Compile Data Set for Download or QSAR
maximum 50k data
Found 73 of ic50 data for polymerid = 9133
LigandPNGBDBM50462596(CHEMBL4242659)
Affinity DataIC50:  0.290nMAssay Description:Inhibition of PI3Kdelta in Balb/c mouse splenocytes-derived B cells assessed as reduction in anti-IgM antibody-stimulated B cell proliferation after ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50462587(CHEMBL4250271)
Affinity DataIC50:  0.410nMAssay Description:Inhibition of PI3Kdelta in Balb/c mouse splenocytes-derived B cells assessed as reduction in anti-IgM antibody-stimulated B cell proliferation after ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50462594(CHEMBL4249087)
Affinity DataIC50:  1.40nMAssay Description:Inhibition of PI3Kdelta in Balb/c mouse splenocytes-derived B cells assessed as reduction in anti-IgM antibody-stimulated B cell proliferation after ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50462588(CHEMBL4248505)
Affinity DataIC50:  1.5nMAssay Description:Inhibition of PI3Kdelta in Balb/c mouse splenocytes-derived B cells assessed as reduction in anti-IgM antibody-stimulated B cell proliferation after ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50462589(CHEMBL4247328)
Affinity DataIC50:  1.5nMAssay Description:Inhibition of PI3Kdelta in Balb/c mouse splenocytes-derived B cells assessed as reduction in anti-IgM antibody-stimulated B cell proliferation after ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50380313(CHEMBL1234354 | US8633204, 286)
Affinity DataIC50:  1.60nMAssay Description:Antagonist activity was determined against beta-1 adrenergic receptor in spontaneously beating rat atriaMore data for this Ligand-Target Pair
In DepthDetails
LigandPNGBDBM50461379(CHEMBL4227156)
Affinity DataIC50:  2.10nMAssay Description:Inhibition of PI3Kdelta in Balb/c mouse splenocytes-derived B cells assessed as reduction in anti-IgM antibody-stimulated B cell proliferation after ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50575900(CHEMBL4853960)
Affinity DataIC50:  2.20nMAssay Description:Inhibition of mouse PI3KdeltaMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
LigandPNGBDBM50403096(CHEMBL2216895)
Affinity DataIC50:  2.5nMAssay Description:Inhibition of PI3Kdelta in Balb/c mouse B cells assessed as inhibition of antiIgM-induced Akt phosphorylation at ser 473 residue preincubated for 45 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50461373(CHEMBL4228899)
Affinity DataIC50:  2.60nMAssay Description:Inhibition of PI3Kdelta in Balb/c mouse splenocytes-derived B cells assessed as reduction in anti-IgM antibody-stimulated B cell proliferation after ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50462595(CHEMBL4250966)
Affinity DataIC50:  2.90nMAssay Description:Inhibition of PI3Kdelta in Balb/c mouse splenocytes-derived B cells assessed as reduction in anti-IgM antibody-stimulated B cell proliferation after ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM346183(US10202371, Example 13)
Affinity DataIC50: <3nMAssay Description:AlphaScreen (Amplified Luminescent Proximity Homogeneous Assay, ALPHA, Perkin Elmer) is a non-radioactive bead-based proximity assay technology to st...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM346184(US10202371, Example 14)
Affinity DataIC50:  4nMAssay Description:AlphaScreen (Amplified Luminescent Proximity Homogeneous Assay, ALPHA, Perkin Elmer) is a non-radioactive bead-based proximity assay technology to st...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM50232430(CHEMBL4061855 | US10214537, Example 262)
Affinity DataIC50:  4nMAssay Description:Inhibition of PI3Kdelta in mouse spleen assessed suppression of CD86More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM346182(US10202371, Example 12)
Affinity DataIC50:  4nMAssay Description:AlphaScreen (Amplified Luminescent Proximity Homogeneous Assay, ALPHA, Perkin Elmer) is a non-radioactive bead-based proximity assay technology to st...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM50557968(CHEMBL4754382)
Affinity DataIC50:  4.20nMAssay Description:Inhibition of PI3Kdelta in Balb/c mouse B cells assessed as inhibition of antiIgM-induced Akt phosphorylation at ser 473 residue preincubated for 45 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50462590(CHEMBL4244862)
Affinity DataIC50:  4.30nMAssay Description:Inhibition of PI3Kdelta in Balb/c mouse splenocytes-derived B cells assessed as reduction in anti-IgM antibody-stimulated B cell proliferation after ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50557972(CHEMBL4790186)
Affinity DataIC50:  4.5nMAssay Description:Inhibition of PI3Kdelta in Balb/c mouse B cells assessed as inhibition of antiIgM-induced Akt phosphorylation at ser 473 residue preincubated for 45 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50557969(CHEMBL4763849)
Affinity DataIC50:  4.60nMAssay Description:Inhibition of PI3Kdelta in Balb/c mouse B cells assessed as inhibition of antiIgM-induced Akt phosphorylation at ser 473 residue preincubated for 45 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50462593(CHEMBL4246031)
Affinity DataIC50:  4.80nMAssay Description:Inhibition of PI3Kdelta in Balb/c mouse splenocytes-derived B cells assessed as reduction in anti-IgM antibody-stimulated B cell proliferation after ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50239718(CHEMBL4064666 | US10214537, Example 639)
Affinity DataIC50:  5.10nMAssay Description:Antisecretory activity evaluated by the inhibition of 14C -AP uptake in isolated rabbit parietal cells stimulated by dibutyryl cyclic adenosine 3', 5...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM346173(US10202371, Example 3)
Affinity DataIC50:  6nMAssay Description:AlphaScreen (Amplified Luminescent Proximity Homogeneous Assay, ALPHA, Perkin Elmer) is a non-radioactive bead-based proximity assay technology to st...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM50462598(CHEMBL4245438)
Affinity DataIC50:  7.80nMAssay Description:Inhibition of PI3Kdelta in Balb/c mouse splenocytes-derived B cells assessed as reduction in anti-IgM antibody-stimulated B cell proliferation after ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50403081(CHEMBL2216855)
Affinity DataIC50: <10nMAssay Description:Inhibition of PI3Kdelta-mediated AKT phosphorylation in mouse Raw 264.7 cells by immunoassayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM118299(US8653092, 67)
Affinity DataIC50:  10nMAssay Description:Inhibition of PI3Kdelta in anti-CD3/CD28 stimulated mouse CD4-positive T cells assessed as reduction in T cell differentiation to Th2 cells by measur...More data for this Ligand-Target Pair
LigandPNGBDBM50203699(CHEMBL3977066)
Affinity DataIC50:  11nMAssay Description:Inhibition of PI3Kdelta in Balb/c mouse in rat B cells assessed as reduction in anti-IgM induced proliferation measured over last 16 hrs of 88 hrs by...More data for this Ligand-Target Pair
LigandPNGBDBM346179(US10202371, Example 9)
Affinity DataIC50:  11nMAssay Description:AlphaScreen (Amplified Luminescent Proximity Homogeneous Assay, ALPHA, Perkin Elmer) is a non-radioactive bead-based proximity assay technology to st...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM346171((4S,5R)-3-(2′-Amino-2-morpholin-4-yl-4′...)
Affinity DataIC50:  11.3nMAssay Description:AlphaScreen (Amplified Luminescent Proximity Homogeneous Assay, ALPHA, Perkin Elmer) is a non-radioactive bead-based proximity assay technology to st...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM217352(GS-9820)
Affinity DataIC50:  12.7nMAssay Description:Biochemical in vitro lipid kinase assays were performed by the SelectScreen® biochemical kinase assay service (Invitrogen Ltd.). A stock solution of ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM118300(US8653092, 68)
Affinity DataIC50:  15nMAssay Description:Inhibition of PI3Kdelta in Balb/c mouse splenocytes assessed as reduction in anti-IgM stimulated CD86 expression pretreated for 1 hr followed by anti...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM346181(US10202371, Example 11)
Affinity DataIC50:  20nMAssay Description:AlphaScreen (Amplified Luminescent Proximity Homogeneous Assay, ALPHA, Perkin Elmer) is a non-radioactive bead-based proximity assay technology to st...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM50462591(CHEMBL4249694)
Affinity DataIC50:  20nMAssay Description:Inhibition of PI3Kdelta in Balb/c mouse splenocytes-derived B cells assessed as reduction in anti-IgM antibody-stimulated B cell proliferation after ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM346180(US10202371, Example 10)
Affinity DataIC50:  22nMAssay Description:AlphaScreen (Amplified Luminescent Proximity Homogeneous Assay, ALPHA, Perkin Elmer) is a non-radioactive bead-based proximity assay technology to st...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM50533775(CHEMBL4588314)
Affinity DataIC50:  26nMAssay Description:Inhibition of PI3Kdelta in Balb/c mouse B cells assessed as reduction in anti-IgM induced CD86 expression preincubated for 1 hr followed by anti-IgM ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM346178(US10202371, Example 8)
Affinity DataIC50:  28nMAssay Description:AlphaScreen (Amplified Luminescent Proximity Homogeneous Assay, ALPHA, Perkin Elmer) is a non-radioactive bead-based proximity assay technology to st...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM118299(US8653092, 67)
Affinity DataIC50:  33nMAssay Description:Inhibition of PI3Kdelta in mouse spleen cells assessed as reduction in cell proliferation by measuring [3H]thymidine incorporation by beta counting b...More data for this Ligand-Target Pair
LigandPNGBDBM50203701(CHEMBL3944013)
Affinity DataIC50:  34nMAssay Description:Inhibition of PI3Kdelta in Balb/c mouse B cells assessed as reduction in anti-IgM induced CD86 expression preincubated for 1 hr followed by anti-IgM ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50203701(CHEMBL3944013)
Affinity DataIC50:  34nMAssay Description:Inhibition of PI3K-delta in mouse splenocytes assessed as inhibition anti-IgM induced CD86 expressionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM118299(US8653092, 67)
Affinity DataIC50:  48nMAssay Description:Inhibition of PI3Kdelta in Balb/c mouse splenocytes assessed as reduction in anti-IgM stimulated CD86 expression pretreated for 1 hr followed by anti...More data for this Ligand-Target Pair
LigandPNGBDBM50203699(CHEMBL3977066)
Affinity DataIC50:  48nMAssay Description:Inhibition of PI3Kdelta in Balb/c mouse splenocytes assessed as reduction in anti-IgM stimulated CD86 expression pretreated for 1 hr followed by anti...More data for this Ligand-Target Pair
LigandPNGBDBM118299(US8653092, 67)
Affinity DataIC50:  48nMAssay Description:Inhibition of PI3Kdelta in Balb/c mouse splenocytes assessed as reduction in anti-IgM stimulated CD86 expression pretreated for 1 hr followed by anti...More data for this Ligand-Target Pair
LigandPNGBDBM50203682(CHEMBL3947814)
Affinity DataIC50:  70nMAssay Description:Inhibition of PI3Kdelta in Balb/c mouse B cells assessed as reduction in anti-IgM induced CD86 expression preincubated for 1 hr followed by anti-IgM ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50203682(CHEMBL3947814)
Affinity DataIC50:  70nMAssay Description:Inhibition of PI3K-delta in mouse splenocytes assessed as inhibition anti-IgM induced CD86 expressionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50203699(CHEMBL3977066)
Affinity DataIC50:  70nMAssay Description:Inhibition of PI3Kdelta in Balb/c mouse B cells assessed as reduction in anti-IgM induced CD86 expression preincubated for 1 hr followed by anti-IgM ...More data for this Ligand-Target Pair
LigandPNGBDBM50203682(CHEMBL3947814)
Affinity DataIC50:  70nMAssay Description:Inhibition of PI3Kdelta in Balb/c mouse splenocytes assessed as reduction in anti-IgM stimulated CD86 expression pretreated for 1 hr followed by anti...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50203699(CHEMBL3977066)
Affinity DataIC50:  74nMAssay Description:Inhibition of PI3K-delta in mouse splenocytes assessed as inhibition anti-IgM induced CD86 expressionMore data for this Ligand-Target Pair
LigandPNGBDBM50533778(CHEMBL4453497)
Affinity DataIC50:  74nMAssay Description:Inhibition of PI3Kdelta in Balb/c mouse B cells assessed as reduction in anti-IgM induced CD86 expression preincubated for 1 hr followed by anti-IgM ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50203696(CHEMBL3896413)
Affinity DataIC50:  82nMAssay Description:Inhibition of PI3K-delta in mouse splenocytes assessed as inhibition anti-IgM induced CD86 expressionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM118293(US8653092, 61)
Affinity DataIC50:  84nMAssay Description:Inhibition of PI3Kdelta in Balb/c mouse splenocytes assessed as reduction in anti-IgM stimulated CD86 expression pretreated for 1 hr followed by anti...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50203685(CHEMBL3966263)
Affinity DataIC50:  85nMAssay Description:Inhibition of PI3K-delta in mouse splenocytes assessed as inhibition anti-IgM induced CD86 expressionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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