Compile Data Set for Download or QSAR
maximum 50k data
Found 107 of ic50 for UniProtKB: Q8HZR1
TargetProstaglandin G/H synthase 1(Canis familiaris)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50137420(2-[5-(4-Ethoxy-phenyl)-3-trifluoromethyl-pyrazol-1...)
Affinity DataIC50:  50nMAssay Description:In vitro inhibitory activity against cannine prostaglandin G/H synthase 1.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Canis familiaris)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50179624(5-(2,3-dimethylphenoxy)-1-(5-(methylsulfonyl)pyrid...)
Affinity DataIC50:  100nMAssay Description:Inhibition of COX1 by canine whole blood assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Canis familiaris)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50179602(1-(5-(methylsulfonyl)pyridin-2-yl)-5-(5,6,7,8-tetr...)
Affinity DataIC50:  100nMAssay Description:Inhibition of COX1 by canine whole blood assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Canis familiaris)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50179609(1-(5-(methylsulfonyl)pyridin-2-yl)-5-(phenylthio)-...)
Affinity DataIC50:  200nMAssay Description:Inhibition of COX1 by canine whole blood assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Canis familiaris)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50137411(2-[3-Difluoromethyl-5-(4-methoxy-phenyl)-pyrazol-1...)
Affinity DataIC50:  200nMAssay Description:In vitro inhibitory activity against cannine prostaglandin G/H synthase 1.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Canis familiaris)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50179598(1-(5-(methylsulfonyl)pyridin-2-yl)-5-(propylthio)-...)
Affinity DataIC50:  200nMAssay Description:Inhibition of COX1 by canine whole blood assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Canis familiaris)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50137423(2-(4-Chloro-3-difluoromethyl-5-phenyl-pyrazol-1-yl...)
Affinity DataIC50:  330nMAssay Description:In vitro inhibitory activity against cannine prostaglandin G/H synthase 1.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Canis familiaris)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50179596(5-(cyclopentylmethoxy)-1-(5-(methylsulfonyl)pyridi...)
Affinity DataIC50:  400nMAssay Description:Inhibition of COX1 by canine whole blood assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Canis familiaris)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50179600(5-(2-fluorobenzylthio)-1-(5-(methylsulfonyl)pyridi...)
Affinity DataIC50:  600nMAssay Description:Inhibition of COX1 by canine whole blood assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Canis familiaris)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50137438(5-Methanesulfonyl-2-[5-(4-methoxy-phenyl)-3-triflu...)
Affinity DataIC50:  830nMAssay Description:In vitro inhibitory activity against cannine prostaglandin G/H synthase 1.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Canis familiaris)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50137428(2-[3-Difluoromethyl-5-(4-methylsulfanyl-phenyl)-py...)
Affinity DataIC50:  900nMAssay Description:In vitro inhibitory activity against cannine prostaglandin G/H synthase 1.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Canis familiaris)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50179616(5-(benzylthio)-1-(5-(methylsulfonyl)pyridin-2-yl)-...)
Affinity DataIC50:  900nMAssay Description:Inhibition of COX1 by canine whole blood assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Canis familiaris)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50137410(2-[5-(4-Bromo-phenyl)-3-difluoromethyl-pyrazol-1-y...)
Affinity DataIC50:  1.00E+3nMAssay Description:In vitro inhibitory activity against cannine prostaglandin G/H synthase 1.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Canis familiaris)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50179631(5-(sec-butylthio)-1-(5-(methylsulfonyl)pyridin-2-y...)
Affinity DataIC50:  1.50E+3nMAssay Description:Inhibition of COX1 by canine whole blood assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Canis familiaris)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50137424(2-[4-Chloro-5-(3-chloro-4-methoxy-phenyl)-3-difluo...)
Affinity DataIC50:  1.50E+3nMAssay Description:In vitro inhibitory activity against cannine prostaglandin G/H synthase 1.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Canis familiaris)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50137437(5-Methanesulfonyl-2-[5-(4-methylsulfanyl-phenyl)-3...)
Affinity DataIC50:  1.90E+3nMAssay Description:In vitro inhibitory activity against cannine prostaglandin G/H synthase 1.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Canis familiaris)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50176555(3-(difluoromethyl)-5-(3-methylpiperidin-1-yl)-1-(5...)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibitory activity against COX1 in canine whole bloodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Canis familiaris)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50137427(2-(4-Bromo-3-difluoromethyl-5-phenyl-pyrazol-1-yl)...)
Affinity DataIC50:  2.00E+3nMAssay Description:In vitro inhibitory activity against cannine prostaglandin G/H synthase 1.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Canis familiaris)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50179608(5-(2-ethoxyethylthio)-1-(5-(methylsulfonyl)pyridin...)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of COX1 by canine whole blood assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Canis familiaris)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50182350(2-(furan-2-yl)-5-(1-(5-(methylsulfonyl)pyridin-2-y...)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of COX1 in canine whole bloodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Canis familiaris)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50182339(2-(furan-2-yl)-5-(1-(5-(methylsulfonyl)pyridin-2-y...)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of COX1 in canine whole bloodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Canis familiaris)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50182349(5-(methylsulfonyl)-2-(5-(4-(thiazol-5-yl)phenyl)-3...)
Affinity DataIC50:  2.70E+3nMAssay Description:Inhibition of COX1 in canine whole bloodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Canis familiaris)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50137439(2-[5-(2-Fluoro-4-methoxy-phenyl)-3-trifluoromethyl...)
Affinity DataIC50:  2.80E+3nMAssay Description:In vitro inhibitory activity against cannine prostaglandin G/H synthase 1.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Canis familiaris)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50179621(5-(cyclohexylthio)-1-(5-(methylsulfonyl)pyridin-2-...)
Affinity DataIC50:  3.20E+3nMAssay Description:Inhibition of COX1 by canine whole blood assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Canis familiaris)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50179613(5-(4-methylpentylthio)-1-(5-(methylsulfonyl)pyridi...)
Affinity DataIC50:  3.30E+3nMAssay Description:Inhibition of COX1 by canine whole blood assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Canis familiaris)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50176547(5-(3-methylbutan-2-ylamino)-1-(5-(methylsulfonyl)p...)
Affinity DataIC50:  3.40E+3nMAssay Description:Inhibitory activity against COX1 in canine whole bloodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Canis familiaris)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50182338(2-(5-(4-(furan-2-yl)-3-methylphenyl)-3-(trifluorom...)
Affinity DataIC50:  3.40E+3nMAssay Description:Inhibition of COX1 in canine whole bloodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Canis familiaris)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50179628(1-(5-(methylsulfonyl)pyridin-2-yl)-5-(pentylthio)-...)
Affinity DataIC50:  3.50E+3nMAssay Description:Inhibition of COX1 by canine whole blood assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Canis familiaris)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50182353(2-(3-(difluoromethyl)-5-(3-methyl-4-(thiazol-4-yl)...)
Affinity DataIC50:  3.80E+3nMAssay Description:Inhibition of COX1 in canine whole bloodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Canis familiaris)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50176532(6-(4-cyano-3-(difluoromethyl)-5-(2-methylbutylamin...)
Affinity DataIC50:  4.00E+3nMAssay Description:Inhibitory activity against COX1 in canine whole bloodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Canis familiaris)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50176541(6-(4-cyano-5-(2-methylbutylamino)-3-(trifluorometh...)
Affinity DataIC50:  4.50E+3nMAssay Description:Inhibitory activity against COX1 in canine whole bloodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Canis familiaris)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50182334(2-(3-(difluoromethyl)-5-(3-fluoro-4-(furan-2-yl)ph...)
Affinity DataIC50:  5.00E+3nMAssay Description:Inhibition of COX1 in canine whole bloodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Canis familiaris)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50182352(2-(5-(3-chloro-4-(furan-2-yl)phenyl)-3-(difluorome...)
Affinity DataIC50:  5.50E+3nMAssay Description:Inhibition of COX1 in canine whole bloodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Canis familiaris)
Pfizer

Curated by ChEMBL
LigandPNGBDBM11639(4-[5-(4-methylphenyl)-3-(trifluoromethyl)-1H-pyraz...)
Affinity DataIC50:  5.57E+3nMAssay Description:In vitro inhibitory activity against cannine prostaglandin G/H synthase 1.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Canis familiaris)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50176533(1-(5-(methylsulfonyl)pyridin-2-yl)-5-(thiophen-2-y...)
Affinity DataIC50:  5.60E+3nMAssay Description:Inhibitory activity against COX1 in canine whole bloodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Canis familiaris)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50176539(1-(5-(methylsulfonyl)pyridin-2-yl)-5-(pentan-3-yla...)
Affinity DataIC50:  6.70E+3nMAssay Description:Inhibitory activity against COX1 in canine whole bloodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Canis familiaris)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50176546(6-(4-cyano-3-(difluoromethyl)-5-((cis)-3,5-dimethy...)
Affinity DataIC50:  7.00E+3nMAssay Description:Inhibitory activity against COX1 in canine whole bloodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Canis familiaris)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50179593(5-(2-methylcyclohexyloxy)-1-(5-(methylsulfonyl)pyr...)
Affinity DataIC50:  7.10E+3nMAssay Description:Inhibition of COX1 by canine whole blood assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Canis familiaris)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50179595(5-(3-methylcyclopentyloxy)-1-(5-(methylsulfonyl)py...)
Affinity DataIC50:  7.60E+3nMAssay Description:Inhibition of COX1 by canine whole blood assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Canis familiaris)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50137435(2-(4-Chloro-5-phenyl-3-trifluoromethyl-pyrazol-1-y...)
Affinity DataIC50:  7.90E+3nMAssay Description:In vitro inhibitory activity against cannine prostaglandin G/H synthase 1.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Canis familiaris)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50179611(5-(cycloheptyloxy)-1-(5-(methylsulfonyl)pyridin-2-...)
Affinity DataIC50:  8.00E+3nMAssay Description:Inhibition of COX1 by canine whole blood assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Canis familiaris)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50137432(2-(3-Difluoromethyl-4-methyl-5-phenyl-pyrazol-1-yl...)
Affinity DataIC50:  9.10E+3nMAssay Description:In vitro inhibitory activity against cannine prostaglandin G/H synthase 1.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Canis familiaris)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50137442(2-[3-Difluoromethyl-5-(3-fluoro-4-methoxy-phenyl)-...)
Affinity DataIC50:  9.90E+3nMAssay Description:In vitro inhibitory activity against cannine prostaglandin G/H synthase 1.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Canis familiaris)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50179592(5-isobutoxy-1-(5-(methylsulfonyl)pyridin-2-yl)-3-(...)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibition of COX1 by canine whole blood assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Canis familiaris)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50137418(2-(3-Difluoromethyl-5-p-tolyl-pyrazol-1-yl)-5-meth...)
Affinity DataIC50:  1.00E+4nMAssay Description:In vitro inhibitory activity against cannine prostaglandin G/H synthase 1.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Canis familiaris)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50179601(5-(cyclohex-3-enylmethoxy)-1-(5-(methylsulfonyl)py...)
Affinity DataIC50:  1.06E+4nMAssay Description:Inhibition of COX1 by canine whole blood assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Canis familiaris)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50176556(5-(2-methylcyclohexylamino)-1-(5-(methylsulfonyl)p...)
Affinity DataIC50:  1.08E+4nMAssay Description:Inhibitory activity against COX1 in canine whole bloodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Canis familiaris)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50182346(2-(5-(3-methyl-4-(oxazol-2-yl)phenyl)-3-(trifluoro...)
Affinity DataIC50:  1.11E+4nMAssay Description:Inhibition of COX1 in canine whole bloodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Canis familiaris)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50179591(5-(3-methylbutan-2-yloxy)-1-(5-(methylsulfonyl)pyr...)
Affinity DataIC50:  1.18E+4nMAssay Description:Inhibition of COX1 by canine whole blood assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Canis familiaris)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50182343(2-(3-(difluoromethyl)-5-(4-(furan-2-yl)phenyl)-1H-...)
Affinity DataIC50:  1.20E+4nMAssay Description:Inhibition of COX1 in canine whole bloodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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