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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
8
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Target
Solute carrier organic anion transporter family member
(Danio rerio (Zebrafish))
Rudjer Boskovic Institute
Ligand
BDBM200235
(Rifampicin | cid_5381226)
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Affinity Data
Ki: 1.27E+4nM
Assay Description:
In the inhibition experiments, the cells were preincubated for 20 s with test compounds, followed by a 5-min incubation with [3H]E3S (5 nM) or 30-min...
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Target
Ubiquitin carboxyl-terminal hydrolase isozyme L1
(Homo sapiens (Human))
University Of Delaware
Ligand
BDBM200235
(Rifampicin | cid_5381226)
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Affinity Data
IC50: 1.95E+4nM
pH: 7.5 T: 2°C
Assay Description:
Ubiquitin-7-amino-4-methylcoumarin (Ub-AMC) was generated as previously described.(7) The enzymatic reaction was conducted in fluorometric assay buff...
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Target Info
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MMDB
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Target
Ubiquitin carboxyl-terminal hydrolase 2
(Homo sapiens (Human))
University Of Delaware
Ligand
BDBM200235
(Rifampicin | cid_5381226)
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Affinity Data
IC50: 2.12E+4nM
pH: 7.5 T: 2°C
Assay Description:
Ubiquitin-7-amino-4-methylcoumarin (Ub-AMC) was generated as previously described.(7) The enzymatic reaction was conducted in fluorometric assay buff...
More data for this Ligand-Target Pair
Target Info
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MMDB
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KEGG
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B.MOAD
antibodypedia
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Target
Ubiquitin carboxyl-terminal hydrolase isozyme L3
(Homo sapiens (Human))
University Of Delaware
Ligand
BDBM200235
(Rifampicin | cid_5381226)
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Affinity Data
IC50: 2.48E+4nM
pH: 7.5 T: 2°C
Assay Description:
Ubiquitin-7-amino-4-methylcoumarin (Ub-AMC) was generated as previously described.(7) The enzymatic reaction was conducted in fluorometric assay buff...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
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KEGG
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B.MOAD
antibodypedia
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Article
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Target
Ubiquitin carboxyl-terminal hydrolase 15
(Homo sapiens (Human))
University Of Delaware
Ligand
BDBM200235
(Rifampicin | cid_5381226)
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Affinity Data
IC50: 4.61E+4nM
pH: 7.5 T: 2°C
Assay Description:
Ubiquitin-7-amino-4-methylcoumarin (Ub-AMC) was generated as previously described.(7) The enzymatic reaction was conducted in fluorometric assay buff...
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Target Info
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Target
Ubiquitin carboxyl-terminal hydrolase isozyme L5
(Homo sapiens (Human))
University Of Delaware
Ligand
BDBM200235
(Rifampicin | cid_5381226)
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Affinity Data
IC50: 6.28E+4nM
pH: 7.5 T: 2°C
Assay Description:
Ubiquitin-7-amino-4-methylcoumarin (Ub-AMC) was generated as previously described.(7) The enzymatic reaction was conducted in fluorometric assay buff...
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Target Info
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Target
Isocitrate lyase
(Mycobacterium tuberculosis)
Birla Institute Of Technology
Ligand
BDBM200235
(Rifampicin | cid_5381226)
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Affinity Data
IC50: >7.59E+4nM
T: 2°C
Assay Description:
Isocitrate lyase activity was determined at 37°C by measuringthe formation of glyoxylate phenylhydrazone at 324 nm [Bai et al., Drug Dev. Res., 6...
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Target
Cystic fibrosis transmembrane conductance regulator
(Homo sapiens (Human))
Southern Research Institute
Curated by
PubChem BioAssay
Ligand
BDBM200235
(Rifampicin | cid_5381226)
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Affinity Data
EC50: >5.00E+4nM
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