Compile Data Set for Download or QSAR
maximum 50k data
Found 4 Enz. Inhib. hit(s) with Target = 'Nuclear receptor subfamily 1 group I member 2' and Ligand = 'BDBM50030477'
TargetNuclear receptor subfamily 1 group I member 2(Homo sapiens (Human))
Phenex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50030477(CHEBI:77317 | CHEMBL458767 | SR-12813)
Affinity DataEC50:  80nMAssay Description:Agonist activity at human pregnane X receptor expressed in HEK293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group I member 2(Homo sapiens (Human))
Phenex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50030477(CHEBI:77317 | CHEMBL458767 | SR-12813)
Affinity DataEC50:  220nMAssay Description:Activation of human PXRMore data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group I member 2(Homo sapiens (Human))
Phenex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50030477(CHEBI:77317 | CHEMBL458767 | SR-12813)
Affinity DataEC50:  60nMAssay Description:Agonist activity at human PXRMore data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group I member 2(Homo sapiens (Human))
Phenex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50030477(CHEBI:77317 | CHEMBL458767 | SR-12813)
Affinity DataEC50:  440nMAssay Description:Competitive binding affinity to human PXR LBD (111 to 434) by TR-FRET assayMore data for this Ligand-Target Pair