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Report error Found 5 Enz. Inhib. hit(s) for PDB: 3KKU
TargetCruzipain(Trypanosoma cruzi)
Universidade Federal Do Rio Grande Do Sul

Curated by ChEMBL
LigandPNGBDBM50322742(CHEMBL1173694 | N-(2-(1H-benzo[d]imidazol-2-yl)eth...)
Affinity DataKi:  2.00E+3nMAssay Description:Binding affinity to Trypanosoma cruzi Cruzain assessed as inhibition constantMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedMMDB
PDB3D3D Structure (crystal)

TargetCruzipain(Trypanosoma cruzi)
Universidade Federal Do Rio Grande Do Sul

Curated by ChEMBL
LigandPNGBDBM50322742(CHEMBL1173694 | N-(2-(1H-benzo[d]imidazol-2-yl)eth...)
Affinity DataKi:  2.00E+3nMAssay Description:Inhibition of Trypanosoma cruzi cruzain assessed as Z-Phe-Arg-aminomethylcoumarin cleavage by competetive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedMMDB
PDB3D3D Structure (crystal)

TargetCruzipain(Trypanosoma cruzi)
Universidade Federal Do Rio Grande Do Sul

Curated by ChEMBL
LigandPNGBDBM50322742(CHEMBL1173694 | N-(2-(1H-benzo[d]imidazol-2-yl)eth...)
Affinity DataIC50:  800nMAssay Description:Inhibition of Trypanosoma cruzi CruzainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedMMDB
PDB3D3D Structure (crystal)

TargetCruzipain(Trypanosoma cruzi)
Universidade Federal Do Rio Grande Do Sul

Curated by ChEMBL
LigandPNGBDBM50322742(CHEMBL1173694 | N-(2-(1H-benzo[d]imidazol-2-yl)eth...)
Affinity DataIC50:  800nMAssay Description:Inhibition of Trypanosoma cruzi cruzaine expressed in Escherichia coli SG13009 using Z-FR-AMC as substrate after 5 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedMMDB
PDB3D3D Structure (crystal)

TargetCruzipain(Trypanosoma cruzi)
Universidade Federal Do Rio Grande Do Sul

Curated by ChEMBL
LigandPNGBDBM50322742(CHEMBL1173694 | N-(2-(1H-benzo[d]imidazol-2-yl)eth...)
Affinity DataIC50:  800nMAssay Description:Inhibition of Trypanosoma cruzi CruzainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedMMDB
PDB3D3D Structure (crystal)