Report error Found 34 Enz. Inhib. hit(s) with all data for entry = 50003653
Affinity DataKi: 0.0631nMAssay Description:Binding affinity against 5-hydroxytryptamine 1A human cloned receptors in HEK293 cells using [3H]8-OH-DPAT as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 0.398nMAssay Description:Binding affinity against 5-hydroxytryptamine 7 human receptorsMore data for this Ligand-Target Pair
Affinity DataKi: 0.631nMAssay Description:Binding affinity against 5-hydroxytryptamine 1A human cloned receptors in HEK293 cells using [3H]8-OH-DPAT as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 1.30nMAssay Description:Binding affinity against 5-hydroxytryptamine 1A human cloned receptors in HEK293 cells using [3H]8-OH-DPAT as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 1.30nMAssay Description:Binding affinity against human 5-hydroxytryptamine 1B receptor cloned receptors in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Binding affinity against 5-hydroxytryptamine 1A human cloned receptors in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 3.20nMAssay Description:Binding affinity against cloned human 5-hydroxytryptamine 1B receptor in CHO cells using [3H]5-CT as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 3.20nMAssay Description:Binding affinity against 5-hydroxytryptamine 7 human receptorsMore data for this Ligand-Target Pair
Affinity DataKi: 3.20nMAssay Description:Binding affinity against 5-hydroxytryptamine 2A receptor human cloned receptors in HEK 293 cells using [3H]ketanserin as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 3.20nMAssay Description:Binding affinity against 5-hydroxytryptamine 7 human receptorsMore data for this Ligand-Target Pair
Affinity DataKi: 3.20nMAssay Description:Binding affinity against human Dopamine receptor D2 in CHO cells using [125I]iodosulpirideMore data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:Binding affinity against 5-hydroxytryptamine 1A human cloned receptors in HEK293 cells using [3H]8-OH-DPAT as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 5nMAssay Description:Binding affinity against 5-hydroxytryptamine 2C receptor human cloned receptors in HEK 293 cells using [3H]mesulergine as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 5nMAssay Description:Binding affinity against cloned human 5-hydroxytryptamine 1B receptor in CHO cells using [3H]5-CT as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 6.30nMAssay Description:Binding affinity against 5-hydroxytryptamine 7 human receptorsMore data for this Ligand-Target Pair
Affinity DataKi: 6.30nMAssay Description:Binding affinity against 5-hydroxytryptamine 7 human receptorsMore data for this Ligand-Target Pair
Affinity DataKi: 6.30nMAssay Description:Binding affinity against 5-hydroxytryptamine 6 human cloned receptors in HeLa cellsMore data for this Ligand-Target Pair
Affinity DataKi: 16nMAssay Description:Binding affinity against 5-hydroxytryptamine 2A receptor human cloned receptorswithouteffect in HEK 293 cells using [3H]ketanserin as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 16nMAssay Description:Binding affinity against 5-hydroxytryptamine 2C receptor human cloned receptorswithouteffect in HEK 293 cells using [3H]mesulergine as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 50nMAssay Description:Binding affinity against 5-hydroxytryptamine 6 human cloned receptors in HeLa cells using [3H]LSD as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 50nMAssay Description:Binding affinity against 5-hydroxytryptamine 2C receptor human cloned receptors in HEK 293 cells using [3H]mesulergine as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 126nMAssay Description:Binding affinity against 5-hydroxytryptamine 6 human cloned receptors in HeLa cells using [3H]LSD as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 126nMAssay Description:Binding affinity against human Dopamine receptor D2 in CHO cells using [125I]iodosulpirideMore data for this Ligand-Target Pair
Affinity DataKi: 126nMAssay Description:Binding affinity against 5-hydroxytryptamine 6 human cloned receptors in HeLa cells using [3H]LSD as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 316nMAssay Description:Binding affinity against human 5-hydroxytryptamine 1B receptor cloned receptors in CHO cells using [3H]5-CT as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 398nMAssay Description:Binding affinity against 5-hydroxytryptamine 2A receptor human cloned receptors in HEK 293 cells using [3H]ketanserin as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 1.00E+3nMAssay Description:Binding affinity against 5-hydroxytryptamine 6 human cloned receptors in HeLa cells using [3H]LSD as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 2.51E+3nMAssay Description:Binding affinity against 5-hydroxytryptamine 2C receptor human cloned receptors in HEK 293 cells using [3H]mesulergine as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: <5.01E+3nMAssay Description:Binding affinity against 5-hydroxytryptamine 2A receptor human cloned receptors in HEK 293 cells using [3H]ketanserin as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 1.00E+4nMAssay Description:Binding affinity against 5-hydroxytryptamine 2A receptor human cloned receptors in HEK 293 cells using [3H]ketanserin as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 1.26E+4nMAssay Description:Binding affinity against 5-hydroxytryptamine 2C receptor human cloned receptors in HEK 293 cells using [3H]mesulergine as radioligandMore data for this Ligand-Target Pair
Affinity DataEC50: 19nMAssay Description:Binding affinity against human 5-hydroxytryptamine 1A receptors HEK 293 cell membranes using [35S]GTP gamma-SMore data for this Ligand-Target Pair
Affinity DataEC50: 2nMAssay Description:Binding affinity against human 5-hydroxytryptamine 1A receptors HEK 293 cell membranes using [35S]GTP gamma-SMore data for this Ligand-Target Pair
Affinity DataEC50: 8.70nMAssay Description:Binding affinity against human 5-hydroxytryptamine 1A receptors HEK 293 cell membranes using [35S]GTP gamma-SMore data for this Ligand-Target Pair