Compile Data Set for Download or QSAR
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Found 2 Enz. Inhib. hit(s) with Target = 'Vasopressin V1a receptor' and Ligand = 'BDBM50319797'
TargetVasopressin V1a receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50319797((4-(benzo[b]thiophen-3-yl)-3-methoxyphenyl)((1S,5R...)
Affinity DataKi:  0.790nMAssay Description:Displacement [3H]Arg human recombinant Vasopressin V1a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50319797((4-(benzo[b]thiophen-3-yl)-3-methoxyphenyl)((1S,5R...)
Affinity DataIC50:  41nMAssay Description:Antagonist activity at human Vasopressin V1a receptor assessed as inhibition of intracellular calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed