM
More data for this Ligand-Target Pair
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Target
D(3) dopamine receptor
(Homo sapiens (Human))
Università
Curated by
ChEMBL
Ligand
BDBM84637
(CAS_85760-74-3 | CHEMBL240773 | NSC_54562 | QUINPI...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 49nM
Assay Description:
Displacement of [3H]spiperone from human cloned dopamine D3 receptor expressed in CHO cells
More data for this Ligand-Target Pair
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Target
D(2) dopamine receptor
(Homo sapiens (Human))
University Of Toronto
Curated by
PDSP K
i
Database
Ligand
BDBM84637
(CAS_85760-74-3 | CHEMBL240773 | NSC_54562 | QUINPI...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 52nM
Assay Description:
In vitro for its ability to displace [3H]- spiperone from cloned human dopamine D2 short receptor expressed in CHO cells; high binding affinity
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D(2) dopamine receptor
(Homo sapiens (Human))
University Of Toronto
Curated by
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Ligand
BDBM84637
(CAS_85760-74-3 | CHEMBL240773 | NSC_54562 | QUINPI...)
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Ki: 52nM
Assay Description:
Effective concentration for [3H]thymidine uptake in growing CHO cells stably expressing the dopamine D4.2 receptor
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D(4) dopamine receptor
(Homo sapiens (Human))
Washington University
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BDBM84637
(CAS_85760-74-3 | CHEMBL240773 | NSC_54562 | QUINPI...)
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Ki: 53nM
Assay Description:
Low inhibition constant against [3H]-spiperone binding to human Dopamine receptor D4.4 expressed in CHO cells
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D(4) dopamine receptor
(Homo sapiens (Human))
Washington University
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BDBM84637
(CAS_85760-74-3 | CHEMBL240773 | NSC_54562 | QUINPI...)
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Ki: 53nM
Assay Description:
In vitro for its ability to displace [3H]- spiperone from cloned human Dopamine receptor D2L expressed in CHO cells
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D(4) dopamine receptor
(Homo sapiens (Human))
Washington University
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BDBM84637
(CAS_85760-74-3 | CHEMBL240773 | NSC_54562 | QUINPI...)
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Ki: 53nM
Assay Description:
Low binding affinity towards human dopamine receptor 4.4 expressed in Chinese hamster ovary cells using [3H]spiperone (0.5 nM) as radioligand
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D(2) dopamine receptor
(Rattus norvegicus (rat))
Dupont Pharmaceuticals
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BDBM84637
(CAS_85760-74-3 | CHEMBL240773 | NSC_54562 | QUINPI...)
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Ki: 54nM
Assay Description:
Compound was evaluated for its ability to displace [3H]raclopride from dopamine receptor D2 in rat striatal homogenates
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D(2) dopamine receptor
(BOVINE)
Universit£
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ChEMBL
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BDBM84637
(CAS_85760-74-3 | CHEMBL240773 | NSC_54562 | QUINPI...)
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Ki: 59nM
Assay Description:
Inhibition of [3H]YM-09151-2 binding to bovine retina membrane Dopamine receptor D2, high affinity site
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D(1A) dopamine receptor
(Homo sapiens (Human))
Friedrich-Alexander University
Curated by
ChEMBL
Ligand
BDBM84637
(CAS_85760-74-3 | CHEMBL240773 | NSC_54562 | QUINPI...)
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Ki: 63nM
Assay Description:
Binding affinity (high) towards human dopamine receptor 2 long against radioligand [3H]spiperone, expressed in Chinese hamster ovary cells
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D(2) dopamine receptor
(Homo sapiens (Human))
University Of Toronto
Curated by
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i
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BDBM84637
(CAS_85760-74-3 | CHEMBL240773 | NSC_54562 | QUINPI...)
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Ki: 63nM
Assay Description:
High inhibition constant against [3H]-spiperone binding to human Dopamine receptor D2L expressed in CHO cells
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D(2) dopamine receptor
(Homo sapiens (Human))
University Of Toronto
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i
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Ligand
BDBM84637
(CAS_85760-74-3 | CHEMBL240773 | NSC_54562 | QUINPI...)
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Ki: 64nM
Assay Description:
In vitro binding affinity to displace [3H]spiperone from the cloned human dopamine receptor D2 long in CHO cells
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Target
D(2) dopamine receptor
(Homo sapiens (Human))
University Of Toronto
Curated by
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i
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Ligand
BDBM84637
(CAS_85760-74-3 | CHEMBL240773 | NSC_54562 | QUINPI...)
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Ki: 64nM
Assay Description:
In vitro for its ability to displace [3H]- spiperone from cloned human dopamine D2 long receptor expressed in CHO cells; high binding affinity
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Target
D(4) dopamine receptor
(Homo sapiens (Human))
Washington University
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BDBM84637
(CAS_85760-74-3 | CHEMBL240773 | NSC_54562 | QUINPI...)
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Ki: 124nM
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Target
D(4) dopamine receptor
(Homo sapiens (Human))
Washington University
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i
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BDBM84637
(CAS_85760-74-3 | CHEMBL240773 | NSC_54562 | QUINPI...)
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Ki: 140nM
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D(2) dopamine receptor
(Mus musculus (Mouse))
Medical Research Service
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i
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Ligand
BDBM84637
(CAS_85760-74-3 | CHEMBL240773 | NSC_54562 | QUINPI...)
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Ki: 204nM
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Target
D(4) dopamine receptor
(Homo sapiens (Human))
Washington University
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i
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Ligand
BDBM84637
(CAS_85760-74-3 | CHEMBL240773 | NSC_54562 | QUINPI...)
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Ki: 250nM
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Target
D(2) dopamine receptor
(Homo sapiens (Human))
University Of Toronto
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i
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Ligand
BDBM84637
(CAS_85760-74-3 | CHEMBL240773 | NSC_54562 | QUINPI...)
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Ki: 260nM
Assay Description:
Displacement of [3H]spiperone from human dopamine D2L receptor expressed in CHO cells
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Target
D(2) dopamine receptor
(Homo sapiens (Human))
University Of Toronto
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i
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Ligand
BDBM84637
(CAS_85760-74-3 | CHEMBL240773 | NSC_54562 | QUINPI...)
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Ki: 260nM
Assay Description:
Displacement of [3H]spiperone from human dopamine D2L receptor expressed in CHO cells
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Target
D(2) dopamine receptor
(Rattus norvegicus (rat))
Dupont Pharmaceuticals
Curated by
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i
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BDBM84637
(CAS_85760-74-3 | CHEMBL240773 | NSC_54562 | QUINPI...)
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Ki: 389nM
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D(3) dopamine receptor
(Homo sapiens (Human))
Università
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ChEMBL
Ligand
BDBM84637
(CAS_85760-74-3 | CHEMBL240773 | NSC_54562 | QUINPI...)
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Ki: 420nM
Assay Description:
Low inhibition constant against [3H]-spiperone binding to human Dopamine receptor D3 expressed in CHO cells
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Target
D(3) dopamine receptor
(Homo sapiens (Human))
Università
Curated by
ChEMBL
Ligand
BDBM84637
(CAS_85760-74-3 | CHEMBL240773 | NSC_54562 | QUINPI...)
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Affinity Data
Ki: 420nM
Assay Description:
In vitro for its ability to displace [3H]- spiperoneI from cloned human Dopamine receptor D3 expressed in CHO cells; Low binding affinity
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Target
D(3) dopamine receptor
(Homo sapiens (Human))
Università
Curated by
ChEMBL
Ligand
BDBM84637
(CAS_85760-74-3 | CHEMBL240773 | NSC_54562 | QUINPI...)
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Ki: 420nM
Assay Description:
Low binding affinity towards human dopamine receptor 3 expressed in Chinese hamster ovary cells using [3H]spiperone (0.5 nM) as radioligand
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D(2) dopamine receptor
(Rattus norvegicus (rat))
Dupont Pharmaceuticals
Curated by
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BDBM84637
(CAS_85760-74-3 | CHEMBL240773 | NSC_54562 | QUINPI...)
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Ki: 576nM
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D(2) dopamine receptor
(Rattus norvegicus (rat))
Dupont Pharmaceuticals
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BDBM84637
(CAS_85760-74-3 | CHEMBL240773 | NSC_54562 | QUINPI...)
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Ki: 576nM
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D(2) dopamine receptor
(Homo sapiens (Human))
University Of Toronto
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i
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BDBM84637
(CAS_85760-74-3 | CHEMBL240773 | NSC_54562 | QUINPI...)
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Ki: 600nM
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Target
D(2) dopamine receptor
(Rattus norvegicus (rat))
Dupont Pharmaceuticals
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i
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BDBM84637
(CAS_85760-74-3 | CHEMBL240773 | NSC_54562 | QUINPI...)
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Ki: 734nM
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D(2) dopamine receptor
(Homo sapiens (Human))
University Of Toronto
Curated by
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i
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BDBM84637
(CAS_85760-74-3 | CHEMBL240773 | NSC_54562 | QUINPI...)
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Ki: 870nM
Assay Description:
Displacement of [3H]spiperone from human cloned dopamine D2short receptor expressed in CHO cells
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Target
D(2) dopamine receptor
(Homo sapiens (Human))
University Of Toronto
Curated by
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i
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BDBM84637
(CAS_85760-74-3 | CHEMBL240773 | NSC_54562 | QUINPI...)
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Ki: 891nM
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Target
D(2) dopamine receptor
(Rattus norvegicus (rat))
Dupont Pharmaceuticals
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i
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BDBM84637
(CAS_85760-74-3 | CHEMBL240773 | NSC_54562 | QUINPI...)
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Ki: 930nM
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Target
D(2) dopamine receptor
(Homo sapiens (Human))
University Of Toronto
Curated by
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i
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Ligand
BDBM84637
(CAS_85760-74-3 | CHEMBL240773 | NSC_54562 | QUINPI...)
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Affinity Data
Ki: 950nM
Assay Description:
Displacement of [3H]spiperone from human cloned dopamine D2long receptor expressed in CHO cells
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Target
D(1A) dopamine receptor
(RAT)
University Of North Carolina
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i
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Ligand
BDBM84637
(CAS_85760-74-3 | CHEMBL240773 | NSC_54562 | QUINPI...)
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Ki: 1.00E+3nM
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Target
Histamine H1 receptor
(Cavia porcellus (domestic guinea pig))
Institut De Recherches Servier
Curated by
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i
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Ligand
BDBM84637
(CAS_85760-74-3 | CHEMBL240773 | NSC_54562 | QUINPI...)
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Ki: 1.05E+3nM
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Target
D(2) dopamine receptor
(Homo sapiens (Human))
University Of Toronto
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i
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BDBM84637
(CAS_85760-74-3 | CHEMBL240773 | NSC_54562 | QUINPI...)
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Ki: 1.19E+3nM
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Target
D(2) dopamine receptor
(Homo sapiens (Human))
University Of Toronto
Curated by
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i
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Ligand
BDBM84637
(CAS_85760-74-3 | CHEMBL240773 | NSC_54562 | QUINPI...)
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Ki: 1.19E+3nM
Assay Description:
Displacement of [3H]YM-09151-2 from human dopamine D2 receptor expressed in CHOp cells
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Target
D(4) dopamine receptor
(Homo sapiens (Human))
Washington University
Curated by
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i
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BDBM84637
(CAS_85760-74-3 | CHEMBL240773 | NSC_54562 | QUINPI...)
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Ki: 1.26E+3nM
Assay Description:
Inhibitory constant for [3H]YM-09151-2 binding to Dopamine receptor D2-like in porcine striatal membranes
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Target
D(2) dopamine receptor
(Homo sapiens (Human))
University Of Toronto
Curated by
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i
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BDBM84637
(CAS_85760-74-3 | CHEMBL240773 | NSC_54562 | QUINPI...)
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Ki: 1.40E+3nM
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Target
D(2) dopamine receptor
(Homo sapiens (Human))
University Of Toronto
Curated by
PDSP K
i
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Ligand
BDBM84637
(CAS_85760-74-3 | CHEMBL240773 | NSC_54562 | QUINPI...)
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Ki: 1.45E+3nM
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Target
D(2) dopamine receptor
(BOVINE)
Universit£
Curated by
ChEMBL
Ligand
BDBM84637
(CAS_85760-74-3 | CHEMBL240773 | NSC_54562 | QUINPI...)
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Affinity Data
Ki: 1.50E+3nM
Assay Description:
Tested for binding affinity against Dopamine receptor D2 like from bovine striatum membranes by using [3H]YM-09151-2 radioligand
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5-hydroxytryptamine receptor 1A
(Homo sapiens (Human))
Institut De Recherches Servier
Curated by
PDSP K
i
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Ligand
BDBM84637
(CAS_85760-74-3 | CHEMBL240773 | NSC_54562 | QUINPI...)
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Ki: 1.70E+3nM
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Target
5-hydroxytryptamine receptor 1A
(Homo sapiens (Human))
Institut De Recherches Servier
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i
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Ligand
BDBM84637
(CAS_85760-74-3 | CHEMBL240773 | NSC_54562 | QUINPI...)
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Ki: 1.71E+3nM
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Target
D(2) dopamine receptor
(Homo sapiens (Human))
University Of Toronto
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i
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Ligand
BDBM84637
(CAS_85760-74-3 | CHEMBL240773 | NSC_54562 | QUINPI...)
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Ki: 2.16E+3nM
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Alpha-2B adrenergic receptor
(Homo sapiens (Human))
Institut De Recherches Servier
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PDSP K
i
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Ligand
BDBM84637
(CAS_85760-74-3 | CHEMBL240773 | NSC_54562 | QUINPI...)
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Ki: 2.51E+3nM
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Target
D(2) dopamine receptor
(Homo sapiens (Human))
University Of Toronto
Curated by
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i
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Ligand
BDBM84637
(CAS_85760-74-3 | CHEMBL240773 | NSC_54562 | QUINPI...)
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Affinity Data
Ki: 2.57E+3nM
Assay Description:
Affinity towards Dopamine receptor D2
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Target
D(2) dopamine receptor
(BOVINE)
Universit£
Curated by
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Ligand
BDBM84637
(CAS_85760-74-3 | CHEMBL240773 | NSC_54562 | QUINPI...)
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Affinity Data
Ki: 2.58E+3nM
Assay Description:
Inhibition of [3H]YM-09151-2 binding to bovine retina membrane Dopamine receptor D2, low affinity site
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D(2) dopamine receptor
(Homo sapiens (Human))
University Of Toronto
Curated by
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i
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Ligand
BDBM84637
(CAS_85760-74-3 | CHEMBL240773 | NSC_54562 | QUINPI...)
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Affinity Data
Ki: 3.00E+3nM
Assay Description:
Low inhibition constant against [3H]-spiperone binding to human Dopamine receptor D2S expressed in CHO cells
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Target
D(2) dopamine receptor
(Homo sapiens (Human))
University Of Toronto
Curated by
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i
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Ligand
BDBM84637
(CAS_85760-74-3 | CHEMBL240773 | NSC_54562 | QUINPI...)
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Affinity Data
Ki: 3.00E+3nM
Assay Description:
Binding affinity (low) towards human dopamine receptor 2 short against radioligand [3H]spiperone, expressed in Chinese hamster ovary cells
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Target
D(2) dopamine receptor
(Homo sapiens (Human))
University Of Toronto
Curated by
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i
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Ligand
BDBM84637
(CAS_85760-74-3 | CHEMBL240773 | NSC_54562 | QUINPI...)
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Affinity Data
Ki: 3.10E+3nM
Assay Description:
Low inhibition constant against [3H]-spiperone binding to human Dopamine receptor D2L expressed in CHO cells
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Target
D(2) dopamine receptor
(Homo sapiens (Human))
University Of Toronto
Curated by
PDSP K
i
Database
Ligand
BDBM84637
(CAS_85760-74-3 | CHEMBL240773 | NSC_54562 | QUINPI...)
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Affinity Data
Ki: 3.10E+3nM
Assay Description:
Binding affinity (low) towards human dopamine receptor 2 (long) against radioligand [3H]spiperone, expressed in Chinese hamster ovary cells
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Target
D(2) dopamine receptor
(Homo sapiens (Human))
University Of Toronto
Curated by
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i
Database
Ligand
BDBM84637
(CAS_85760-74-3 | CHEMBL240773 | NSC_54562 | QUINPI...)
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Affinity Data
Ki: 4.00E+3nM
Assay Description:
In vitro for its ability to displace [3H]- spiperone from cloned human dopamine D2 long receptor expressed in CHO cells
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D(2) dopamine receptor
(Rattus norvegicus (rat))
Dupont Pharmaceuticals
Curated by
PDSP K
i
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Ligand
BDBM84637
(CAS_85760-74-3 | CHEMBL240773 | NSC_54562 | QUINPI...)
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Ki: 7.70E+3nM
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Target
5-hydroxytryptamine receptor 2C
(Rattus norvegicus (Rat))
Sri International
Curated by
PDSP K
i
Database
Ligand
BDBM84637
(CAS_85760-74-3 | CHEMBL240773 | NSC_54562 | QUINPI...)
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Ki: >1.00E+4nM
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Target
5-hydroxytryptamine receptor 3A
(Mus musculus (house mouse))
Sri International
Curated by
PDSP K
i
Database
Ligand
BDBM84637
(CAS_85760-74-3 | CHEMBL240773 | NSC_54562 | QUINPI...)
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Ki: >1.00E+4nM
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Target
D(1A) dopamine receptor
(BOVINE)
University Of Nebraska
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i
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Ligand
BDBM84637
(CAS_85760-74-3 | CHEMBL240773 | NSC_54562 | QUINPI...)
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Ki: >1.00E+4nM
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Target
D(1A) dopamine receptor
(Homo sapiens (Human))
Friedrich-Alexander University
Curated by
ChEMBL
Ligand
BDBM84637
(CAS_85760-74-3 | CHEMBL240773 | NSC_54562 | QUINPI...)
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Affinity Data
Ki: >1.00E+4nM
Assay Description:
Displacement of [3H]SCH-23390 from human dopamine D1 receptor expressed in LHD1 cells
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Target
D(1B) dopamine receptor
(Homo sapiens (Human))
Institut De Recherches Servier
Curated by
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i
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Ligand
BDBM84637
(CAS_85760-74-3 | CHEMBL240773 | NSC_54562 | QUINPI...)
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Ki: >1.00E+4nM
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Target
D(1A) dopamine receptor
(Homo sapiens (Human))
Friedrich-Alexander University
Curated by
ChEMBL
Ligand
BDBM84637
(CAS_85760-74-3 | CHEMBL240773 | NSC_54562 | QUINPI...)
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Ki: >1.00E+4nM
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Target
Beta-2 adrenergic receptor
(Homo sapiens (Human))
Institut De Recherches Servier
Curated by
PDSP K
i
Database
Ligand
BDBM84637
(CAS_85760-74-3 | CHEMBL240773 | NSC_54562 | QUINPI...)
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Ki: >1.00E+4nM
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Target
D(1A) dopamine receptor
(Homo sapiens (Human))
Friedrich-Alexander University
Curated by
ChEMBL
Ligand
BDBM84637
(CAS_85760-74-3 | CHEMBL240773 | NSC_54562 | QUINPI...)
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Ki: >1.00E+4nM
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Target
5-hydroxytryptamine receptor 2A
(Rattus norvegicus (rat))
Sri International
Curated by
PDSP K
i
Database
Ligand
BDBM84637
(CAS_85760-74-3 | CHEMBL240773 | NSC_54562 | QUINPI...)
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Ki: >1.00E+4nM
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Target
5-hydroxytryptamine receptor 1B
(Homo sapiens (Human))
Institut De Recherches Servier
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i
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Ligand
BDBM84637
(CAS_85760-74-3 | CHEMBL240773 | NSC_54562 | QUINPI...)
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Ki: >1.00E+4nM
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Target
5-hydroxytryptamine receptor 1D
(Homo sapiens (Human))
Institut De Recherches Servier
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i
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Ligand
BDBM84637
(CAS_85760-74-3 | CHEMBL240773 | NSC_54562 | QUINPI...)
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Ki: >1.00E+4nM
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Target
5-hydroxytryptamine receptor 2A
(Homo sapiens (Human))
Institut De Recherches Servier
Curated by
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i
Database
Ligand
BDBM84637
(CAS_85760-74-3 | CHEMBL240773 | NSC_54562 | QUINPI...)
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Ki: >1.00E+4nM
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Target
5-hydroxytryptamine receptor 2B
(Homo sapiens (Human))
Institut De Recherches Servier
Curated by
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i
Database
Ligand
BDBM84637
(CAS_85760-74-3 | CHEMBL240773 | NSC_54562 | QUINPI...)
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Ki: >1.00E+4nM
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Target
5-hydroxytryptamine receptor 2C
(Homo sapiens (Human))
Institut De Recherches Servier
Curated by
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i
Database
Ligand
BDBM84637
(CAS_85760-74-3 | CHEMBL240773 | NSC_54562 | QUINPI...)
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Ki: >1.00E+4nM
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Target
Alpha-1A adrenergic receptor
(Homo sapiens (Human))
Institut De Recherches Servier
Curated by
PDSP K
i
Database
Ligand
BDBM84637
(CAS_85760-74-3 | CHEMBL240773 | NSC_54562 | QUINPI...)
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Ki: >1.00E+4nM
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Target
Alpha-1B adrenergic receptor
(Homo sapiens (Human))
Institut De Recherches Servier
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i
Database
Ligand
BDBM84637
(CAS_85760-74-3 | CHEMBL240773 | NSC_54562 | QUINPI...)
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Ki: >1.00E+4nM
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Target
Alpha-1D adrenergic receptor
(Homo sapiens (Human))
Institut De Recherches Servier
Curated by
PDSP K
i
Database
Ligand
BDBM84637
(CAS_85760-74-3 | CHEMBL240773 | NSC_54562 | QUINPI...)
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Ki: >1.00E+4nM
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Target
Alpha-2A adrenergic receptor
(Homo sapiens (Human))
Institut De Recherches Servier
Curated by
PDSP K
i
Database
Ligand
BDBM84637
(CAS_85760-74-3 | CHEMBL240773 | NSC_54562 | QUINPI...)
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Ki: >1.00E+4nM
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Target
Alpha-2C adrenergic receptor
(Homo sapiens (Human))
Institut De Recherches Servier
Curated by
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i
Database
Ligand
BDBM84637
(CAS_85760-74-3 | CHEMBL240773 | NSC_54562 | QUINPI...)
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Ki: >1.00E+4nM
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Target
Alpha-2A adrenergic receptor [16-465]
(Rattus norvegicus (rat))
Institut De Recherches Servier
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i
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Ligand
BDBM84637
(CAS_85760-74-3 | CHEMBL240773 | NSC_54562 | QUINPI...)
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Ki: >1.00E+4nM
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Target
Beta-1 adrenergic receptor
(Homo sapiens (Human))
Institut De Recherches Servier
Curated by
PDSP K
i
Database
Ligand
BDBM84637
(CAS_85760-74-3 | CHEMBL240773 | NSC_54562 | QUINPI...)
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Ki: >1.00E+4nM
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Target
D(1A) dopamine receptor
(BOVINE)
University Of Nebraska
Curated by
PDSP K
i
Database
Ligand
BDBM84637
(CAS_85760-74-3 | CHEMBL240773 | NSC_54562 | QUINPI...)
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Affinity Data
Ki: >2.00E+4nM
Assay Description:
Inhibition constant against [3H]-SCH-23,390 binding to Dopamine receptor D1 in bovine striatal membranes
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Target
D(1A) dopamine receptor
(BOVINE)
University Of Nebraska
Curated by
PDSP K
i
Database
Ligand
BDBM84637
(CAS_85760-74-3 | CHEMBL240773 | NSC_54562 | QUINPI...)
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Affinity Data
Ki: >2.00E+4nM
Assay Description:
Binding affinity (low) towards bovine dopamine receptor 1 by using [3H]-SCH- 23390 (0.3 nM) as radioligand
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Target
D(2) dopamine receptor
(Homo sapiens (Human))
University Of Toronto
Curated by
PDSP K
i
Database
Ligand
BDBM84637
(CAS_85760-74-3 | CHEMBL240773 | NSC_54562 | QUINPI...)
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Affinity Data
Ki: 3.10E+4nM
Assay Description:
In vitro for its ability to displace [3H]- spiperone from cloned human dopamine D2 long receptor expressed in CHO cells; Low binding affinity
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Target
D(1A) dopamine receptor
(Sus scrofa)
Friedrich-Alexander University
Curated by
ChEMBL
Ligand
BDBM84637
(CAS_85760-74-3 | CHEMBL240773 | NSC_54562 | QUINPI...)
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Ki: 7.20E+4nM
Assay Description:
Displacement of [3H]SCH23390 from dopamine D1 receptor in pig striatal membranes
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Target
D(1A) dopamine receptor
(Sus scrofa)
Friedrich-Alexander University
Curated by
ChEMBL
Ligand
BDBM84637
(CAS_85760-74-3 | CHEMBL240773 | NSC_54562 | QUINPI...)
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Affinity Data
Ki: 8.70E+4nM
Assay Description:
Displacement of [3H]SCH23390 from dopamine D1 receptor in porcine striatal membranes
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D(1A) dopamine receptor
(Homo sapiens (Human))
Friedrich-Alexander University
Curated by
ChEMBL
Ligand
BDBM84637
(CAS_85760-74-3 | CHEMBL240773 | NSC_54562 | QUINPI...)
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Affinity Data
Ki: 5.25E+5nM
Assay Description:
Affinity towards Dopamine receptor D1
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Target
D(2) dopamine receptor
(Rattus norvegicus (rat))
Dupont Pharmaceuticals
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PDSP K
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Ligand
BDBM84637
(CAS_85760-74-3 | CHEMBL240773 | NSC_54562 | QUINPI...)
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IC50: 100nM
Assay Description:
Displacement of [3H]- -spiperone from Dopamine receptor D2 in rat striatum
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Target
D(2) dopamine receptor
(Homo sapiens (Human))
University Of Toronto
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PDSP K
i
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Ligand
BDBM84637
(CAS_85760-74-3 | CHEMBL240773 | NSC_54562 | QUINPI...)
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Affinity Data
IC50: 462nM
T: 2°C
Assay Description:
Each medicament was dissolved in serum-free F12 culture medium containing 100 μM of IBMX. CHO cells which can stably express D2 receptor were pre-...
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Target
D(1A) dopamine receptor
(RAT)
University Of North Carolina
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Ligand
BDBM84637
(CAS_85760-74-3 | CHEMBL240773 | NSC_54562 | QUINPI...)
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Affinity Data
IC50: >3.00E+4nM
Assay Description:
Displacement of [3H]- #NAME? from binding Dopamine receptor D1 in rat striatum
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Target
D(2) dopamine receptor
(Homo sapiens (Human))
University Of Toronto
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i
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Ligand
BDBM84637
(CAS_85760-74-3 | CHEMBL240773 | NSC_54562 | QUINPI...)
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Affinity Data
EC50: 19nM
Assay Description:
Agonist activity at human dopamine D2 receptor expressed in CHOp cells assessed as stimulation of mitogenesis incubated for 24 hrs by [3H]thymidine i...
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Target
D(2) dopamine receptor
(Rattus norvegicus (rat))
Dupont Pharmaceuticals
Curated by
PDSP K
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Ligand
BDBM84637
(CAS_85760-74-3 | CHEMBL240773 | NSC_54562 | QUINPI...)
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Affinity Data
EC50: 48nM
Assay Description:
Effective concentration to stimulate rat Dopamine receptor D2L mediated [3H]-thymidine incorporation into growing cells using mitogenesis assay
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Target
D(4) dopamine receptor
(Homo sapiens (Human))
Washington University
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PDSP K
i
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Ligand
BDBM84637
(CAS_85760-74-3 | CHEMBL240773 | NSC_54562 | QUINPI...)
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Affinity Data
EC50: 8.70nM
Assay Description:
Effective concentration to stimulate human Dopamine receptor D4.2 mediated [3H]-thymidine incorporation into growing cells using mitogenesis assay
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Target
D(2) dopamine receptor
(Rattus norvegicus (rat))
Dupont Pharmaceuticals
Curated by
PDSP K
i
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Ligand
BDBM84637
(CAS_85760-74-3 | CHEMBL240773 | NSC_54562 | QUINPI...)
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EC50: 17nM
Assay Description:
Effective concentration to stimulate rat Dopamine receptor D2S mediated [3H]-thymidine incorporation into growing cells using mitogenesis assay
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Target
D(3) dopamine receptor
(Homo sapiens (Human))
Università
Curated by
ChEMBL
Ligand
BDBM84637
(CAS_85760-74-3 | CHEMBL240773 | NSC_54562 | QUINPI...)
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Affinity Data
EC50: 2.60nM
Assay Description:
Effective concentration to stimulate human Dopamine receptor D3 mediated [3H]-thymidine incorporation into growing cells using mitogenesis assay
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D(2) dopamine receptor
(Homo sapiens (Human))
University Of Toronto
Curated by
PDSP K
i
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Ligand
BDBM84637
(CAS_85760-74-3 | CHEMBL240773 | NSC_54562 | QUINPI...)
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EC50: 330nM
Assay Description:
Intrinsic activity against dopamine D2(long) receptor expressed in CHO cells by GTPgammaS assay
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Target
D(3) dopamine receptor
(Homo sapiens (Human))
Università
Curated by
ChEMBL
Ligand
BDBM84637
(CAS_85760-74-3 | CHEMBL240773 | NSC_54562 | QUINPI...)
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EC50: 3.40nM
Assay Description:
Intrinsic activity against dopamine D3 receptor assessed as [3H]thymidine uptake in CHO cells by mitogenesis assay
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D(2) dopamine receptor
(Homo sapiens (Human))
University Of Toronto
Curated by
PDSP K
i
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Ligand
BDBM84637
(CAS_85760-74-3 | CHEMBL240773 | NSC_54562 | QUINPI...)
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EC50: 7.40nM
Assay Description:
Intrinsic activity against dopamine D2(long) receptor assessed as [3H]thymidine uptake in CHO cells by mitogenesis assay
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D(2) dopamine receptor
(Homo sapiens (Human))
University Of Toronto
Curated by
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i
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Ligand
BDBM84637
(CAS_85760-74-3 | CHEMBL240773 | NSC_54562 | QUINPI...)
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EC50: 230nM
Assay Description:
Intrinsic activity against dopamine D2(short) receptor expressed in CHO cells by GTPgammaS assay
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D(4) dopamine receptor
(Homo sapiens (Human))
Washington University
Curated by
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Ligand
BDBM84637
(CAS_85760-74-3 | CHEMBL240773 | NSC_54562 | QUINPI...)
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EC50: 11nM
Assay Description:
Intrinsic activity against dopamine D4 receptor assessed as [3H]thymidine uptake in CHO cells by mitogenesis assay
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D(2) dopamine receptor
(Homo sapiens (Human))
University Of Toronto
Curated by
PDSP K
i
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Ligand
BDBM84637
(CAS_85760-74-3 | CHEMBL240773 | NSC_54562 | QUINPI...)
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EC50: 10nM
Assay Description:
Intrinsic activity against dopamine D2(short) receptor assessed as [3H]thymidine uptake in CHO cells by mitogenesis assay
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D(4) dopamine receptor
(Homo sapiens (Human))
Washington University
Curated by
PDSP K
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Ligand
BDBM84637
(CAS_85760-74-3 | CHEMBL240773 | NSC_54562 | QUINPI...)
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EC50: 23nM
Assay Description:
Intrinsic activity against dopamine D4 receptor expressed in CHO cells by GTPgammaS assay
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Target
D(3) dopamine receptor
(Homo sapiens (Human))
Università
Curated by
ChEMBL
Ligand
BDBM84637
(CAS_85760-74-3 | CHEMBL240773 | NSC_54562 | QUINPI...)
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EC50: 2.60nM
Assay Description:
Intrinsic activity at human D3 receptor expressed in CHO dhfr- cells assessed as rate of [3H]thymidine incorporation by mitogenesis assay
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D(3) dopamine receptor
(Homo sapiens (Human))
Università
Curated by
ChEMBL
Ligand
BDBM84637
(CAS_85760-74-3 | CHEMBL240773 | NSC_54562 | QUINPI...)
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Affinity Data
EC50: 5.20nM
Assay Description:
Agonist activity at human dopamine D3 receptor expressed in CHO dhfr mutant cells assessed as stimulation of mitogenesis after 4 hrs
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D(3) dopamine receptor
(Homo sapiens (Human))
Università
Curated by
ChEMBL
Ligand
BDBM84637
(CAS_85760-74-3 | CHEMBL240773 | NSC_54562 | QUINPI...)
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Affinity Data
EC50: 2.10nM
Assay Description:
Intrinsic activity at human D3 receptor expressed in CHO dhfr- cells by [3H]thymidine incorporation assay
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D(3) dopamine receptor
(Homo sapiens (Human))
Università
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ChEMBL
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BDBM84637
(CAS_85760-74-3 | CHEMBL240773 | NSC_54562 | QUINPI...)
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Affinity Data
EC50: 2.90nM
Assay Description:
Intrinsic activity at human D3 receptor expressed in CHO dhfr- cells assessed as inhibition of forskolin-induced cAMP release
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D(3) dopamine receptor
(Homo sapiens (Human))
Università
Curated by
ChEMBL
Ligand
BDBM84637
(CAS_85760-74-3 | CHEMBL240773 | NSC_54562 | QUINPI...)
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EC50: 1.40nM
Assay Description:
Agonist activity at human dopamine D3 receptor expressed in dhfr-deficient CHO cells assessed as [3H]thymidine incorporation
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Target
D(2) dopamine receptor
(Homo sapiens (Human))
University Of Toronto
Curated by
PDSP K
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Ligand
BDBM84637
(CAS_85760-74-3 | CHEMBL240773 | NSC_54562 | QUINPI...)
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EC50: 140nM
Assay Description:
Agonist activity at DRD2 Long receptor expressed in CHO cells assessed as inhibition of forskolin-stimulated cAMP accumulation by bioluminescence ass...
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D(4) dopamine receptor
(Homo sapiens (Human))
Washington University
Curated by
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BDBM84637
(CAS_85760-74-3 | CHEMBL240773 | NSC_54562 | QUINPI...)
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EC50: 2.20nM
Assay Description:
Effective concentration of compound required against human Dopamine D4.2 receptor
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D(4) dopamine receptor
(Homo sapiens (Human))
Washington University
Curated by
PDSP K
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Ligand
BDBM84637
(CAS_85760-74-3 | CHEMBL240773 | NSC_54562 | QUINPI...)
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EC50: 2nM
Assay Description:
Tested for the effective concentration against CHO 10001 cells in human D4.2 receptor established in mitogenesis assay
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Target
D(2) dopamine receptor
(Homo sapiens (Human))
University Of Toronto
Curated by
PDSP K
i
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BDBM84637
(CAS_85760-74-3 | CHEMBL240773 | NSC_54562 | QUINPI...)
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EC50: 7.60nM
Assay Description:
In vitro inhibition of forskolin-stimulated cAMP accumulation in GH4C1 cells transfected with the human Dopamine D2 receptor
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Target
D(2) dopamine receptor
(Homo sapiens (Human))
University Of Toronto
Curated by
PDSP K
i
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Ligand
BDBM84637
(CAS_85760-74-3 | CHEMBL240773 | NSC_54562 | QUINPI...)
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EC50: 3.70nM
Assay Description:
Effective dose was measured by the stimulation of mitogenesis at Dopamine receptor D4.2
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Target
D(2) dopamine receptor
(Rattus norvegicus (rat))
Dupont Pharmaceuticals
Curated by
PDSP K
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Ligand
BDBM84637
(CAS_85760-74-3 | CHEMBL240773 | NSC_54562 | QUINPI...)
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Affinity Data
EC50: 2.20nM
Assay Description:
Agonist activity by measuring the [3H]thymidine uptake against Dopamine receptor D2L from rat
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Target
D(3) dopamine receptor
(Rattus norvegicus (Rat))
U. 109
Curated by
PDSP K
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Ligand
BDBM84637
(CAS_85760-74-3 | CHEMBL240773 | NSC_54562 | QUINPI...)
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Affinity Data
EC50: 1.70nM
Assay Description:
Agonist activity by measuring the [3H]thymidine uptake against Dopamine receptor D3 from rat
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Target
D(2) dopamine receptor
(Rattus norvegicus (rat))
Dupont Pharmaceuticals
Curated by
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BDBM84637
(CAS_85760-74-3 | CHEMBL240773 | NSC_54562 | QUINPI...)
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Affinity Data
Kd: 2.30E+3nM
Assay Description:
In vitro affinity at mutant D2 receptor (S197A) in C6 (glioma) cell membranes.
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D(2) dopamine receptor
(Homo sapiens (Human))
University Of Toronto
Curated by
PDSP K
i
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Ligand
BDBM84637
(CAS_85760-74-3 | CHEMBL240773 | NSC_54562 | QUINPI...)
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Affinity Data
EC50: 2.20nM
Assay Description:
Effective concentration was determined as thymidine uptake in CHO-L6 cells transfected with the rat Dopamine receptor D2L by mitogenesis assay (intri...
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D(3) dopamine receptor
(Homo sapiens (Human))
Università
Curated by
ChEMBL
Ligand
BDBM84637
(CAS_85760-74-3 | CHEMBL240773 | NSC_54562 | QUINPI...)
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Affinity Data
EC50: 1.70nM
Assay Description:
Effective concentration was determined as thymidine uptake in CHO-L6 cells transfected with the rat Dopamine receptor D3 by mitogenesis assay (intrin...
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D(3) dopamine receptor
(Homo sapiens (Human))
Università
Curated by
ChEMBL
Ligand
BDBM84637
(CAS_85760-74-3 | CHEMBL240773 | NSC_54562 | QUINPI...)
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Affinity Data
EC50: 3.10nM
Assay Description:
Intrinsic activity in mitogenesis assay using Dopamine receptor D3 expressing CHO cells
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Target
D(3) dopamine receptor
(Rattus norvegicus (Rat))
U. 109
Curated by
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Ligand
BDBM84637
(CAS_85760-74-3 | CHEMBL240773 | NSC_54562 | QUINPI...)
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Affinity Data
EC50: 80nM
Assay Description:
Basal binding towards Dopamine receptor D3 was evaluated using [35S]- GTP-gamma S radioligand
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D(4) dopamine receptor
(Homo sapiens (Human))
Washington University
Curated by
PDSP K
i
Database
Ligand
BDBM84637
(CAS_85760-74-3 | CHEMBL240773 | NSC_54562 | QUINPI...)
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Affinity Data
EC50: 19nM
Assay Description:
Effective concentration from [3H]thymidine uptake assay in CHO10001 cells expressing human Dopamine receptor D4.2
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D(3) dopamine receptor
(Homo sapiens (Human))
Università
Curated by
ChEMBL
Ligand
BDBM84637
(CAS_85760-74-3 | CHEMBL240773 | NSC_54562 | QUINPI...)
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Affinity Data
EC50: 1.40nM
Assay Description:
Effective concentration in [3H]thymidine uptake assay by CHO dhfr- mutant cells expressing human D3 receptor
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Target
D(4) dopamine receptor
(Homo sapiens (Human))
Washington University
Curated by
PDSP K
i
Database
Ligand
BDBM84637
(CAS_85760-74-3 | CHEMBL240773 | NSC_54562 | QUINPI...)
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Affinity Data
EC50: 49nM
Assay Description:
Effective concentration for [35S]GTP-gamma-S, binding in CHO-K1 cells expressing human dopamine D4 receptor
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D(3) dopamine receptor
(Homo sapiens (Human))
Università
Curated by
ChEMBL
Ligand
BDBM84637
(CAS_85760-74-3 | CHEMBL240773 | NSC_54562 | QUINPI...)
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Affinity Data
EC50: 2.60nM
Assay Description:
Effective concentration against dopamine D3 receptor
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Target
D(4) dopamine receptor
(Homo sapiens (Human))
Washington University
Curated by
PDSP K
i
Database
Ligand
BDBM84637
(CAS_85760-74-3 | CHEMBL240773 | NSC_54562 | QUINPI...)
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Affinity Data
EC50: 1.40nM
Assay Description:
Activity at human D4.2 receptor assessed as [3H]thymidine incorporation in CHO 10001 cells by mitogenesis assay
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Target
D(4) dopamine receptor
(Homo sapiens (Human))
Washington University
Curated by
PDSP K
i
Database
Ligand
BDBM84637
(CAS_85760-74-3 | CHEMBL240773 | NSC_54562 | QUINPI...)
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Affinity Data
EC50: 49nM
Assay Description:
Activity at human D4.4 receptor expressed in CHOK1 cells assessed as stimulation of [35S]GTP-gammaS binding
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Target
D(2) dopamine receptor
(Rattus norvegicus (rat))
Dupont Pharmaceuticals
Curated by
PDSP K
i
Database
Ligand
BDBM84637
(CAS_85760-74-3 | CHEMBL240773 | NSC_54562 | QUINPI...)
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Affinity Data
EC50: 9nM
Assay Description:
Activity at rat dopamine D2L receptor expressed in HEK293 cells assessed as inhibition of forskolin-stimulated cAMP production
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Target
D(4) dopamine receptor
(Homo sapiens (Human))
Washington University
Curated by
PDSP K
i
Database
Ligand
BDBM84637
(CAS_85760-74-3 | CHEMBL240773 | NSC_54562 | QUINPI...)
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Affinity Data
EC50: 5nM
Assay Description:
Binding affinity to human cloned dopamine D4 receptor
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Target
D(4) dopamine receptor
(Homo sapiens (Human))
Washington University
Curated by
PDSP K
i
Database
Ligand
BDBM84637
(CAS_85760-74-3 | CHEMBL240773 | NSC_54562 | QUINPI...)
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Affinity Data
EC50: 9.90nM
Assay Description:
Effective concentration for [3H]thymidine uptake in growing CHO cells stably expressing the dopamine D4.2 receptor
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D(2) dopamine receptor
(Homo sapiens (Human))
University Of Toronto
Curated by
PDSP K
i
Database
Ligand
BDBM84637
(CAS_85760-74-3 | CHEMBL240773 | NSC_54562 | QUINPI...)
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Affinity Data
EC50: 240nM
Assay Description:
Agonist activity at dopamine D2 receptor expressed in HEK293 cells by by [35S]GTPgammaS binding assay
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Target
D(3) dopamine receptor
(Homo sapiens (Human))
Università
Curated by
ChEMBL
Ligand
BDBM84637
(CAS_85760-74-3 | CHEMBL240773 | NSC_54562 | QUINPI...)
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Affinity Data
EC50: 8.40nM
Assay Description:
Agonist activity at human dopamine D3 receptor expressed in CHOp cells assessed as stimulation of mitogenesis incubated for 24 hrs by [3H]thymidine i...
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D(4) dopamine receptor
(Homo sapiens (Human))
Washington University
Curated by
PDSP K
i
Database
Ligand
BDBM84637
(CAS_85760-74-3 | CHEMBL240773 | NSC_54562 | QUINPI...)
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EC50: 31nM
Assay Description:
In vitro for its ability to displace [3H]- spiperone from cloned human Dopamine receptor D4 expressed in CHO cells
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D(2) dopamine receptor
(Homo sapiens (Human))
University Of Toronto
Curated by
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i
Database
Ligand
BDBM84637
(CAS_85760-74-3 | CHEMBL240773 | NSC_54562 | QUINPI...)
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EC50: 1.20nM
Assay Description:
Agonist activity at N-terminal flag-tagged D2S receptor (unknown origin) expressed in HEK293 cells coexpressing renilla luciferase 2-tagged GalphaoA ...
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D(2) dopamine receptor
(Homo sapiens (Human))
University Of Toronto
Curated by
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i
Database
Ligand
BDBM84637
(CAS_85760-74-3 | CHEMBL240773 | NSC_54562 | QUINPI...)
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EC50: 64nM
Assay Description:
Agonist activity at ARMS2-PK2 tagged D2S receptor (unknown origin) expressed in HEK293 cells assessed as induction of EA-tagged beta-arrestin-2 recru...
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D(2) dopamine receptor
(Homo sapiens (Human))
University Of Toronto
Curated by
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i
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Ligand
BDBM84637
(CAS_85760-74-3 | CHEMBL240773 | NSC_54562 | QUINPI...)
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EC50: 151nM
Assay Description:
Agonist activity at N-terminal flag-tagged D2S receptor (unknown origin) expressed in HEK293 cells assessed as induction of renilla luciferase 2-tagg...
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D(2) dopamine receptor
(Homo sapiens (Human))
University Of Toronto
Curated by
PDSP K
i
Database
Ligand
BDBM84637
(CAS_85760-74-3 | CHEMBL240773 | NSC_54562 | QUINPI...)
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EC50: 295nM
Assay Description:
Agonist activity at N-terminal flag-tagged D2S receptor (unknown origin) expressed in HEK293 cells assessed as induction of renilla luciferase 2-tagg...
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D(2) dopamine receptor
(Homo sapiens (Human))
University Of Toronto
Curated by
PDSP K
i
Database
Ligand
BDBM84637
(CAS_85760-74-3 | CHEMBL240773 | NSC_54562 | QUINPI...)
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Affinity Data
EC50: 5.90nM
Assay Description:
Agonist activity at N-terminal flag-tagged D2S receptor (unknown origin) expressed in HEK293 cells coexpressing renilla luciferase 2-tagged Galphai3 ...
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D(2) dopamine receptor
(Homo sapiens (Human))
University Of Toronto
Curated by
PDSP K
i
Database
Ligand
BDBM84637
(CAS_85760-74-3 | CHEMBL240773 | NSC_54562 | QUINPI...)
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EC50: 3nM
Assay Description:
Agonist activity at N-terminal flag-tagged D2S receptor (unknown origin) expressed in HEK293 cells coexpressing renilla luciferase 2-tagged Galphai1 ...
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D(2) dopamine receptor
(Homo sapiens (Human))
University Of Toronto
Curated by
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i
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Ligand
BDBM84637
(CAS_85760-74-3 | CHEMBL240773 | NSC_54562 | QUINPI...)
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EC50: 5.10nM
Assay Description:
Agonist activity at N-terminal flag-tagged D2S receptor (unknown origin) expressed in HEK293 cells coexpressing renilla luciferase 2-tagged Galphai2 ...
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D(2) dopamine receptor
(Rattus norvegicus (rat))
Dupont Pharmaceuticals
Curated by
PDSP K
i
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Ligand
BDBM84637
(CAS_85760-74-3 | CHEMBL240773 | NSC_54562 | QUINPI...)
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Kd: 6.70E+3nM
Assay Description:
In vitro affinity at mutant D2 receptor (S194A) in C6 (glioma) cell membranes.
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D(2) dopamine receptor
(Rattus norvegicus (rat))
Dupont Pharmaceuticals
Curated by
PDSP K
i
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Ligand
BDBM84637
(CAS_85760-74-3 | CHEMBL240773 | NSC_54562 | QUINPI...)
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Kd: 1.90E+3nM
Assay Description:
In vitro affinity at wild type Dopamine receptor D2 on C6 (glioma) cell membranes.
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D(2) dopamine receptor
(Homo sapiens (Human))
University Of Toronto
Curated by
PDSP K
i
Database
Ligand
BDBM84637
(CAS_85760-74-3 | CHEMBL240773 | NSC_54562 | QUINPI...)
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Affinity Data
EC50: 1.20nM
Assay Description:
Agonist activity at human Dopamine D2S receptor expressed in HEK293T cell membranes coexpressing GalphaoA incubated for 30 mins measured after 75 min...
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D(2) dopamine receptor
(Rattus norvegicus (rat))
Dupont Pharmaceuticals
Curated by
PDSP K
i
Database
Ligand
BDBM84637
(CAS_85760-74-3 | CHEMBL240773 | NSC_54562 | QUINPI...)
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Affinity Data
Kd: 3.50E+3nM
Assay Description:
In vitro affinity at mutant D2 receptor (S194A) in C6 (glioma) cell membranes.
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