Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 30 hits in this display
BDBM3033(3-{23-methyl-14-oxo-3,13,23-triazahexacyclo[14.7.0...)
BDBM3033(3-{23-methyl-14-oxo-3,13,23-triazahexacyclo[14.7.0...)
BDBM3033(3-{23-methyl-14-oxo-3,13,23-triazahexacyclo[14.7.0...)
BDBM3033(3-{23-methyl-14-oxo-3,13,23-triazahexacyclo[14.7.0...)
BDBM3033(3-{23-methyl-14-oxo-3,13,23-triazahexacyclo[14.7.0...)
Ki: >1.90E+4nMAssay Description:Kinase was assayed in 384-well polypropylene plate format. The compound was mixed with kinase and biotinylated peptide substrate and incubated. After...More data for this Ligand-Target Pair
BDBM3033(3-{23-methyl-14-oxo-3,13,23-triazahexacyclo[14.7.0...)
BDBM3033(3-{23-methyl-14-oxo-3,13,23-triazahexacyclo[14.7.0...)
BDBM3033(3-{23-methyl-14-oxo-3,13,23-triazahexacyclo[14.7.0...)
BDBM3033(3-{23-methyl-14-oxo-3,13,23-triazahexacyclo[14.7.0...)
BDBM3033(3-{23-methyl-14-oxo-3,13,23-triazahexacyclo[14.7.0...)
BDBM3033(3-{23-methyl-14-oxo-3,13,23-triazahexacyclo[14.7.0...)
BDBM3033(3-{23-methyl-14-oxo-3,13,23-triazahexacyclo[14.7.0...)
BDBM3033(3-{23-methyl-14-oxo-3,13,23-triazahexacyclo[14.7.0...)
BDBM3033(3-{23-methyl-14-oxo-3,13,23-triazahexacyclo[14.7.0...)
BDBM3033(3-{23-methyl-14-oxo-3,13,23-triazahexacyclo[14.7.0...)
BDBM3033(3-{23-methyl-14-oxo-3,13,23-triazahexacyclo[14.7.0...)
BDBM3033(3-{23-methyl-14-oxo-3,13,23-triazahexacyclo[14.7.0...)
BDBM3033(3-{23-methyl-14-oxo-3,13,23-triazahexacyclo[14.7.0...)
BDBM3033(3-{23-methyl-14-oxo-3,13,23-triazahexacyclo[14.7.0...)
BDBM3033(3-{23-methyl-14-oxo-3,13,23-triazahexacyclo[14.7.0...)
BDBM3033(3-{23-methyl-14-oxo-3,13,23-triazahexacyclo[14.7.0...)
BDBM3033(3-{23-methyl-14-oxo-3,13,23-triazahexacyclo[14.7.0...)
IC50: 5.80E+3nMpH: 7.2 T: 2°CAssay Description:The activity of MLCK is measured by its ability to transfer 32P from [gamma-32P]ATP to myosin light-chain.More data for this Ligand-Target Pair
BDBM3033(3-{23-methyl-14-oxo-3,13,23-triazahexacyclo[14.7.0...)
BDBM3033(3-{23-methyl-14-oxo-3,13,23-triazahexacyclo[14.7.0...)
BDBM3033(3-{23-methyl-14-oxo-3,13,23-triazahexacyclo[14.7.0...)
IC50: 6.20E+3nMAssay Description:The activity of cGPK, activated by cGMP, is measured by its ability to transfer phosphate from [gamma-32P]ATP to histone.More data for this Ligand-Target Pair
BDBM3033(3-{23-methyl-14-oxo-3,13,23-triazahexacyclo[14.7.0...)
BDBM3033(3-{23-methyl-14-oxo-3,13,23-triazahexacyclo[14.7.0...)
BDBM3033(3-{23-methyl-14-oxo-3,13,23-triazahexacyclo[14.7.0...)
BDBM3033(3-{23-methyl-14-oxo-3,13,23-triazahexacyclo[14.7.0...)
IC50: >1.00E+5nMAssay Description:The activity of PKA, activated by cAMP, is measured by its ability to transfer phosphate from [gamma-32P]ATP to histone.More data for this Ligand-Target Pair
BDBM3033(3-{23-methyl-14-oxo-3,13,23-triazahexacyclo[14.7.0...)