Compile Data Set for Download or QSAR
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Report error Found 4 Enz. Inhib. hit(s) for PDB: 3HVL
TargetNuclear receptor subfamily 1 group I member 2(Human)
Phenex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50030477(CHEBI:77317 | CHEMBL458767 | SR-12813)
Affinity DataEC50:  80nMAssay Description:Agonist activity at human pregnane X receptor expressed in HEK293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group I member 2(Human)
Phenex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50030477(CHEBI:77317 | CHEMBL458767 | SR-12813)
Affinity DataEC50:  220nMAssay Description:Activation of human PXRMore data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group I member 2(Human)
Phenex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50030477(CHEBI:77317 | CHEMBL458767 | SR-12813)
Affinity DataEC50:  60nMAssay Description:Agonist activity at human PXRMore data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group I member 2(Human)
Phenex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50030477(CHEBI:77317 | CHEMBL458767 | SR-12813)
Affinity DataEC50:  440nMAssay Description:Competitive binding affinity to human PXR LBD (111 to 434) by TR-FRET assayMore data for this Ligand-Target Pair