Affinity DataKi: 0.0290nMAssay Description:Binding affinity against Rat 5-hydroxytryptamine 7 receptor using [3H]-5-HTMore data for this Ligand-Target Pair
Affinity DataKi: 0.120nMAssay Description:Binding affinity at rat 5-hydroxytryptamine 7 receptor.More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Roche Bioscience
Curated by PDSP Ki Database
Roche Bioscience
Curated by PDSP Ki Database
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Roche Bioscience
Curated by PDSP Ki Database
Roche Bioscience
Curated by PDSP Ki Database
Affinity DataKi: 0.300nMAssay Description:Displacement of [3H]-5-CT from human cloned 5HT7 receptorMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Roche Bioscience
Curated by PDSP Ki Database
Roche Bioscience
Curated by PDSP Ki Database
Affinity DataKi: 0.350nMAssay Description:Displacement of [3H]-5-CT from human 5-HT7R expressed in human HEK293 cells assessed as inhibitory constant incubated for 60 mins by radioligand bind...More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Roche Bioscience
Curated by PDSP Ki Database
Roche Bioscience
Curated by PDSP Ki Database
Affinity DataKi: 0.398nMAssay Description:Binding affinity against 5-hydroxytryptamine 7 human receptorsMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Roche Bioscience
Curated by PDSP Ki Database
Roche Bioscience
Curated by PDSP Ki Database
Affinity DataKi: 0.490nMAssay Description:Binding affinity to human recombinant 5-hydroxytryptamine 7 receptor in mammalian cells using [3H]5-CT as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 0.5nM ΔG°: -55.2kJ/molepH: 7.4 T: 2°CAssay Description:IC50 values for each test compound were determined from nonlinear regression analysis of data collected from ligand binding experiments. The inhibiti...More data for this Ligand-Target Pair
Affinity DataKi: 0.5nMAssay Description:Displacement of [3H]LSD from rat cloned 5HT7 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.510nMAssay Description:Displacement of [3H]LSD from rat recombinant 5HT7 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.510nMAssay Description:Binding affinity to the rat 5-hydroxytryptamine 7 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.510nMAssay Description:Displacement of [3H]LSD from rat recombinant 5HT7 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Roche Bioscience
Curated by PDSP Ki Database
Roche Bioscience
Curated by PDSP Ki Database
Affinity DataKi: 0.900nMAssay Description:Displacement of [3H]5-HT from human 5-hydroxytryptamine 7 receptorMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Roche Bioscience
Curated by PDSP Ki Database
Roche Bioscience
Curated by PDSP Ki Database
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Roche Bioscience
Curated by PDSP Ki Database
Roche Bioscience
Curated by PDSP Ki Database
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Roche Bioscience
Curated by PDSP Ki Database
Roche Bioscience
Curated by PDSP Ki Database
Affinity DataKi: 0.930nMAssay Description:Binding affinity to 5-HT7 receptor (unknown origin)More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Roche Bioscience
Curated by PDSP Ki Database
Roche Bioscience
Curated by PDSP Ki Database
Target5-hydroxytryptamine receptor 7(Mus musculus (Mouse))
University of Alberta
Curated by PDSP Ki Database
University of Alberta
Curated by PDSP Ki Database
Target5-hydroxytryptamine receptor 7(Mus musculus (Mouse))
University of Alberta
Curated by PDSP Ki Database
University of Alberta
Curated by PDSP Ki Database
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Roche Bioscience
Curated by PDSP Ki Database
Roche Bioscience
Curated by PDSP Ki Database
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Roche Bioscience
Curated by PDSP Ki Database
Roche Bioscience
Curated by PDSP Ki Database
Affinity DataKi: <10nMAssay Description:Binding affinity of compound towards rodent 5-hydroxytryptamine 7 receptorMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Roche Bioscience
Curated by PDSP Ki Database
Roche Bioscience
Curated by PDSP Ki Database
Affinity DataEC50: 630nMAssay Description:Activity at 5HT7 receptor assessed as relaxation of substance P-induced contraction of Dunkin-Hartley guinea pig ileumMore data for this Ligand-Target Pair
Affinity DataEC50: 630nMAssay Description:Agonist activity at 5HT7 receptor assessed as relaxation of substance P-induced Dunkin-Hartley guinea pig ileum contractionMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Roche Bioscience
Curated by PDSP Ki Database
Roche Bioscience
Curated by PDSP Ki Database
Affinity DataEC50: 5.10nMAssay Description:Agonist activity at human 5HT7 receptor expressed in CHO-K1 cells by calcium 4 dye based FLIPR assayMore data for this Ligand-Target Pair