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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 4 hits in this display   

TargetMu-type opioid receptor(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50286102(CHEMBL353736 | Morphinan Cyclic Imine analogue)
Affinity DataIC50:  0.890nMAssay Description:Compound was tested for its ability to displace [3H]-DAMGO from mu opioid receptor in hartley guinea pig brain membrane in the presence of 100 nM of ...More data for this Ligand-Target Pair
In DepthDetails Article
TargetDelta-type opioid receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50286102(CHEMBL353736 | Morphinan Cyclic Imine analogue)
Affinity DataIC50:  12nMAssay Description:Compound was tested for its ability to displace [3H]-Cl-DPDPE from delta opioid receptor in hartley guinea pig brain membrane in the presence of 100 ...More data for this Ligand-Target Pair
In DepthDetails Article
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
TBA

Curated by ChEMBL
LigandPNGBDBM50286102(CHEMBL353736 | Morphinan Cyclic Imine analogue)
Affinity DataIC50:  97nMAssay Description:Compound was tested for its ability to displace bremazocine from Opioid receptor kappa 2 in hartley guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails Article
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
TBA

Curated by ChEMBL
LigandPNGBDBM50286102(CHEMBL353736 | Morphinan Cyclic Imine analogue)
Affinity DataIC50:  331nMAssay Description:Compound was tested for its ability to displace bremazocine from Opioid receptor kappa 2 in hartley guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails Article